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methyl 4-({4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)benzoate
{[6-(4-ethylpiperazin-1-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}[(2-fluorophenyl)methyl]amine
1-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
N-[1-methyl-4-(pyridin-3-yloxy)-1H-indazol-3-yl]oxane-4-carboxamide
N-{[7-(2-cyclohexylacetyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}oxolane-3-carboxamide
2-(dimethylamino)-2-(3-methylphenyl)-N-[2-(3-methylpyridin-2-yl)ethyl]acetamide
2-(dimethylamino)-N-[1-(hydroxymethyl)cyclohexyl]-2-(4-methylphenyl)acetamide
[5-({[3-(1H-imidazol-1-yl)propyl](pyridin-4-ylmethyl)amino}methyl)furan-2-yl]methanol
ethyl 1-{2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]acetyl}-4-(3-phenylpropyl)piperidine-4-carboxylate
N-(3,4-difluorophenyl)-1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-3-amine
1-(3,4-difluorophenyl)-5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
2-methyl-6-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
3,5-dimethyl-N-{[5-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1,2-oxazole-4-carboxamide
1-(1-benzoxepine-4-carbonyl)-4-[(3-fluorophenyl)methyl]piperazine
1-{2,7-diazaspiro[4.5]decan-7-yl}-4-phenylbutane-1,4-dione
N-[2-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]cyclohexanecarboxamide
3-(2,3-dihydro-1H-inden-2-yl)-5-[1-(1H-indol-2-ylmethyl)piperidin-4-yl]-5-methylimidazolidine-2,4-dione
8-[(2,6-dimethoxyphenyl)methyl]-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)acetamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(2-methoxyethyl)pyrrolidin-3-yl]-1H-indole-2-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[3-(1H-1,2,4-triazol-1-yl)propyl]piperidin-2-one
N-[1-(furan-2-carbonyl)piperidin-4-yl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
N-[2-(4-methoxyphenyl)phenyl]-1-(pyridin-4-yl)piperidine-3-carboxamide
2-ethyl-8-[2-(2-hydroxyphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[(3-phenyl-1H-pyrazol-4-yl)methyl]amine
5-cyclopropanecarbonyl-1'-(3-fluorobenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(oxan-4-ylmethyl)-6-(pyridin-4-ylmethoxy)-4-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]-1,4-diazepan-2-one
N-{2-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}oxolane-2-carboxamide
2-(2,4-difluorophenoxy)-N-[1-(3-methoxyphenyl)-5-oxopyrrolidin-3-yl]acetamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-2-methoxypyridine-4-carboxamide
1-{3-[4-(1-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]piperidin-1-yl}ethan-1-one
4-[1-(3-methoxyphenyl)piperidin-4-yl]-2-(trifluoromethyl)morpholine
4-[1-(3,5-dimethylbenzoyl)pyrrolidin-3-yl]-2-(pyridin-3-yl)pyridine
methyl 2-(2-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)propanamido]methyl}-5-methyl-2,3-dihydro-1-benzofuran-7-yl)benzoate
2,6-dimethyl-4-(thiomorpholine-4-carbonyl)quinoline
N-[2-hydroxy-1-(pyridin-3-yl)ethyl]-5-(1H-indol-1-ylmethyl)-1H-pyrazole-3-carboxamide
N-{5H,6H,7H-cyclopenta[b]pyridin-3-ylmethyl}-2-(dimethylamino)-2-(3-fluorophenyl)acetamide
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[(3,5-dimethylphenyl)methyl]-1-[(4-hydroxyphenyl)methyl]piperidine-3,5-dicarboxamide
2,4-dimethyl-N-{[5-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1,3-thiazole-5-carboxamide
{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}({2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl})amine
5-[(4-methyl-3-phenylpiperazin-1-yl)methyl]-N-propylpyrimidin-2-amine
N-[(2R,3R)-2-hydroxy-1'-(quinolin-6-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
(1R,2R)-2-[ethyl({[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl})amino]cyclohexan-1-ol
1-{2-[3-(2-methoxybenzoyl)piperidine-1-carbonyl]phenyl}ethan-1-one
(1S,5R)-6-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-(dimethylamino)-1-{4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-N-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-{1-[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]azetidin-3-yl}morpholine
1-(2-{1-[2-(dimethylamino)-2-(3-methylphenyl)acetyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
methyl 4-(4-{2,5-dioxo-4-propyl-1-[2-(thiophen-2-yl)ethyl]imidazolidin-4-yl}piperidine-1-carbonyl)benzoate