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N-[(3S)-1-benzylpyrrolidin-3-yl]-4-methyl-1,3-oxazole-5-carboxamide
2-({3-[4-(2,4-difluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-5-methoxyphenol
7-(3-chlorophenyl)-4-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[2-methyl-3-({[1-(4-methylpyridin-2-yl)propyl]amino}methyl)-1H-indol-1-yl]acetamide
N-(2-hydroxyethyl)-N-methyl-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
N-[4-methoxy-3-(methylcarbamoyl)phenyl]-2-oxo-1-oxa-3,8-diazaspiro[4.6]undecane-8-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-(2,3-dihydro-1H-inden-2-yl)pyrrolidin-3-yl]-2-methoxyacetamide
(3R)-1-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}pyrrolidin-3-ol
4-[5-(2-butylpyrrolidine-1-carbonyl)-1H-pyrazol-3-yl]pyridine
(3S,4S)-4-(4-fluorophenyl)-1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-ol
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]quinoline-3-carboxamide
1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-2-(3-methoxypropyl)piperidine
7-(2,2-dimethylpropyl)-2-{[5-(hydroxymethyl)furan-2-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
1-{1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}azepan-4-ol
1-{4-[(3-chlorophenyl)methyl]piperazin-1-yl}-2-(oxolan-2-ylmethoxy)ethan-1-one
1-[(2E)-3-phenylprop-2-en-1-yl]-4-(1H-1,2,3-triazole-5-carbonyl)piperazine
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-(2-methoxyethyl)-5-(methoxymethyl)-N-(propan-2-yl)-1H-pyrazole-4-carboxamide
4-[(2-ethoxyphenyl)methyl]-9-methoxy-7-(4-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
8-acetyl-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-(cyclohexylmethyl)-3-hydroxy-3-({[(6-methylpyridin-2-yl)methyl]amino}methyl)piperidin-2-one
3-(5-fluoro-2-methoxybenzoyl)piperidine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(1-methyl-1H-pyrazol-5-yl)propanamide
2-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pyridine-3-carboxamide
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-1-methyl-1H-1,2,3-triazol-4-amine
2-{2-[6-amino-5-cyano-4-(pyridin-3-yl)pyridin-2-yl]phenoxy}acetamide
(1R,5S)-6-(1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carbonyl)-6-azabicyclo[3.2.1]octane
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-(3-methylphenoxy)piperidine-4-carboxylic acid
3-{methyl[(2-methyl-1,3-oxazol-4-yl)methyl]amino}-1-phenylpropan-1-ol
1-[(1,3-dimethylpyrrolidin-3-yl)methyl]-1-methyl-3-(2-phenyl-1,3-benzoxazol-5-yl)urea
N-(cyclohex-1-en-1-ylmethyl)-2-(1,1-dioxo-1λ6-thiomorpholin-4-yl)benzamide
5-methoxy-2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
2-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
N-[2-(cyclohex-1-en-1-yl)ethyl]-5-methyl-6-(pyrrolidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
{3-[(3-methoxyphenyl)methyl]-1-[(3,4,5-trimethoxyphenyl)methyl]piperidin-3-yl}methanol
N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-[3-(2-methyl-1H-imidazol-4-yl)phenyl]ethan-1-one
5-fluoro-2-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]phenol
3-(3-fluorophenoxymethyl)-1-methyl-5-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-1,2,4-triazole
4-{3-ethyl-5-[(pyridin-2-ylsulfanyl)methyl]-1H-1,2,4-triazol-1-yl}benzene-1-sulfonamide
4-(2-methyl-1H-imidazol-1-yl)-1-(4-methylpyrimidin-2-yl)piperidine-4-carboxylic acid
2-[1-(2-methylpropyl)-4-(pyridin-4-ylmethyl)piperazin-2-yl]ethan-1-ol
3-cyclopentaneamido-N,4-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]benzamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2,3-dihydro-1-benzofuran-7-carboxamide
1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-ethyl-N-methylacetamide
(1S,5R)-3-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(1R)-1-(4-chlorophenyl)ethyl]-4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carboxamide
4-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-ylmethyl}benzamide
N-[2-(azepan-1-yl)ethyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)thiophene-2-carboxamide