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5-{1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
6-(4-methoxyphenyl)-N,N-dimethyl-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[(3-ethoxy-4-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-{7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(pyrazin-2-yl)propan-1-one
N-{[5-fluoro-7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(morpholin-4-yl)propanamide
(4aR,7aS)-1-[2-(dimethylamino)acetyl]-4-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
3-{[4-(3-hydroxypyrrolidin-1-yl)pyrimidin-2-yl]amino}-1-[4-(propan-2-yl)piperazin-1-yl]propan-1-one
6-[1-butyl-3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
N-{[4-fluoro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
N-(1-methyl-1H-pyrazol-5-yl)-3-({methyl[1-(pyridin-2-yl)propan-2-yl]amino}methyl)benzamide
1-(4-fluorophenyl)-N-methyl-N-[1-(1,3-thiazol-5-yl)ethyl]cyclopropane-1-carboxamide
(2S,4R)-N-(1-benzothiophen-2-ylmethyl)-1-[(2-fluorophenyl)methyl]-N-methyl-4-[(4-methylpyrimidin-2-yl)sulfanyl]pyrrolidine-2-carboxamide
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-{imidazo[1,2-a]pyridine-2-carbonyl}piperidine
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(propan-2-ylsulfanyl)ethan-1-one
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
N-(adamantan-1-ylmethyl)-1-[(2,6-difluorophenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
7-{[bis(2-methoxyethyl)amino]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-6-(4-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)-2-[(prop-2-en-1-yl)amino]benzamide
8-(1,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N3-ethyl-N5-[1-(4-fluorophenyl)ethyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2,3-dimethyl-7-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
2,5-dimethyl-N-({5-methyl-2-[3-(propane-2-sulfonamido)phenyl]-1,3-oxazol-4-yl}methyl)benzamide
(2E)-N-({3-methyl-7-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-phenylprop-2-enamide
1-(2-fluorophenyl)-4-[(2S,4R)-4-[(4-methoxyphenyl)sulfanyl]-1-(1-methylpiperidin-4-yl)pyrrolidine-2-carbonyl]piperazine
N,N-dimethyl-6-(2-methylphenyl)-3-(4-methylpiperidine-1-carbonyl)pyridin-2-amine
N-({1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]pyrrolidin-3-yl}methyl)acetamide
N-(1-{imidazo[1,2-a]pyridine-6-carbonyl}piperidin-4-yl)pyrimidin-2-amine
N-(cyclopropylmethyl)-N-propyl-2-(pyridine-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
3-ethyl-1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-ol
2-[({[(2R,3R,5S)-2-(4-chlorophenyl)-1-ethyl-5-(hydroxymethyl)-5-methylpyrrolidin-3-yl]methyl}amino)methyl]phenol
N-({3,5-dimethoxy-4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-4-(3-fluorophenyl)-N-(pyridin-4-ylmethyl)benzamide
4-{[2-(methylsulfanyl)phenyl]methyl}-1-phenylpiperazin-2-one
2-(4-fluorophenyl)-1-[9-(oxan-2-ylmethoxy)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
(4aR,8aS)-1-[(3-fluorophenyl)methyl]-6-[4-(4-methylphenyl)benzoyl]-decahydro-1,6-naphthyridin-2-one
2-[4-(1-cyano-1-methylethyl)phenyl]-2-[4-(pyridin-2-yl)piperazin-1-yl]acetic acid
[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)methylamine
[(3-cyclohexyl-1H-pyrazol-4-yl)methyl][(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)amine
5-oxo-1-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}pyrrolidine-3-carboxylic acid
1-[(4-chlorophenyl)methyl]-4-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazole
(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-2-(pyrazin-2-yl)-decahydroisoquinoline
1-{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-2-(methoxymethyl)piperidine
4-[1-(2,3-dihydro-1-benzofuran-2-carbonyl)piperidin-3-yl]-2-methyl-5-(3-methylphenyl)pyrimidine
1-ethyl-3-(2-methylpropyl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-pyrazole-5-carboxamide
7-oxo-2-(2-phenylacetamido)-N-[1-(1,3-thiazol-2-yl)ethyl]-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
3-[2-(1,3-benzothiazol-2-yl)pyrrolidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
1-(dimethylamino)-2-{4-[4-(furan-2-yl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}propan-2-ol
2-{2-oxo-2-[4-(1,3-thiazol-2-yl)piperazin-1-yl]ethyl}-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one