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(3S,4S)-4-[(2-hydroxyethyl)(methyl)amino]-1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]pyrrolidin-3-ol
5-[(2E)-3-phenylprop-2-en-1-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
3-(piperidine-1-sulfonyl)-N-[3-(1H-1,2,4-triazol-1-yl)propyl]benzamide
(3S,4S)-1-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
1-{[(1R,9aR)-1-hydroxy-octahydro-1H-quinolizin-1-yl]methyl}-1H-indole-4-carbonitrile
methyl({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)(thiophen-2-ylmethyl)amine
N-[1-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
3-(1,1-dioxo-1λ6-thiomorpholin-4-yl)-N-[(1S,2R)-2-[(propan-2-yl)amino]cyclobutyl]benzamide
N-{[2-(cyclohex-1-en-1-ylmethyl)-6-oxo-1,6-dihydropyrimidin-4-yl]methyl}-2-(methylsulfanyl)pyridine-3-carboxamide
methyl 3-acetamido-1-[2-(1H-indol-3-yl)ethyl]-5-[(2-methylbutyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(2-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)-2-(pyridin-2-yl)pyrimidine-5-carboxamide
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
5-(azepan-1-yl)-1-methyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
(2R,3R)-1'-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(pyrrolidin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-[(2-fluorophenyl)methyl]-1-methyl-5-[methyl(1,2-oxazol-3-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-1,4-oxazepan-6-ol
5-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-N-methyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3-carboxamide
4-[6-(piperidin-1-yl)pyrimidin-4-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
2-butyl-N-(2,6-diethylphenyl)-4-methyl-3-oxopiperazine-1-carboxamide
3-{2-[3-(3-fluorophenoxymethyl)piperidin-1-yl]-2-oxoethyl}-3-(2-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
2-cyclopentyl-4-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
(1R,5R)-N-(3-cyanophenyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
7-[(3,4-difluorophenyl)methyl]-2-(1,3-thiazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,3λ6,4-oxathiazinane-3,3-dione
N-[3-methyl-1-(4-methylphenyl)-1H-pyrazol-5-yl]thiomorpholine-4-carboxamide
methyl 3-methoxy-5-[2-(3-methoxypropyl)piperidine-1-carbonyl]benzoate
N-[2-(dimethylamino)ethyl]-3-{1-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}propanamide
4-{1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}pyridine
N-[(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-fluorobenzamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
1,3-dimethyl-5-{2-oxo-2-[4-(2-phenoxyethyl)piperazin-1-yl]ethyl}imidazolidine-2,4-dione
4-{[2-(benzylsulfanyl)pyrimidin-5-yl]methyl}morpholine-2-carboxamide
1-[(4aR,8aR)-7-[5-fluoro-2-(hydroxymethyl)pyridin-4-yl]-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]ethan-1-one
9-[3-(2-fluorophenyl)propanoyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[5-fluoro-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methoxybenzamide
1-{[1-(2H-1,3-benzodioxol-5-yl)-3-phenyl-1H-1,2,4-triazol-5-yl]methyl}-1H-1,2,3,4-tetrazol-5-amine
1-(2-{methyl[(4-phenylphenyl)methyl]amino}ethyl)-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
3-(3-chlorobenzoyl)-1-(thiophene-3-sulfonyl)piperidine
N-methyl-N-[(3-methylpyridin-2-yl)methyl]-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
3-(3-methoxyphenyl)-1-(pyridin-2-ylmethyl)-6-(thiolan-3-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
4-[2-(dimethylamino)ethyl]-N-[4-(4-fluorophenoxy)phenyl]piperazine-1-carboxamide
9-[2-(benzyloxy)ethyl]-2-cyclopentyl-2,9-diazaspiro[5.5]undecan-3-one
5-{[(8-fluoroquinolin-2-yl)formamido]methyl}thiophene-2-carboxylic acid
N-benzyl-N-ethyl-2-[1-(2-methoxyethyl)-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]acetamide
6-[1-(2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}acetyl)piperidin-4-yl]-2-methyl-3,4-dihydropyrimidin-4-one
4-(4-methoxyphenoxy)-N-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]benzamide
2-(1-methylpyrrolidin-3-yl)-9-(5-propyl-1,3,4-thiadiazol-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 9-(cyclopentyloxy)-3-[(2-fluoro-5-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate