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1-cyclohexyl-4-[(4-methanesulfonylphenyl)methyl]-1,4-diazepane
(2E)-N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(2,5-difluorophenyl)prop-2-enamide
N-[2-(1H-imidazol-4-yl)ethyl]-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
2-{5-[1-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)piperidin-4-yl]-1H-pyrazol-3-yl}acetic acid
1-(pyridin-2-ylmethyl)-N-{thieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methylpiperidin-3-amine
N,8-dimethyl-N-(oxan-4-yl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
5-[(3-fluorophenyl)methyl]-5-{1-[(4-methoxyphenyl)methyl]piperidin-4-yl}-3-(2-methylpropyl)imidazolidine-2,4-dione
3-(furan-3-yl)-2,4,5-triazatetracyclo[11.4.0.02,6.07,12]heptadeca-1(17),3,5,7,9,11,13,15-octaene
4-[7-(1H-imidazole-2-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
5-cyclohexyl-2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
8-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{[4-(1H-imidazol-1-yl)phenyl]methyl}-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
N-[2-(3-phenylpiperidin-1-yl)ethyl]-4-(1H-pyrazol-3-yl)benzamide
N-[(1-hydroxycyclohexyl)methyl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
1-(oxolane-2-carbonyl)-4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1,4-diazepane
methyl 3-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propanoate
N-({5-[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-2-({6-methylthieno[2,3-d]pyrimidin-4-yl}sulfanyl)acetamide
1-cyclopentyl-3-{2-[4-(4-methyl-1,2,5-oxadiazol-3-yl)piperazin-1-yl]-2-oxoethyl}-3-(2-methylphenyl)pyrrolidine-2,5-dione
ethyl 7-(2-chlorobenzamido)-1,2,3,4-tetrahydroisoquinoline-2-carboxylate
1-(1-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)pyrrolidin-2-one
2-methyl-4-phenyl-9-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecane
2-[1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)pyrrolidin-2-yl]pyridine
(3aR,6aR)-2-methanesulfonyl-5-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(1,3-oxazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-[1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
2-methoxy-N-{1-[1-(2-oxopropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-phenylacetamide
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyridin-2-yl)ethyl]acetamide
2-{[8-(2-methylquinolin-4-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}phenol
4-[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]benzene-1-sulfonamide
3-[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-4-yl]-1-(4-phenylpiperazin-1-yl)propan-1-one
N-[2-hydroxy-2-(pyridin-2-yl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
methyl 2-[8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
5-{4-[(3-propyl-1,2,4-oxadiazol-5-yl)methoxy]phenyl}-1,3,4-oxadiazol-2-amine
4-(4-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)quinazoline
N-[(8-{[2-(furan-2-yl)phenyl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]-2-methylpropanamide
N-(2-methoxyphenyl)-6-{[4-(2-methylpropyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-3-[3-(1H-1,2,4-triazol-1-yl)phenyl]urea
N-[(3,4-difluorophenyl)methyl]-3-[1-(3-methylthiophene-2-carbonyl)piperidin-3-yl]propanamide
(1-{[1-(furan-3-ylmethyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)(phenyl)methanol
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-4-(1H-pyrazol-1-yl)-N-(pyridin-4-ylmethyl)benzamide
5-fluoro-2-(1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)-1H-1,3-benzodiazole
N-(4-{[(3R,4R)-4-(azepan-1-yl)-3-hydroxypiperidin-1-yl]methyl}phenyl)acetamide
1-{2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole-5-carbonyl}piperidin-4-ol
3-(3-hydroxyquinoxalin-2-yl)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-3-(4-phenylbenzoyl)piperidine
4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]-1-(1H-pyrazole-3-carbonyl)piperidine
2-chloro-N-(cyclopropylmethyl)-N-(propan-2-yl)-4-(4H-1,2,4-triazol-4-yl)benzamide