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(1S,5R)-3-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-(1-phenylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
2-(adamantan-1-yl)-N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}acetamide
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-N,5-dimethyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
N-methyl-3-phenyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-1,2,4-oxadiazol-5-amine
1-[(4-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}phenyl)methyl]-5-methyl-1H-1,2,3,4-tetrazole
(2S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-4-{[(2,5-dimethylphenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
4-(2-methoxyphenyl)-1-(1,3-thiazol-4-ylmethyl)piperidine
7-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
[(2S,6S)-11-methoxy-4-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
5-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]pyrazin-2-ol
2-tert-butyl-6-(2,2,3,3-tetramethylcyclopropanecarbonyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
6-(2,5-dimethylfuran-3-yl)-N-(2-hydroxypropyl)-N,7-dimethyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
8-chloro-2-(furan-2-yl)-N-[(5-methyl-1,2-oxazol-3-yl)methyl]quinoline-4-carboxamide
5,7-dimethyl-N-(piperidin-4-ylmethyl)pyrido[2,3-d]pyrimidin-4-amine
N-(1-{1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-4-yl}-2-phenylethyl)-N-methylpyridine-2-carboxamide
[(1-ethyl-1H-pyrazol-4-yl)methyl][(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl](2-methylpropyl)amine
3-ethyl-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-1-methyl-N-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propanamide
N-{[7-chloro-2-(dimethylamino)quinolin-3-yl]methyl}-3,4-dimethoxy-N-(2-methoxyethyl)benzamide
{4-[1-(cyclohexylmethyl)-1H-1,2,4-triazol-5-yl]phenyl}methanol
2-hydroxy-4-methoxy-N-{[1-(oxan-4-yl)piperidin-3-yl]methyl}benzamide
1-phenyl-N-({1-[2-(phenylsulfanyl)acetyl]piperidin-3-yl}methyl)methanesulfonamide
methyl 3-[9-hydroxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanoate
4-(3-chloro-4-{[(2R)-2-methylpyrrolidin-1-yl]methyl}phenyl)pyridine
methyl 2-{[5-(2-methoxyacetamido)-1-(2-phenylethyl)-1H-1,3-benzodiazol-7-yl]formamido}-4-(methylsulfanyl)butanoate
4-(2,2-diethylmorpholine-4-carbonyl)-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
3-cyclopropyl-5-(4-methanesulfonylphenyl)-1-(2-phenylethyl)-1H-1,2,4-triazole
1-methyl-N-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(2S)-2-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)-2-phenylethan-1-ol
1-[1-(3-cyano-4,6-dimethylpyridin-2-yl)piperidin-4-yl]-N-cyclopropylpiperidine-3-carboxamide
3-(1-benzyl-1H-imidazol-2-yl)-1-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperidine
methyl 3-{[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]carbamoyl}propanoate
1-cyclopropyl-N-[3-(1H-indazol-1-yl)propyl]-5-oxopyrrolidine-3-carboxamide
1-(carbamoylmethyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]piperidine-4-carboxamide
2-(cyclopropylamino)-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}acetamide
4-(4,6-dimethylpyrimidin-2-yl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
2-({[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl)amino}methyl)-3-methoxyphenol
1-{7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(pyrazin-2-yl)propan-1-one
4-[1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-methyl-2-oxo-8-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylic acid
dimethyl({[(1R,5S,6S)-3-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]-3-azabicyclo[3.1.0]hexan-6-yl]methyl})amine
(3aR,6aS)-2-[(5-chloro-2,4-dimethoxyphenyl)methyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole
(E)-2-phenyl-N-{2-[4-(propan-2-yl)morpholin-2-yl]ethyl}ethene-1-sulfonamide
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
3-(3-chlorophenyl)-3-(2-hydroxyphenyl)-N-[(1r,4r)-4-hydroxycyclohexyl]propanamide
3-ethyl-N-(2-methoxyethyl)-4-methyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-5-carboxamide
9-(cyclopropylmethyl)-1-methyl-4-(4,4,4-trifluorobutyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
4-methyl-5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyrimidine
N-[(5-chloro-2-ethoxyphenyl)methyl]-N,1-dimethyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide