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N-{[1-(2-methyl-1-benzofuran-5-carbonyl)piperidin-3-yl]methyl}-1H-indole-2-carboxamide
8-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-ethyl-5-(1-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-4-phenyl-1H-imidazol-5-yl)-1H-1,2,4-triazole
(3S,4S)-4-(dimethylamino)-1-({3-[(3-fluorophenyl)methoxy]-4-methoxyphenyl}methyl)pyrrolidin-3-ol
N-[(4-hydroxyphenyl)methyl]-4-(1H-pyrazol-3-yl)benzamide
methyl 6-(4-fluorobenzoyl)-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-butyl-1-methyl-4-[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]piperazin-2-one
2-(morpholin-4-yl)-N-(1,2-oxazol-3-ylmethyl)pyrimidine-5-carboxamide
1-[(4-chlorophenyl)methyl]-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-oxopiperidine-3-carboxamide
N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-4-(piperidin-1-yl)butanamide
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]cyclohex-3-ene-1-carboxamide
2-(4-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
4-[(2-chloro-4-fluorophenyl)methyl]-3-[2-(4-cyclopentyl-1,4-diazepan-1-yl)-2-oxoethyl]piperazin-2-one
N'1-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]cyclopropane-1,1-dicarboxamide
1-cycloheptyl-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-6-oxopiperidine-3-carboxamide
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-(1,3-thiazol-2-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
N-benzyl-N-butyl-3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
6,6-dimethyl-1-(4-methylphenyl)-N-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-4-(3-methoxybenzoyl)piperazine
5-{2-[1-(3,4-dimethylphenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]ethyl}imidazolidine-2,4-dione
15-methyl-12-[4-(propan-2-yl)piperazine-1-carbonyl]-9-(thiophen-2-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaen-13-one
6-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}pyridine-2-carbonitrile
methyl 7-oxo-3-[(4-phenylphenyl)methyl]-9-(pyridin-4-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[(2R,3R)-2-ethoxy-1'-[(3-fluorophenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
5-ethyl-N4-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidine-2,4-diamine
5-methyl-5-(4-methylpent-3-en-1-yl)-1-[1-(pyrazin-2-yl)piperidin-4-yl]piperidin-2-one
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-{2-[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-oxoethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
2-(1-ethyl-1H-pyrazol-4-yl)-N-[1-(pyridin-4-yl)propyl]quinoline-4-carboxamide
5-(3,5-dimethyl-4-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-1H-pyrazol-1-yl)-1H-1,2,3,4-tetrazole
methyl 3-acetamido-1-ethyl-5-[(3-methylbutyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
[(3S,5R)-5-[(dimethylamino)methyl]-1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl]methanol
2-[(2,3-dimethoxyphenyl)methyl]-4-{4-[2-(2-methoxyphenyl)acetyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
5-(2-fluorophenyl)-N-[2-(1H-imidazol-1-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-[1-(ethanesulfonyl)azepan-3-yl]-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetamide
2-(2H-indazol-2-yl)-1-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]ethan-1-one
4-{[5-(2-chlorophenyl)furan-2-yl]methyl}-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(1-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-2-yl)propan-1-ol
3-fluoro-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylbenzamide
2-{[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}pyridine
4-benzyl-3-[1-(5-methyl-1,3,4-oxadiazole-2-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-[2-(ethylamino)ethyl]-1-[(2-fluorophenyl)methyl]pyrrolidin-2-one
2-(furan-2-yl)-5-{1-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-imidazol-2-yl}pyrimidine
4-chloro-2-{[7-(2,3-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenol
N-[(1-ethyl-5-oxopyrrolidin-3-yl)methyl]-4-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
3-{[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]sulfamoyl}-N-(oxolan-3-yl)benzamide
6-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]pyridine-2-carbonitrile
N-cyclopropyl-1-[1-(6-methylpyridine-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
N-[2-(4-hydroxyphenyl)ethyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
N-methyl-N-(1-methylpiperidin-4-yl)-3-(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)propanamide