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6-methyl-3-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
(1R,2S)-N1-tert-butyl-N2-[(2,5-dimethoxyphenyl)methyl]cyclohexane-1,2-dicarboxamide
2-(methylsulfanyl)-1-{3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidin-1-yl}ethan-1-one
N-[2-(2,4-difluorophenyl)-1-{1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}ethyl]-N-methylpropanamide
N-[2-(dimethylamino)ethyl]-3-[(furan-3-ylmethyl)amino]-5-[(4-methoxyphenyl)sulfamoyl]benzamide
N-({1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-3-yl}methyl)-3-(trifluoromethyl)benzamide
(2S)-2-hydroxy-N-{2-[5-(hydroxymethyl)-1,2,4-oxadiazol-3-yl]ethyl}-3-phenylpropanamide
2-({[1-({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-3-yl]oxy}methyl)pyridine
N-[4-(4-{[1-(1H-1,3-benzodiazol-2-yl)ethyl]amino}piperidin-1-yl)phenyl]-4-methoxybenzamide
1-(pyrimidin-2-yl)-4-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-1,4-diazepane
2-{[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}-N-propylacetamide
13-(5-chloro-2,4-dimethoxyphenyl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
ethyl 2-(4-{2-[4-(3-phenoxypropanamido)-1H-pyrazol-1-yl]acetyl}morpholin-3-yl)acetate
1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-2-(1,3-thiazol-2-yl)piperidine
ethyl 3-[(1-methylazepan-2-yl)formamido]propanoate
2-[(isoquinolin-5-yloxy)methyl]-N-[2-(pyridin-2-yl)ethyl]-1,3-oxazole-4-carboxamide
1-(4-methoxyphenyl)-6,6-dimethyl-4-[(1R,2S)-2-propylcyclopropanecarbonyl]piperazin-2-one
3,5-dimethyl-2-[4-(pyridin-4-yl)piperazine-1-carbonyl]-1H-indole
N-[2-(4-chlorophenyl)ethyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-methyl-2-(methylsulfanyl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}pyridine-3-carboxamide
4-{[(dimethyl-1,3-thiazol-5-yl)methyl]amino}pyrimidine-5-carboxylic acid
N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-1-(pyrimidin-2-yl)piperidin-4-amine
(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-4-yl)(pyridin-2-yl)methanol
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}[(3-fluorophenyl)methyl]methylamine
8-(4-hydroxy-4-methylpentan-2-yl)-1-methyl-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[1-(2,5-dimethoxybenzoyl)piperidin-3-yl]-N-[(5-methylfuran-2-yl)methyl]propanamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxy-N-methyl-N-(pyridin-2-ylmethyl)benzamide
2-{1-benzyl-4-[6-methyl-2-(methylamino)pyrimidin-4-yl]piperazin-2-yl}ethan-1-ol
4-(5-{[(3-hydroxypropyl)amino]methyl}-1,2,4-oxadiazol-3-yl)benzoic acid
2-{4-[(2,4-dimethoxy-3-methylphenyl)methyl]-1-[(2-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-methyl-4-({5-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl}methyl)piperidine
(2E)-3-(2-chlorophenyl)-N-{[8-(4-fluorobenzoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}prop-2-enamide
2-[2-(4-chloro-1H-pyrazol-1-yl)acetamido]-N-[(3-methylphenyl)methyl]benzamide
6-[3-(2-ethoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-9H-purine
1-cycloheptyl-5-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
2-{4-[2-(2,3-dimethylphenoxy)ethyl]piperazin-1-yl}-4,6-dimethylpyrimidine
3-[(4-fluorophenyl)methyl]-N-{[1-(propan-2-yl)piperidin-4-yl]methyl}-1,2-oxazole-5-carboxamide
1-[2-(1-benzothiophen-2-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-(furan-2-ylmethyl)-N-methylpiperidine-4-carboxamide
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
5-cyclopropyl-N-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-1,3-oxazole-4-carboxamide
1-(2-{[3-(4-hydroxyphenyl)phenyl]formamido}ethyl)piperidine-3-carboxamide
4-cyclopentyl-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]pyrimidin-2-amine
1-(2-cycloheptyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)-N-methyl-N-(propan-2-yl)piperidine-4-carboxamide
N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1,2,3,4-tetrahydronaphthalene-2-carboxamide
5-(3-benzyl-1,2,4-oxadiazol-5-yl)-N-[(5-methyl-1,2-oxazol-3-yl)methyl]pyridin-2-amine
(3R,5R)-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
methyl 4-(5-{[benzyl(butyl)amino]methyl}-1,2,4-oxadiazol-3-yl)benzoate
5-(2,4-difluorophenoxymethyl)-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1,2-oxazole-3-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopropyl-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide