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(3S,4R)-1-[2-(methylsulfanyl)acetyl]-4-phenylpyrrolidine-3-carboxylic acid
3-[1-(1-cyclobutanecarbonylpiperidine-4-carbonyl)pyrrolidin-2-yl]pyridine
(3R,4S)-4-(4-methoxyphenyl)-1-(morpholine-4-sulfonyl)pyrrolidin-3-amine
(2S)-2-({1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-7-oxoazepan-4-yl}amino)-4-methylpentanamide
[1-(1-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)ethyl]dimethylamine
(3R,5S)-N-[2-(morpholin-4-yl)ethyl]-5-(morpholin-4-ylmethyl)-1-(naphthalen-2-ylmethyl)piperidine-3-carboxamide
1-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-5-methyl-5-(4-methylpent-3-en-1-yl)piperidin-2-one
(3R,9R)-11-(naphthalene-2-carbonyl)-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
6-(difluoromethyl)-2-(4-{[methyl(1,2,3,4-tetrahydronaphthalen-1-yl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N-[(3R,4S)-1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]butane-1-sulfonamide
N-[(2-methylpyridin-4-yl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(piperidin-4-ylmethyl)acetamide
N-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-2-{4-[(E)-2-phenylethenyl]-1H-pyrazol-1-yl}acetamide
4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]piperidine
(3R,4R)-4-ethyl-1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidine-3,4-diol
4-[(5-ethylpyridin-2-yl)methyl]-9-(2-methoxyethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1'-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidine-1-carbonyl]benzonitrile
2-(3-methoxypropyl)-4-(4-{[4-(propan-2-yl)phenyl]methyl}piperazin-1-yl)-2,3-dihydro-1H-isoindole-1,3-dione
3-methyl-8-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(azepane-1-sulfonyl)-5-(1H-1,2,3-triazol-1-yl)benzoic acid
N-{[7-chloro-2-(4-methoxyphenyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)furan-3-carboxamide
5-{[3-(2-methoxybenzoyl)piperidin-1-yl]methyl}quinoxaline
N,5-dimethyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
2-{[4-(pyridin-3-yl)-5-[(trimethyl-1H-pyrazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
1-{1-[4-methyl-6-(propan-2-yl)quinazolin-2-yl]piperidine-4-carbonyl}-4-(pyridin-3-yl)piperidin-4-ol
[(3,5-dimethoxyphenyl)methyl](2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)amine
5-[2-(3,4-difluorophenyl)pyrimidin-4-yl]-2-ethoxybenzoic acid
3-[(3-hydroxypiperidin-1-yl)methyl]-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
6-methyl-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
(4aR,7aS)-1-[2-(1,4-diazepan-1-yl)pyrimidin-4-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S,4S)-1-[(2-chloro-5-ethoxy-4-methoxyphenyl)methyl]-4-(piperidin-1-yl)pyrrolidin-3-ol
(1s,4s)-4-[3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]cyclohexan-1-ol
N-(4-methoxyphenyl)-1-(2-methyl-1,3-benzothiazole-5-carbonyl)piperidin-3-amine
2-tert-butyl-4-hydroxy-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]pyrimidine-5-carboxamide
3-{2-[2-(1-ethylpiperidin-3-yl)-1H-imidazol-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(1H-imidazol-2-ylmethyl)({[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
N-[2-(4-methoxyphenyl)ethyl]-1-methyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(2,3-dihydro-1H-inden-2-yl)-2-methyl-N-propylimidazo[1,2-a]pyrimidine-3-carboxamide
N-[(3S,4R)-4-(propan-2-yl)-1-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetyl]pyrrolidin-3-yl]methanesulfonamide
2-methyl-5-(3-methylphenyl)-4-[1-(naphthalene-2-carbonyl)piperidin-3-yl]pyrimidine
4-{1-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-3-yl}-5-methyl-2-(pyridin-3-yl)pyrimidine
N-{[5-fluoro-7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methyl-4-oxo-3,4-dihydrophthalazine-1-carboxamide
1-[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
3-[1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]-1-(4-ethylpiperazin-1-yl)propan-1-one
2-methyl-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}thieno[2,3-d]pyrimidin-4-amine
N-[(3R,4S)-4-cyclopropyl-1-methanesulfonylpyrrolidin-3-yl]-5-fluoro-2-methoxybenzamide
({1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-1H-imidazol-5-yl}methyl)(prop-2-en-1-yl)(prop-2-yn-1-yl)amine
N-{[4-(oxolan-2-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)-2-(trifluoromethyl)benzamide
2-(2,4-difluorophenoxy)-N-[1-(thiophen-2-ylmethyl)piperidin-3-yl]acetamide