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N-[(8-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]oxolane-2-carboxamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-2-phenyl-N-(pyridin-3-ylmethyl)acetamide
4-{7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}pyridin-1-ium-1-olate
N-[(2-fluorophenyl)methyl]-5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
5-methyl-1-propyl-N-(thiophen-3-ylmethyl)-1H-pyrazole-4-carboxamide
N-{2-[3-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]propyl}-2-(trifluoromethyl)benzamide
N-(furan-2-ylmethyl)-1-(pyrimidin-2-yl)piperidin-3-amine
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
2,2-dimethyl-N-{2-methyl-4-[2-(1H-1,2,4-triazol-1-yl)propanamido]phenyl}propanamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-ethyl-5-[1-(2-phenoxypropanoyl)piperidin-4-yl]imidazolidine-2,4-dione
2-{5-[1-(1H-imidazol-1-ylmethyl)cyclopropyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}-6-methylpyridine
2-amino-3-cyano-4-(1H-imidazol-4-yl)-5H,6H-furo[2,3-h]quinoline-9-carboxylic acid
3-chloro-N-cyclopentyl-4-({1-[3-(furan-2-yl)propanoyl]piperidin-4-yl}oxy)benzamide
2-methyl-6-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
1-{[1-(benzenesulfonyl)-1H-pyrrol-2-yl]methyl}-3-(1H-imidazol-1-ylmethyl)piperidine
4-[3-(cyclopentylcarbamoyl)-1-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyridin-1-ium-1-olate
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(5-methyl-1H-indazole-3-carbonyl)pyrrolidin-3-yl]methanol
N,1-dimethyl-N-[2-phenyl-1-(1-{[4-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)ethyl]-1H-pyrazole-3-carboxamide
({1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-1H-imidazol-5-yl}methyl)(methyl)(1,3-thiazol-2-ylmethyl)amine
N-cyclopentyl-4-oxo-4-(3-oxo-4-phenylpiperazin-1-yl)butanamide
3-cyclopropyl-N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1H-pyrazole-5-carboxamide
5-[2-(2-aminoethyl)morpholin-4-yl]-2-[2-(2,4-dimethylphenoxy)ethyl]-2,3-dihydropyridazin-3-one
N,1-dimethyl-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[2-(dimethylamino)ethyl]-5-[1-(4-methyl-2-oxopentanoyl)piperidin-4-yl]-5-(3-methylbutyl)imidazolidine-2,4-dione
2-ethyl-5-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyrimidine
2-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-(2-methoxyethyl)-N-(propan-2-yl)benzamide
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-2-oxo-2-phenylacetamide
2-[1-cyclopentyl-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-(cyclopropylmethyl)-N-propylacetamide
N-(3,4-dimethylphenyl)-1-(3,4,5-trimethoxybenzoyl)piperidin-3-amine
butyl 2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidine-1-carboxylate
2-(4-chloro-3-fluorophenyl)-2-[(2-methoxyethyl)(methyl)amino]acetic acid
ethyl 5-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[(4-{[(2S,5R)-5-(1,4-oxazepan-4-ylmethyl)oxolan-2-yl]methyl}phenyl)methyl]cyclopropanamine
N-({8-[(2-fluorophenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-phenoxypropanamide
[1-(6-chloro-2-methylquinoline-4-carbonyl)piperidin-2-yl]methanamine
4-[1-(1-methylcyclopropanecarbonyl)piperidin-4-yl]-5-phenyl-2-(pyridin-3-yl)pyrimidine
2-(dimethyl-1,2-oxazol-4-yl)-1-[1-(2-methylpropyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
2-(2,3-difluorophenoxymethyl)-N-(3-hydroxypropyl)-N-methyl-1,3-oxazole-4-carboxamide
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(2,5-difluorophenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(2S,4R)-N-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-1-[(3-methoxyphenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
6-[(2-methoxyphenyl)methyl]-N-(3-phenylpropyl)-6-azaspiro[2.5]octane-1-carboxamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylpent-4-enamide
(1R,6S)-9-methyl-3-(4-methyl-2-phenylpyrimidine-5-carbonyl)-3,9-diazabicyclo[4.2.1]nonane
N,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)-N-(pyridin-3-ylmethyl)quinoline-4-carboxamide
1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-({3-methyl-7-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(methylsulfanyl)benzamide
1-[2-({[(5-chlorothiophen-2-yl)methyl]amino}methyl)-5-methoxyphenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
4-[3-(2-oxo-5,5-diphenylpiperidin-1-yl)propyl]piperazin-2-one
N-(2-ethyl-3-methyl-1-benzofuran-7-yl)-1,1-dioxo-1λ6-thiomorpholine-4-carboxamide
3-(but-2-yn-1-yl)-5-{1-[(2E)-4-methylpent-2-en-1-yl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione