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(4-{[1-(2-methoxyphenoxy)propan-2-yl]amino}quinazolin-2-yl)methanol
N-(3-cyano-4,5-dimethylfuran-2-yl)-4-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}benzamide
1-({4-methyl-5-[1-(1,3-thiazol-2-ylmethyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
(1H-1,3-benzodiazol-2-ylmethyl)({[1-(cyclohexylmethyl)-2-methanesulfonyl-1H-imidazol-5-yl]methyl})methylamine
2-[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]-6-methyl-1H-1,3-benzodiazole
4-{[1-(3,5-dichloro-4-methylbenzoyl)piperidin-3-yl]methyl}morpholine
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-[2-(methylsulfanyl)pyridine-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(morpholin-4-yl)ethyl]acetamide
4-{[3-(2-chlorophenyl)pyrrolidin-1-yl]methyl}-1,3-thiazole
2-{4-[(6-ethoxypyridin-3-yl)methyl]piperazin-1-yl}-6-methylpyridine-3-carboxamide
2-benzyl-4-(1H-pyrazole-4-carbonyl)morpholine
7-{[3-(methoxymethyl)piperidin-1-yl]methyl}-4-[(4-methoxynaphthalen-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(3-phenylpropyl)-4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}morpholine
N-(1H-imidazol-2-ylmethyl)-N-methyl-3-[(2R)-2-methylpiperazine-1-carbonyl]benzene-1-sulfonamide
methyl 2-(azocane-1-sulfonyl)-6-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-(azetidine-1-carbonyl)-N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methylbenzene-1-sulfonamide
3-(3-cyanopiperidine-1-carbonyl)-N-(1H-pyrazol-3-ylmethyl)benzene-1-sulfonamide
2-{4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
1-({3-methoxy-4-[(3-methylbut-2-en-1-yl)oxy]phenyl}methyl)-2-(methoxymethyl)piperidine
4-methoxy-6-(3-{1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrimidine
1-[1-(4-cyclohexylpiperazine-1-carbonyl)-6-azaspiro[2.5]octan-6-yl]-3-(furan-2-yl)propan-1-one
3-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1-[4-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]urea
(5-{1-[(2-ethoxypyridin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}furan-2-yl)methanol
1-({5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-7-yl}methyl)-1,2-dihydroquinoxalin-2-one
2-({[(3R,4R)-1-(2-chloro-6-fluorobenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-[(3R)-3-phenylbutyl]-4-(pyridin-2-ylmethyl)piperazine
N-[5-({[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]carbamoyl}amino)-2-methoxyphenyl]propanamide
N-[(3R,4S)-4-cyclopropyl-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-3-methanesulfonamidopropanamide
8-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
5-({4-[(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)-2-hydroxybenzoic acid
4-[(1S,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]butanamide
2-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
N-methyl-3-(2-methylpropyl)-N-(thiophen-2-ylmethyl)-1,2-oxazole-5-carboxamide
N-(2-hydroxyethyl)-N-(thiophen-2-ylmethyl)oxolane-3-carboxamide
4-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-2-methyl-1,3-thiazole
1-[1-methyl-5-(thiophen-2-yl)-1H-pyrazole-3-carbonyl]-4-[(2-methylphenyl)methyl]piperazine
1-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-3-[1-(pentan-3-yl)-1H-pyrazol-5-yl]urea
ethyl 2-{[3-(3-chlorobenzoyl)piperidine-1-carbonyl]amino}acetate
1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-amine
5-acetyl-N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)thiophene-3-carboxamide
N-(1-{1-[(4-hydroxy-3,5-dimethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2,2-dimethylpropanamide
4-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-1-methyl-2-phenylpiperazine
N-methyl-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-(quinoxalin-2-ylmethyl)propanamide
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[1-(pyrazin-2-yl)propan-2-yl]acetamide
1-[(2,6-difluorophenyl)methyl]-4-(2-methylphenoxy)piperidine-4-carboxylic acid
1-[(2,3-difluorophenyl)methyl]-4-(pyrrolidin-3-yl)piperazine
N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-3-azaspiro[5.5]undecan-9-amine
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-methyl-N-[1-(pyridin-3-yl)propyl]benzamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-(2-methoxyethyl)-N-(pyridin-3-ylmethyl)acetamide
5-methyl-4-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-2-[(oxolan-2-ylmethyl)sulfanyl]pyrimidine