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1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-2-(1-methyl-1H-pyrazol-3-yl)piperidine
N-butyl-6-(4-methoxyphenyl)-N,7-dimethyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-[(1S,2R)-2-hydroxy-1,2-diphenylethyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
4-[(3S,5R)-5-[4-(4-methyl-1H-pyrazol-3-yl)piperidine-1-carbonyl]piperidine-3-carbonyl]morpholine
3,3,3-trifluoro-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}propane-1-sulfonamide
1-(oxan-4-yl)-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
2-{4-benzyl-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
4-(2-{[(3,5-dimethylphenyl)methyl]sulfanyl}acetyl)piperazine-2-carboxylic acid
[(3-{2-[4-(3-chloro-2-methylbenzenesulfonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)(thiophen-2-ylmethyl)amine
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2-[3-(trifluoromethyl)phenyl]ethan-1-one
3-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-[4-(furan-2-carbonyl)piperazin-1-yl]propan-1-one
1-[(3-ethenylphenyl)methyl]-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazine
2-{3-[1-(3-methoxypropyl)-1H-pyrazol-3-yl]phenyl}-6-methylpyridine-3-carbonitrile
ethyl 2-({4-[2-(3-chlorophenyl)ethyl]-3-oxo-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-11-yl}(methyl)amino)acetate
7-methoxy-N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}-1,2,3,4-tetrahydronaphthalen-2-amine
[(4-fluorophenyl)methyl](methyl){[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}amine
[(3R,4R)-1-(5-methoxypyrimidin-2-yl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-(dimethyl-1,2-oxazol-4-yl)-1,1-dioxo-1λ6-thiomorpholine-4-carboxamide
N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
methyl N-{2-[2-(4-chlorophenyl)morpholin-4-yl]-2-oxoethyl}carbamate
(1-{[1-(thian-4-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
1-{1-[2-(ethylsulfanyl)ethyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-6-aminopyridine-2-carboxamide
(3R,4R)-1-[(3-chloro-4-ethoxyphenyl)methyl]-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
5-[1-(2,1,3-benzothiadiazol-5-ylmethyl)pyrrolidin-2-yl]-N-(propan-2-yl)thiophene-2-carboxamide
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-2-(dimethylamino)-2-(3-methylphenyl)acetamide
1-{1-[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2,5-dimethylfuran-3-carboxamide
1-(1,3-dihydro-2-benzofuran-5-yl)-3-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-3-methylurea
3-[({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1H-1,2,4-triazol-5-amine
2-({3-[5-(4-fluorophenyl)-2-methylpyrimidin-4-yl]piperidin-1-yl}methyl)-1,3-benzothiazole
N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-3-[(oxolan-3-yl)sulfamoyl]benzamide
(2S)-2-({1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-4-methylpentan-1-ol
1-methyl-N-[3-(methylsulfanyl)propyl]-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
(4aS,8aR)-6-{2-[4-(methylsulfanyl)phenyl]acetyl}-decahydro-1,6-naphthyridine-4a-carboxylic acid
1-[(4-methoxyphenyl)methyl]-4-[2-(methylsulfanyl)acetyl]piperazin-2-one
{3-[(dimethylamino)methyl]-1-{[2-(5-methylfuran-2-yl)phenyl]methyl}piperidin-3-yl}methanol
3-(2-ethyl-1H-imidazol-1-yl)-1-[(3S)-3-ethylmorpholin-4-yl]propan-1-one
2-(3-methoxypropyl)-N-(3-methylphenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
1-({1-[(2-chloro-6-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}methyl)azepan-2-one
(2S,4R)-1-(cyclohexylmethyl)-N-ethyl-4-(5-methylthiophene-3-amido)pyrrolidine-2-carboxamide
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-4-(4H-1,2,4-triazol-4-yl)benzamide
3-(2-methoxyphenyl)-5-[2-(methylsulfanyl)ethyl]-1,2,4-oxadiazole
1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-4-(pyridin-4-ylmethyl)-1,4-diazepane
N,N-dimethyl-1-{[3-(thiophen-3-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-3-amine
1-[4-(furan-2-yl)pyrimidin-2-yl]-N-(1-methoxybutan-2-yl)-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
1-[7-(3-chlorophenyl)-9-(furan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methylpropan-1-one
6-(4-methoxyphenyl)-2-[2-(1,4-oxazepan-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
2-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N,N-bis(prop-2-en-1-yl)acetamide