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1-(azepan-1-yl)-3-(3-{[3-(morpholin-4-yl)azetidin-1-yl]methyl}phenoxy)propan-2-ol
1-[3-(4-fluorophenyl)benzoyl]-4-(hydroxymethyl)azepan-4-ol
{1-[(2-chloro-4,5-dimethoxyphenyl)methyl]-3-[(2-fluorophenyl)methyl]piperidin-3-yl}methanol
1-(3-chlorophenyl)-4-[2-(4-methoxyphenyl)acetyl]piperazin-2-one
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-5-methyl-1,2-oxazole-4-carboxamide
(3R,4R)-1-(2-benzyl-1,3-thiazole-4-carbonyl)-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-methylacetamide
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-4-(pyrrolidin-1-yl)benzamide
1-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)-3-(pyrrolidin-1-yl)propan-2-ol
1-benzyl-8-propyl-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-[(4-methoxyphenyl)methyl]piperidine
2-(piperidin-1-yl)-N-(pyrrolidin-3-yl)-2,3-dihydro-1H-indene-2-carboxamide
1-{2-[(4-fluorophenyl)methyl]morpholin-4-yl}-2-(1H-pyrazol-1-yl)ethan-1-one
3-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1H-pyrazol-5-amine
ethyl 3-benzyl-1-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}piperidine-3-carboxylate
N-[2-({3-azaspiro[5.5]undecan-9-yl}amino)ethyl]-2-chlorobenzamide
N,2,8-trimethyl-N-[2-(oxan-2-yl)ethyl]quinoline-4-carboxamide
2-(2-aminoethyl)-N-[6-(dimethylamino)-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl]morpholine-4-carboxamide
1-(3-cyanopyrazin-2-yl)-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
1-[(diethylcarbamoyl)methyl]-N-methyl-N-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
(1S,5R)-6-(cyclopropylmethyl)-3-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
2-{5-[1-(3-phenoxypropyl)pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
2-(methylamino)-N-(2-methylphenyl)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidine-6-carboxamide
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pentane-1,4-dione
2-{[(1R,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzoic acid
2-[4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl]ethan-1-ol
N-{[7-(4,6-dimethylpyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propanamide
4-benzyl-3-ethyl-1-(3-hydroxypyridine-2-carbonyl)-1,4-diazepan-5-one
N-[1-({[(4-phenyloxan-4-yl)methyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-2-(phenylsulfanyl)acetamide
3-({4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)benzonitrile
4-(2-methoxypyridine-4-carbonyl)-1,4-oxazepan-6-ol
6-(azepane-1-carbonyl)-N-[2-(4-methoxyphenyl)ethyl]-5-methylthieno[2,3-d]pyrimidin-4-amine
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(1H-indol-3-yl)propanamide
methyl 4-{4-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]piperazin-1-yl}benzoate
2-(4-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}morpholin-3-yl)acetic acid
methyl 4-{5-[1-(1-methyl-6-oxopiperidin-3-yl)-1H-imidazol-2-yl]furan-2-yl}benzoate
1-({3-[3-(azepan-1-yl)-2-hydroxypropoxy]phenyl}methyl)azetidin-3-ol
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
9-[2-(6-methoxy-2-oxo-2,3-dihydro-1H-indol-3-yl)acetyl]-6-(4-methoxyphenyl)-6,9-diazaspiro[4.5]decan-7-one
8-[(5-methylfuran-2-yl)methyl]-1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2-methoxyethyl)-N-[(4-methoxyphenyl)methyl]-3-(piperidin-3-yl)benzamide
6-(4-chlorophenyl)-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
(1r,4r)-4-methyl-N-{2-[4-(propan-2-yl)morpholin-2-yl]ethyl}cyclohexane-1-carboxamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-1-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)propan-1-one
3-(4-fluorophenyl)-N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)benzamide
1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(1,2-oxazolidin-2-yl)propan-1-one
2-phenyl-1-{1-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperidin-4-yl}ethan-1-ol
5-(4-cyclohexylpiperazine-1-carbonyl)-1,3-benzothiazol-2-amine
7-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-[2-(azepane-1-carbonyl)phenyl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide