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2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]ethan-1-one
(3S,4S)-1-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-4-(piperidin-1-yl)pyrrolidin-3-ol
1-(furan-2-yl)-2-[4-(pyridin-4-yl)piperidin-1-yl]ethane-1,2-dione
1-(3-{[(3-methoxypropyl)(methyl)amino]methyl}-6-methylquinolin-2-yl)piperidin-3-ol
[(3R,4R)-1-[(1-ethyl-1H-indol-6-yl)methyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
methyl[1-(4-methyl-1,3-thiazol-2-yl)ethyl]{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
5-[1-(2,4-dimethylbenzoyl)piperidin-4-yl]-3-(oxolan-2-ylmethyl)-5-(pyridin-3-yl)imidazolidine-2,4-dione
2-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]acetamide
3-[2-(ethylsulfanyl)-1,3-benzoxazol-6-yl]-1-(2-methoxyethyl)-1-(pyridin-4-ylmethyl)urea
2-methyl-6-(1-methyl-1H-1,3-benzodiazol-2-yl)phenol
methyl 7-oxo-3-(pyridin-3-ylmethyl)-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(dimethylamino)-7-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(3-{[(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)amino]methyl}-2-methyl-1H-indol-1-yl)acetamide
9-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
methyl 3-[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl]-9-(cyclopentyloxy)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N4-(2H-1,3-benzodioxol-5-ylmethyl)-6-(propan-2-yloxy)pyrimidine-2,4-diamine
N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
2-[(1S,5R)-3-(3-methoxypyrazin-2-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
(3S,4S)-1-cyclohexanecarbonyl-4-cyclopropylpyrrolidine-3-carboxylic acid
2-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine
3-{[1-(1H-pyrazol-3-ylmethyl)piperidin-4-yl]oxy}-N-(pyridin-3-ylmethyl)benzamide
5-(2,3-dimethoxyphenyl)-4-phenyl-1H-imidazole
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl][2-(2-fluorophenyl)-1-[1-(1H-indole-2-carbonyl)piperidin-4-yl]ethyl]methylamine
3-[2-(2H-1,3-benzodioxol-5-ylmethyl)-5-oxopyrrolidin-2-yl]-N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)propanamide
N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-3-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamide
N-(5-methyl-1,2-oxazol-3-yl)-2-(4-methylpentanoyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-4-phenoxybutan-1-one
4-({5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,2,4-oxadiazol-3-yl}methyl)-1-methylpiperidine
7-(1,3-benzothiazol-2-yl)-4-(pyrimidine-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(cyclohexylmethyl)-2-[(1-methylpiperidin-4-yl)(pyridin-3-ylmethyl)amino]acetamide
N-{2-[(pyridin-2-ylmethyl)carbamoyl]phenyl}-1H-imidazole-2-carboxamide
(4S,4aS,8aS)-1-(4-methylpiperazine-1-carbonyl)-4-phenyl-decahydroquinolin-4-ol
3-(azocan-1-yl)-N-(furan-2-ylmethyl)-N-(pyridin-3-ylmethyl)propanamide
3-methyl-2-oxo-N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pentanamide
1-{1-[(2-aminopyrimidin-5-yl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
N-(2-methylbutyl)-2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
3-(1-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)propan-1-ol
5-({3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}methyl)-N-methylfuran-2-carboxamide
1-benzyl-4-[2-(3,4-dimethoxyphenyl)acetyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
5-chloro-6-[4-(2-methoxybenzoyl)piperazin-1-yl]pyridine-3-carboxylic acid
(2S)-N-{[7-(3,6-dimethylpyrazin-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-acetamido-4-methylpentanamide
2-(4,5-dichloro-1H-imidazol-1-yl)-N-[1-(pentan-2-yl)-1H-pyrazol-5-yl]acetamide
1-[2-(2-chlorophenyl)ethyl]-2-(methoxymethyl)-6-methyl-N-[1-(naphthalen-1-yl)ethyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
N-[(2R,3R)-2-methoxy-1'-[4-(2-methylpropyl)benzoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-2-carboxamide
7-methoxy-3-({[2-(2-methoxyphenyl)ethyl]amino}methyl)-1-(prop-2-yn-1-yl)-1,2-dihydroquinolin-2-one
7-[(3-acetyl-2,4,6-trimethylphenyl)methyl]-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
4-[2-(1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-4-oxo-N-[2-(propan-2-yl)phenyl]butanamide
N-(2-methoxyethyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methylpyridazine-4-carboxamide
1-(2-methoxy-5-{[3-(pyridin-3-yl)azetidin-1-yl]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol