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2-(dimethylamino)-N-(1-{7-[3-(2-methoxyphenyl)propanoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)acetamide
2-{2-[1-(2,4-difluorophenyl)-1H-1,2,4-triazol-5-yl]ethyl}-1-methylpiperidine
2,3-dimethyl-N-{[5-methyl-7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
(2S,4R)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]-N-(2-methyl-1,3-benzothiazol-5-yl)-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
(4aS,8aR)-1-(2-aminoethyl)-6-(3-methyl-1H-indole-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
5-acetamido-1-ethyl-2-(3-methoxyphenyl)-N-(oxolan-2-ylmethyl)-N-propyl-1H-1,3-benzodiazole-7-carboxamide
N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-1H-indole-5-carboxamide
{4-[4-(3-fluorophenyl)benzoyl]-1-methylpiperazin-2-yl}methanol
2-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]acetic acid
ethyl 2-{1-[4-(difluoromethoxy)benzoyl]piperidin-2-yl}acetate
2-hydroxy-N-methyl-4-(methylsulfanyl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}butanamide
N-{3-[(pyridin-3-yl)amino]propyl}pyridine-3-carboxamide
5-{3-[(2-fluorophenyl)formamido]propanoyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
2-ethyl-N,4-dimethyl-N-(quinolin-5-ylmethyl)-1,3-thiazole-5-carboxamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-1-cyclohexanecarbonylpyrrolidine-2-carboxamide
[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]({[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})amine
3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-1-[4-(pyrimidin-2-yl)piperazin-1-yl]propan-1-one
4-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-1,2-dihydroisoquinolin-1-one
2-[(4aR,7aS)-4-(2-cyclopentylacetyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
5-fluoro-N-[(3R,4R)-3-hydroxypiperidin-4-yl]-2-methylbenzamide
N-(3-methoxypropyl)-6-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
4-[5-(4-methoxyphenyl)furan-2-carbonyl]-1-(2-methylpropyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
(1R,2R,6S,7S)-4-[5-(oxolan-2-yl)thiophene-2-carbonyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
7-chloro-N-(2-methoxyethyl)-N-[(2-methoxyphenyl)methyl]-1-methyl-1H-indole-2-carboxamide
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(2-methyl-1,3-thiazol-4-yl)acetamide
4-(2-methoxyphenoxy)-1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}piperidine
4-(1-methyl-1H-imidazol-2-yl)-1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]piperidine
2-(morpholin-4-yl)-N-{[7-(pyrimidin-2-yl)-1H,2H-naphtho[2,1-b]furan-2-yl]methyl}propanamide
3,5-dimethyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-4,5-dihydro-1,2-oxazole-5-carboxamide
2-hydroxy-4-methoxy-N-[(2-phenoxypyridin-3-yl)methyl]benzamide
N-[(3R,4R)-1-(3-ethoxypropanoyl)-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
(2R,3R)-3-amino-1'-(3-methoxy-2-methylbenzoyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-[4-(2-methoxyphenyl)-1,3-dimethyl-1H-pyrazol-5-yl]-1-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]urea
1-{pyrazolo[1,5-a]pyridine-3-carbonyl}-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
(2R,6R)-10-methoxy-4-(pyridin-2-ylmethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-[(3S,4R)-4-(4-methylphenyl)-1-(1H-pyrrole-2-carbonyl)pyrrolidin-3-yl]cyclopropanecarboxamide
1-{2-[1-(3-fluoro-4-methylbenzenesulfonyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-1-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
2-{4-[5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]piperazin-1-yl}pyrimidine
N,N,4-trimethyl-5-[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyrimidin-2-amine
8-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-{5-[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinoline-1-carbonyl]-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl}butanamide
1-(cyclopropylmethyl)-3-(2,3-dimethoxyphenyl)-6-(2-phenoxypropanoyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
(1R,3S)-N1,N1,2,2,3-pentamethyl-N3-[3-(4-methyl-1,3-thiazol-2-yl)propyl]cyclopentane-1,3-dicarboxamide
methyl 2-{[5-(4-fluorophenyl)-4-{1-[(4R)-2-oxo-1,3-thiazolidine-4-carbonyl]piperidin-3-yl}pyrimidin-2-yl]sulfanyl}acetate
1-[2-(1H-imidazol-1-yl)propyl]-3-(trimethyl-1H-pyrazol-4-yl)urea
N-(2,4-dimethoxyphenyl)-3-{1-[(2S)-pyrrolidine-2-carbonyl]piperidin-4-yl}propanamide
3-(furan-2-yl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]benzamide
1-(2-methyl-6-propylpyrimidin-4-yl)-4-(pyridin-2-ylmethyl)-1,4-diazepane
N-({7-[2-(3,5-difluorophenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-methoxy-2-phenylacetamide