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2-(methylsulfanyl)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyridine-3-carboxamide
1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-3-[(methylsulfanyl)methyl]piperidine
1-(carbamoylmethyl)-N-[2-(2-chlorophenoxy)ethyl]piperidine-3-carboxamide
ethyl 1-[2-(dimethylamino)-2-(2-methylphenyl)acetyl]-4-(2-methoxyethyl)piperidine-4-carboxylate
1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-2-(2-methoxyethyl)piperidine
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-4-(1H-1,2,4-triazol-3-yl)benzamide
(4aS,7aR)-1-[3-(1H-1,2,3-benzotriazol-1-yl)propanoyl]-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-4-carboxamide
2-{1-[5-(methoxymethyl)thiophene-2-carbonyl]piperidin-4-yl}-4-methyl-1H-1,3-benzodiazole
3-{1-[3-(2-oxoimidazolidin-1-yl)benzoyl]piperidin-4-yl}benzonitrile
N-cyclobutyl-4-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)pyrimidin-2-amine
(4aR,7aS)-4-[(4-methoxyphenyl)methyl]-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-[(3-methoxyphenyl)methyl]-4-(1-methyl-1H-pyrazole-4-carbonyl)piperazin-2-one
1-[4-(1-benzofuran-2-yl)pyrimidin-2-yl]-5-cyclopropyl-N-[3-(morpholin-4-yl)propyl]-1H-pyrazole-4-carboxamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propyl-1-benzothiophene-5-carboxamide
5-chloro-15-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-13-oxo-9-(thiophen-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
5-[1-methyl-3-(2-methylpropyl)-1H-pyrazol-5-yl]-3-[(methylsulfanyl)methyl]-1,2,4-oxadiazole
6-(4-chlorophenyl)-N-ethyl-N-(pyridin-2-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
9-methoxy-7-(5-methylthiophen-2-yl)-4-[2-(1H-pyrazol-4-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-(2,5-dimethoxyphenyl)-1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}pyrrolidine
(5S,9aS,9bS)-5-[2-(2-phenylethynyl)phenyl]-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-2-[2-(3-methoxyphenyl)pyrrolidin-1-yl]pyridine
2-{5-[(phenylsulfanyl)methyl]-1,2,4-oxadiazol-3-yl}pyrazine
N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-4-methoxybenzamide
1-(carbamoylmethyl)-N-ethyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}piperidine-3-carboxamide
N-[(2-fluorophenyl)methyl]-2-({[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}amino)acetamide
(5S)-5-[3-(3,3-diphenylpiperidin-1-yl)-3-oxopropyl]imidazolidine-2,4-dione
ethyl 2-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)acetate
N-[2-(4-fluorophenyl)ethyl]-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-1,3-thiazole-5-carboxamide
6-ethyl-5-methyl-N4-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}pyrimidine-2,4-diamine
1,3-dimethyl-6-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(cyclobutylmethyl)-3-hydroxy-3-[(4-hydroxypiperidin-1-yl)methyl]piperidin-2-one
1-{2-[4-(3-chloro-5-fluoro-4-methoxyphenyl)-1H-1,2,3-triazol-1-yl]ethyl}piperazine
1-[(3R,4R)-4-amino-3-hydroxypiperidin-1-yl]-2-(3-chlorophenyl)ethan-1-one
(1R,2S,6R,7S)-4-(1,5-dimethyl-1H-pyrrole-2-carbonyl)-4-azatricyclo[5.2.2.02,6]undecane
4-[4-(1H-imidazol-1-yl)benzoyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
{1-[(4,5-diphenyl-1H-imidazol-1-yl)methyl]cyclobutyl}methanol
(1R,3S)-3-ethoxy-7-(quinoxaline-5-carbonyl)-7-azaspiro[3.5]nonan-1-ol
4-({2-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]phenyl}methyl)morpholine
2-benzyl-4-(2-chlorobenzenesulfonyl)morpholine
1-methyl-4-[2-(4-propoxyphenoxy)ethyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(4-fluorophenyl)-N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}acetamide
N-[(3S,4R)-1-[5-(ethylsulfanyl)thiophene-2-carbonyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
9-(8-methoxyquinolin-2-yl)-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
3-ethoxy-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)benzamide
4-[5-(methoxymethyl)-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-1-yl]benzene-1-sulfonamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-{3-[3-(1,3-benzoxazol-2-yl)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
2-{2-[(4-methyl-3-phenylpiperazin-1-yl)methyl]phenoxy}ethan-1-ol
4-methoxy-2-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)phenol
N-methyl-N-(oxan-2-ylmethyl)-4-(pyridin-2-yl)pyrimidin-2-amine