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N-[5-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)-2-methylphenyl]-2-ethylbutanamide
1-[(2-chlorophenyl)methyl]-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-(2-methyl-1H-imidazol-1-yl)-1-[5-(propan-2-yl)-1,3-oxazole-4-carbonyl]piperidine-4-carboxylic acid
4-({4-[(3,4-difluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-2-methoxyphenol
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-2-propoxypropan-1-one
(4aR,7aS)-1-(2-methylpropyl)-4-(2-propyl-1,3-thiazole-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(3-fluorophenyl)methyl]-4-{[4-(pyridin-3-yl)phenyl]methyl}piperazine
2-[3-({[(4-tert-butyl-1,3-thiazol-2-yl)methyl]amino}methyl)-2-methyl-1H-indol-1-yl]acetamide
1-[benzyl(methyl)amino]-3-{4-[(2,2-dimethylmorpholin-4-yl)methyl]phenoxy}propan-2-ol
4-[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
3-hydroxy-5-(5-methyl-1H-indol-3-yl)benzoic acid
3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-(1-methylpiperidin-4-yl)urea
N-methyl-2-[4-(3-methylphenyl)piperazin-1-yl]-N-(pyrazin-2-ylmethyl)acetamide
1-(3-{9-methoxy-7-[4-(methylsulfanyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl}phenyl)imidazolidin-2-one
ethyl 4-[4-(2,4-dioxoimidazolidin-1-yl)benzamido]piperidine-1-carboxylate
N-({4-hydroxy-1-[2-(piperidin-1-yl)acetyl]azepan-4-yl}methyl)pyridine-3-carboxamide
(1R,2S,3S,4R,5S)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}tricyclo[3.2.1.02,4]octane-3-carboxamide
(2R,3R)-3-[4-(2,4-difluorophenyl)-1H-1,2,3-triazol-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-N-(pentan-3-yl)piperidine-4-carboxamide
7-(oxan-4-yl)-2-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
(2S,3S)-2-amino-3-methyl-1-[7-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]pentan-1-one
3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}-N-(2-fluorophenyl)piperidine-1-carboxamide
4-amino-2-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]pyrimidine-5-carbonitrile
(2S,4S)-4-[4-(3-cyanobenzenesulfonamidomethyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
N-methyl-3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]propanamide
1-cyclohexyl-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]piperidine-3-carboxamide
N-[(3S,4R)-4-(4-methylphenyl)-1-[3-(pyridin-3-yl)propanoyl]pyrrolidin-3-yl]cyclopropanecarboxamide
2-[(4aS,8aR)-1-(2-aminoethyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]-4,6-dimethylpyridine-3-carbonitrile
3-(oxolan-3-yl)-5-(2,4,5-trimethylphenyl)-1,2,4-oxadiazole
1-{4-[(5-hydroxy-4,4-dimethylpentyl)amino]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
2-[3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)propanamido]acetic acid
2-chloro-4-{[3-(2-hydroxyethyl)-4-(propan-2-yl)piperazin-1-yl]methyl}phenol
dimethyl(2-{3-[3-(3-methylpyrazin-2-yl)phenyl]-1H-pyrazol-1-yl}ethyl)amine
(3R,4R)-1-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]-3,4-dimethylpyrrolidin-3-ol
2-(2-methyl-1H-1,3-benzodiazol-1-yl)-N-[1-phenyl-3-(propan-2-yl)-1H-pyrazol-5-yl]acetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
N-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)pyridin-3-yl]-2-methylpropanamide
N-[3-(2-aminopyridin-4-yl)phenyl]acetamide
N-{1-azabicyclo[2.2.2]octan-3-yl}-5-{[(5-chloropyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
ethyl 2-(8-methylquinolin-5-yl)pyridine-3-carboxylate
N-{1-[(2R)-2-amino-2-phenylacetyl]piperidin-4-yl}methanesulfonamide
2-(2,5-dimethoxyphenyl)-1H-1,3-benzodiazole-5-carbonitrile
(2S,4R)-4-(cycloheptylamino)-N-[2-(2-fluorophenyl)ethyl]-1-(propan-2-yl)pyrrolidine-2-carboxamide
3-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)-N-{[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}benzamide
4-{[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]amino}-5-methyl-N-(propan-2-yl)thieno[2,3-d]pyrimidine-6-carboxamide
4-[(2-hydroxyethyl)sulfanyl]-N-methyl-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}benzamide
N-cyclopentyl-N-({4-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)methanesulfonamide
3-(azocan-1-yl)-N-[(3,4-dimethoxyphenyl)methyl]propanamide