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1-[4-(2-amino-6-methylpyrimidin-4-yl)piperazin-1-yl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
2-{4-methyl-3-oxo-1H,2H,3H-pyrazolo[3,4-b]pyridine-6-carbonyl}-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
3-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)-1-[(1-hydroxycyclohexyl)methyl]urea
1-[(4aR,8aS)-1-(1-methylcyclopropanecarbonyl)-decahydro-1,6-naphthyridin-6-yl]-4-phenylbutan-1-one
methyl 1-{2-hydroxy-3-[4-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]propyl}piperidine-4-carboxylate
N-(4-methoxy-2-methylphenyl)-2-[2-(pyrrolidin-1-yl)ethyl]piperidine-1-carboxamide
ethyl 2-{1-[5-(2-chloro-4-fluorophenoxymethyl)-1,2-oxazol-3-yl]-N-methylformamido}acetate
3-(pentan-2-yl)-8-[2-(pyrimidin-2-ylsulfanyl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-(2-methylpropyl)-1'-(6-methylpyridine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]-6-(propan-2-yl)pyridine-3-carbonitrile
[(3S,5R)-1-(2-chloro-5-methylbenzoyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
7-(4-chlorophenyl)-2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-(1-{3-[(2-methoxyphenyl)methyl]-1-methyl-1H-1,2,4-triazol-5-yl}cyclohexyl)morpholine
3-cyclopentyl-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N,4-dimethyl-4-[(2-methyl-4-oxo-1,4-dihydroquinolin-8-yl)formamido]pentanamide
13-[3-(3-methylbutoxy)phenyl]-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
N5-[(2,5-dimethoxyphenyl)methyl]-N2,N2-dimethyl-5,6,7,8-tetrahydroquinazoline-2,5-diamine
4-{1-[(1,3-dimethyl-1H-pyrazol-5-yl)sulfonyl]piperidin-3-yl}benzoic acid
4-cyclohexyl-1-[2-(1H-imidazol-1-yl)-1-phenylethyl]-1H-1,2,3-triazole
(2R,4S)-4-hydroxy-1-(3-phenylpropyl)piperidine-2-carboxylic acid
2-[({1-[1-(2-cyclohexylethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-3-yl}oxy)methyl]pyridine
2-{3,9-diazaspiro[5.5]undecan-3-ylmethyl}benzoic acid
N-[3-({[(6-hydroxypyrimidin-4-yl)methyl]carbamoyl}amino)phenyl]cyclopentanecarboxamide
N-benzyl-5-(4-benzylpiperidine-1-carbonyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
(1S,4S)-5-(1-benzylpiperidin-4-yl)-2-(2-fluorophenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
N-{[1-(methoxymethyl)cyclopropyl]methyl}-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
2-ethyl-1-{[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}piperidine
6,7-dimethyl-2-{[4-(pyridin-3-yl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-1,3-benzodiazole
1-{2-[methyl({[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl})amino]ethyl}piperidin-2-one
8-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-{4-[(3-cyclopropyl-1H-1,2,4-triazol-5-yl)methyl]phenyl}imidazolidin-2-one
2-(3-acetyl-1H-indol-1-yl)-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]butanamide
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-1H-pyrazole-4-carboxamide
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-3-propyl-1H-pyrazole-5-carboxamide
7-(2-phenylbenzoyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
4-(2-methoxypyridin-3-yl)-6-(4-methylpiperazin-1-yl)pyrimidin-2-amine
1-[(2,4-difluorophenyl)methyl]-3-[4-(2-methylpropyl)-1H-pyrazol-5-yl]piperidine
3-{1-[(5-cyclopentylthiophen-2-yl)methyl]piperidin-3-yl}-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
N-methyl-3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-[(5-propyl-1H-pyrazol-3-yl)methyl]propanamide
2-({4-[5-(2-methylpropyl)-1H-pyrazol-3-yl]-1H-1,2,3-triazol-1-yl}methyl)morpholine
(3R,5S)-N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
N-(3-{[(1-methylpiperidin-3-yl)methyl]sulfamoyl}phenyl)acetamide
8-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-2-methyl-2,8-diazaspiro[4.5]decane
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-(3-methoxypiperidin-1-yl)pyridine-3-carboxamide
(3R,5R)-N-[(3-phenylphenyl)methyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
1-(2-aminopyridine-4-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[(3S,4S)-3-hydroxy-4-(4-hydroxypiperidin-1-yl)pyrrolidin-1-yl]ethan-1-one
2-(2-oxo-1,2-dihydropyridin-1-yl)-N-[2-(propane-2-sulfonyl)ethyl]acetamide
9-{[2-(butan-2-yloxy)-3-methoxyphenyl]methyl}-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-[(trifluoromethyl)sulfanyl]ethan-1-one