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N-[(3R,4S)-4-cyclopropyl-1-[4-(piperidin-1-yl)butanoyl]pyrrolidin-3-yl]methanesulfonamide
1-(5-methyl-1,3,4-oxadiazol-2-yl)-4-(pyridin-4-yl)piperazine
[1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-2-yl]methanol
3-[5-(oxolane-3-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl]pyridine
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N,2,8-trimethylquinoline-4-carboxamide
1-(2-oxo-2-{2-oxo-1-oxa-3,8-diazaspiro[4.6]undecan-8-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-ethyl-1-[(2E)-3-phenylprop-2-en-1-yl]-1,4-diazepan-5-one
(3S,4R)-3-benzyl-4-methyl-1-(4-methylpyrimidin-2-yl)piperidin-4-ol
N-methyl-N-[(1-methyl-5-oxopyrrolidin-3-yl)methyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
4-[3-(hydroxymethyl)morpholine-4-carbonyl]-1,2-dihydroquinolin-2-one
1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-4-[(3-methylphenyl)methyl]piperazine
methyl 2-[1-(2-butyl-1,3-benzoxazole-5-carbonyl)-3-oxopiperazin-2-yl]acetate
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]acetamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(propan-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-methyl-6-{1-[3-(methylsulfanyl)propyl]piperidin-4-yl}pyrimidin-4-ol
1'-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,2-dihydrospiro[indole-3,4'-piperidine]
2-{2-[4-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-1H-1,2,3-triazol-1-yl]ethyl}-5,6-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-{[4-(but-3-yn-1-yloxy)phenyl]methyl}-N-(oxolan-2-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
2-amino-N-{2-[4-(hydroxymethyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-5-yl}-2-methylpropanamide
N-[2-(azepane-1-carbonyl)phenyl]-3-(3-methyl-1H-1,2,4-triazol-5-yl)propanamide
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-N,N-bis(prop-2-en-1-yl)pyridin-2-amine
(2S,4S)-1-benzyl-N-methyl-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
[2,4,6-trimethyl-3-({[(1-methyl-1H-pyrazol-5-yl)methyl]amino}methyl)phenyl]methyl acetate
3-[(3S,5R)-3-(hydroxymethyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidine-1-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one
8-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-oxa-8-azaspiro[4.6]undecane
1-{2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole-5-carbonyl}azetidin-3-ol
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-5-methoxyfuran-2-carboxamide
(2R,3S,6R)-5-(3-methoxypropyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(3-fluorophenyl)-6-(hydroxymethyl)-1,4-oxazepane-4-carboxamide
3-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-1-(furan-2-ylmethyl)-1-(thiophen-2-ylmethyl)urea
1-(2,3-dihydro-1H-inden-2-yl)-4-{[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}pyrrolidin-2-one
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[(1R,2S)-2-phenylcyclopropyl]acetamide
6-methyl-1-(propan-2-yl)-4-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-1H-pyrazolo[3,4-b]pyridine
2-[(3S)-3-aminopiperidine-1-carbonyl]-6-(4-fluorophenyl)-7-methyl-7H,8H-imidazo[1,2-a]pyrazin-8-one
4-{3-[2-(4-methoxyphenyl)ethyl]piperidine-1-carbonyl}-2,6-dimethylpyrimidine
N-(2-methoxyethyl)-1-[1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
(3R,4R)-4-(azepan-1-yl)-1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]piperidin-3-ol
(8aS)-2-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-(1H-indazol-1-yl)-N-[(2-phenoxypyridin-3-yl)methyl]acetamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-3-ol
N-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}acetamide
6-methyl-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
3-(2,6-dimethylphenoxy)-1-(3-fluoro-4-methylbenzoyl)azetidine
(4aS,8aS)-2-[6-(methoxymethyl)pyrimidin-4-yl]-7-propyl-decahydro-2,7-naphthyridin-4a-ol
3-(2-methylpropyl)-N-[2-(pyridin-4-yl)ethyl]-1,2-oxazole-5-carboxamide
2-{[4-(4-chlorophenoxy)piperidin-1-yl]methyl}pyridine
[(3S,5R)-5-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(pyrimidin-2-yl)piperidin-3-yl]methanol
1-ethyl-8-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
{[3,5-dichloro-4-(prop-2-en-1-yloxy)phenyl]methyl}(ethyl)[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]amine