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3-(1-benzyl-1H-imidazol-2-yl)-1-(1-methyl-1H-pyrazole-3-carbonyl)piperidine
2-butyl-N-(6-hydroxy-6-methylheptan-2-yl)-1,3-benzoxazole-5-carboxamide
1-(1H-imidazol-2-ylmethyl)-4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine
3-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]-1-(5-fluoropyridin-3-yl)urea
N-(2-{7-[(3,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-3-carboxamide
1-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
methyl 8-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]-1-methoxy-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
2-{[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]({[4-(methylsulfanyl)phenyl]methyl})amino}ethan-1-ol
1-{6-[4-(adamantan-1-yl)piperazin-1-yl]pyridin-2-yl}ethan-1-ol
N-[1-(methoxymethyl)cyclopentyl]-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[(2-methylpyrimidin-5-yl)methyl]-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
2-amino-4-(1-ethyl-1H-pyrazol-4-yl)-6-(1-phenyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-[2-(pyridin-4-yl)ethyl]-1,9-dioxaspiro[5.5]undecan-4-amine
methyl 1-{[1-(3-fluoro-4-hydroxyphenyl)ethyl]carbamoyl}cyclopropane-1-carboxylate
[(3S,5R)-1-(3-fluorobenzoyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
2-{2-[2-(aminomethyl)morpholin-4-yl]-2-oxoethyl}-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
9-(5-chloro-2-hydroxybenzoyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
2,3-dimethyl-N-{[4-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)-1H-indole-7-carboxamide
5-[3-(1-tert-butyl-3-methyl-1H-1,2,4-triazol-5-yl)propyl]-3-(2-methoxyphenyl)-1,2,4-oxadiazole
N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
N-[3-(methylsulfanyl)propyl]-1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(2S)-2-amino-6-hydroxy-1-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}hexan-1-one
N'-(prop-2-en-1-yl)-N'-(pyridin-4-ylmethyl)-N-(2,4,6-trimethylphenyl)butanediamide
N-{[4-(cycloheptyloxy)-3-methoxyphenyl]methyl}-N-(pyridin-2-ylmethyl)cyclopropanecarboxamide
(1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-3-(2-phenylethyl)piperidin-3-yl)methanol
(1R,6S)-N-butyl-6-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}cyclohex-3-ene-1-carboxamide
8-(3-methoxy-4-methylbenzoyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
3-[3-(4-ethylpiperazin-1-yl)propyl]-8-(thiolan-3-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
9-methoxy-N-methyl-7-oxo-3-(3-phenoxypropanoyl)-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-methyl-N-{2-[methyl(phenyl)amino]propyl}-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
2-[3-(2-methylphenoxy)azetidine-1-carbonyl]benzonitrile
1-ethyl-2-{1-[3-(1H-pyrazol-1-yl)propyl]-1H-imidazol-2-yl}-1H-imidazole
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-3-[(oxolan-3-ylmethyl)sulfamoyl]benzamide
8-chloro-2-(furan-2-yl)-N-[1-(pyrimidin-4-yl)ethyl]quinoline-4-carboxamide
1-{1-[3-(methylsulfanyl)propanoyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
(3S,4R)-1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
N-[1-(4-methanesulfonylphenyl)ethyl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
3-[1-(1-aminocyclopropanecarbonyl)piperidin-4-yl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
5-{2-[4-(benzenesulfonyl)piperazin-1-yl]-2-oxoethyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
1-(benzenesulfonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
3-methoxy-1-{4-[4-(3-methylpiperidine-1-carbonyl)phenoxy]piperidin-1-yl}propan-1-one
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-4-methyl-1,3-thiazole-5-carboxamide
N-{[(2S,4S)-4-fluoro-1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}pyrrolidin-2-yl]methyl}methanesulfonamide
3-{[7-acetyl-2-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}-1-(pyrrolidin-1-yl)propan-1-one
(1S,2S)-2-{4-[(5-methyl-2-phenyl-1H-imidazol-4-yl)methyl]piperazin-1-yl}cyclohexan-1-ol
1-{[1-butyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}pyrrolidin-2-one
1-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-(3-hydroxy-1,2-oxazol-5-yl)propan-1-one
3-[1-(2-chlorophenyl)-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-5-yl]-1λ6-thiolane-1,1-dione
4-tert-butyl-6-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-1,2-dihydropyrimidin-2-one