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2-methoxy-3-{[3-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}quinoline
1-(cyclohexylmethyl)-3-[(cyclopentylamino)methyl]-3-hydroxypiperidin-2-one
2-[3-(1-{[6-(trifluoromethyl)pyridin-3-yl]methyl}-1H-pyrazol-3-yl)phenyl]pyrazine
1-[6-(4-methoxyphenyl)-7-oxo-6,9-diazaspiro[4.5]decan-9-yl]-2-phenylethane-1,2-dione
2-fluoro-6-hydroxy-N-[(3-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)benzamide
N-(isoquinolin-5-ylmethyl)-N-methyl-2-(morpholin-4-yl)pyrimidine-5-carboxamide
5-methoxy-3-methyl-2-{[4-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-1H-indole
1-(3,3-diphenylpiperidin-1-yl)-2-(oxolan-2-ylmethoxy)ethan-1-one
2-(4-methyl-1H-imidazole-2-carbonyl)-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
1-ethyl-N-[(3-methoxyphenyl)methyl]-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
methyl 4-{[(1-{4-[2-(4-methoxyphenyl)acetamido]phenyl}piperidin-4-yl)amino]methyl}benzoate
(1R,5R)-6-(1-ethyl-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-[(3-chlorophenyl)methyl]-2-[4-(3-methyl-1H-pyrazole-5-carbonyl)morpholin-3-yl]acetamide
1-[3-(4-tert-butylbenzoyl)piperidin-1-yl]-2-(2H-1,2,3,4-tetrazol-2-yl)ethan-1-one
1-{5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-4-ethylpiperazine
N-(furan-2-ylmethyl)-N,1-dimethyl-5-{[(2-methylphenyl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
7-methoxy-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,2,3,4-tetrahydronaphthalen-2-amine
7-methoxy-3-({methyl[(1-methylpiperidin-3-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-N'-(4-methylphenyl)propanediamide
1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-4-[(4-fluorophenyl)methyl]piperidine
5,6,7-trimethoxy-N,N-dimethyl-3-{[(2-methylpropyl)amino]methyl}quinolin-2-amine
N-cyclopropyl-2-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}acetamide
N-cyclopropyl-6-ethyl-2-methyl-N-(pyridin-2-ylmethyl)quinoline-4-carboxamide
5-hydroxy-1,2-dimethyl-N-[2-(pyrrolidin-1-yl)ethyl]-1H-indole-3-carboxamide
1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-3-(pyridin-2-yl)propan-1-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}acetamide
2-[(3,5-difluorophenyl)methyl]-8-(1-methylpiperidin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
2-(2-aminoethyl)-N-[(4-methoxyphenyl)methyl]-N-(prop-2-yn-1-yl)quinazolin-4-amine
3-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]pyridine
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-(6,7-dimethyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetamide
3-(benzyloxy)-1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
1-{3-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-4-(piperidin-1-yl)butanamide
5-(2-chlorophenyl)-2-methyl-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]furan-3-carboxamide
4-(3-methylpiperidine-1-carbonyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine
8-(5,6-dimethylpyrimidin-4-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(2E)-1-(3-{[(dimethylsulfamoyl)amino]methyl}piperidin-1-yl)-4-methylpent-2-en-1-one
N-tert-butyl-5-{1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
N-[(1-cyclopentylpiperidin-3-yl)methyl]-3-methyl-N-[2-(piperidin-1-yl)ethyl]thiophene-2-carboxamide
5-methyl-3-phenyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1,2-oxazole-4-carboxamide
1-methyl-1'-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[2-(naphthalen-1-yl)pyrimidin-5-yl]methyl})amine
N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
1-(1-methylpiperidin-4-yl)-N-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
2-[({3-methoxy-2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)amino]acetamide
N-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-3-yl)pyrimidin-2-amine
1-cyclohexyl-N-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
8-[2-(2-methyl-1H-imidazol-1-yl)acetyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[2-(2-chlorophenyl)ethyl]-5-[2-(ethylamino)ethyl]pyrrolidin-2-one
2-cyclopentanecarbonyl-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-6-one