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1-cyclopropanecarbonyl-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]piperidine-4-carboxamide
(3S,4S)-4-(4-fluorophenyl)-1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-3-ol
1,3-dimethyl-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-[(4-fluoro-3-methoxyphenyl)methyl]-3-[4-(methylsulfanyl)benzoyl]piperidine
N-(pyridin-3-ylmethyl)-1-[1-(thiophen-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
4-ethyl-1-[(2,3,6-trifluorophenyl)methyl]-1,4-diazepan-5-one
2-benzyl-9-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-2,9-diazaspiro[5.5]undecan-3-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-4-hydroxy-N-methyl-2-(thiophen-2-yl)pyrimidine-5-carboxamide
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(1,2,5-trimethyl-1H-pyrrole-3-carbonyl)pyrrolidin-3-yl]methanol
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
1-(3-{[4-benzyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenyl)ethan-1-one
N-(prop-2-en-1-yl)-N-(propan-2-yl)-2-(1H-1,2,4-triazol-1-yl)benzamide
3-{1-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-3-yl}benzoic acid
3-hydroxy-1-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
1-(2-{4-[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-1H-1,2,3-triazol-1-yl}ethyl)imidazolidin-2-one
4-(2H-1,3-benzodioxol-4-ylmethyl)-1-(oxan-4-ylmethyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
N-{[7-methoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-4-methyl-N-(oxolan-2-ylmethyl)benzamide
(2R,6R)-11-methoxy-4-(1H-pyrrole-2-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-cyclopentyl-4-({[(2,3-difluoro-6-methoxyphenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
4-[3-(3-ethylphenoxy)azetidine-1-carbonyl]-1-(2-methoxyethyl)piperidine
3-{5-[1-(2-methoxyethyl)piperidin-3-yl]-1,2,4-oxadiazol-3-yl}pyridazine
(3S,9aR)-3-benzyl-8-(quinolin-5-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[1-(1-{[3-(2-hydroxyethoxy)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]oxolane-3-carboxamide
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-1H-indole-5-carboxamide
3-methyl-N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)-2-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)pentanamide
1-[2-(azetidin-1-yl)-2-oxo-1-phenylethyl]-4-butylpiperazine-2,3-dione
1-(4-methanesulfonylphenyl)-3-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]urea
7-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-2-(2-oxopiperidin-1-yl)-N-(pyridin-3-ylmethyl)acetamide
methyl 2-{[1-(4-cyclopentaneamidophenyl)piperidin-4-yl]amino}acetate
[1-(1-{[2,5-dimethyl-1-(pyridin-3-yl)-1H-pyrrol-3-yl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]methanol
4-(1-{1-[2-(pyridin-2-yl)ethyl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
6-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(2,4-difluorophenyl)methyl]-2-[4-(propan-2-yl)morpholin-2-yl]acetamide
methyl 5-[(2,2-dimethylpropyl)amino]-3-acetamido-1-[2-(1H-indol-3-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[1-(pyridin-4-yl)propyl]-1H-pyrazole-3-carboxamide
2-[1-(2-ethylpyrimidine-5-carbonyl)piperidin-4-yl]-1,3-benzoxazole
[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)[(6-methylpyridin-2-yl)methyl]amine
2-methyl-4-[4-(pyrrolidin-1-ylmethyl)phenyl]butan-2-ol
methyl 6-(pyrazine-2-carbonyl)-2-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
ethyl 4-[1-(6-ethoxy-4-methylquinazolin-2-yl)piperidine-4-amido]piperidine-1-carboxylate
2-(1H-1,3-benzodiazol-1-yl)-1-[3-(3-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}phenoxymethyl)piperidin-1-yl]ethan-1-one
N'-(4-methylphenyl)-N-{[(1,3-thiazol-2-yl)carbamoyl]methyl}propanediamide
9-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-[1-(pyrrolidin-1-yl)ethyl]piperidine
2-{4-[(3aR,6aR)-2-cyclopropanecarbonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]piperazin-1-yl}-N,N-dimethylacetamide
1-[2-(3-methylphenyl)benzoyl]-4-(1-methylpiperidin-4-yl)piperazine
4-(cyclopentylamino)-1-[2-(4-methoxyphenyl)ethyl]pyrrolidin-2-one
methyl 2-[4-(2-{[(2-chlorophenyl)methyl]sulfanyl}acetamido)piperidin-1-yl]acetate