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[(5-ethylfuran-2-yl)methyl](methyl)[4-(morpholin-4-yl)butyl]amine
5-(propan-2-yl)-N-[2-(pyrrolidin-1-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-(4-phenylphenyl)-5-(thiolan-3-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-(2-methyl-1,3-benzothiazol-5-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
1-(3-phenylpropyl)-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
(3R,4S)-4-[4-(2-amino-6-ethyl-5-methylpyrimidin-4-yl)-1,4-diazepan-1-yl]oxolan-3-ol
N-ethyl-1-(4-ethylbenzenesulfonyl)-N-(pyridin-4-ylmethyl)piperidin-3-amine
2-{[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
8-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-cyclopentyl-5-oxo-N-[1-(pyrazin-2-yl)piperidin-4-yl]pyrrolidine-3-carboxamide
ethyl 3-benzyl-1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidine-3-carboxylate
(2-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-oxoethyl)urea
N,5-dimethyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
2-(adamantan-1-ylsulfanyl)-N-[(1-methylpiperidin-3-yl)methyl]acetamide
2-(2-hydroxyethyl)-9-(naphthalen-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-{1-[(2E)-3-(1-methyl-1H-pyrazol-4-yl)prop-2-enoyl]pyrrolidin-2-yl}-N-(propan-2-yl)thiophene-2-carboxamide
6-(3-fluorophenyl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-{[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]methyl}-1,3-thiazole
3-[(3R,4S)-4-(dimethylamino)-1-[(1-methyl-1H-indol-2-yl)methyl]piperidin-3-yl]propan-1-ol
1-{[3-(phenoxymethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]methyl}piperidin-3-ol
1-[(4aS,8aS)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-3-(benzenesulfonyl)propan-1-one
3-(5-amino-1H-1,2,4-triazol-3-yl)-1-{2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}propan-1-one
N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
N-(4-{[3-(methanesulfonylmethyl)piperidin-1-yl]methyl}phenyl)acetamide
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]quinoxaline-5-carboxamide
8-[2-(4-fluoro-3-methylphenyl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(1-hydroxy-2-methylpropan-2-yl)acetamide
2-(methylamino)-1-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
3-(2-{2-methylimidazo[1,2-a]pyridin-3-yl}acetyl)-3,9-diazaspiro[5.6]dodecan-10-one
3-{1-[2-(5-acetylthiophen-3-yl)acetyl]piperidin-3-yl}-1-(morpholin-4-yl)propan-1-one
1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-2-(5-methyl-1,2-oxazol-3-yl)piperidine
4-chloro-1-methyl-N-({1-[(4-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-1H-pyrazole-3-carboxamide
N-(1-cycloheptylpiperidin-3-yl)butanamide
1-[(3-{[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]-4-(2-fluorophenyl)piperazine
N-{2-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-oxoethyl}acetamide
3-[1-(cyclohex-1-ene-1-carbonyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)propanamide
1-[4-(2,5-dihydro-1H-pyrrol-1-yl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-2-(pyridin-3-yl)ethan-1-one
N,N-dimethyl-5-{2-oxo-1-oxaspiro[4.5]decane-4-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(2R,3R)-3-{methyl[2-(oxan-4-yl)ethyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-chloro-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylbenzamide
4-[5-cyclopropyl-4-(4-ethylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]-3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaene
N-[1-(4-methoxyphenyl)ethyl]-N-methyl-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
9-(cyclopropylmethyl)-1-methyl-4-[(1-methyl-1H-imidazol-2-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
7-methyl-2-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2,7-diazaspiro[4.5]decan-6-one
N-(3-chloro-4-methoxyphenyl)-3-{1-[(5-cyano-1H-pyrrol-3-yl)methyl]piperidin-3-yl}propanamide
4-(2,5-dimethylfuran-3-carbonyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
(3S)-N,N-dimethyl-1-(4-methyl-1H-imidazole-2-carbonyl)azepan-3-amine
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
{1-[({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)methyl]cyclopropyl}methanol