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4'-[3-(3-methylpiperidin-1-yl)-3-oxopropyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)pyridine-3-sulfonamide
1-ethyl-4-{[4-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-4-phenoxybutanamide
1-{[4-(2-chloro-6-methoxyphenyl)thiophen-2-yl]methyl}piperazine
N-(2H-1,3-benzodioxol-5-yl)-1-[(2-fluorophenyl)methyl]piperidin-3-amine
7-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-2-oxa-7-azaspiro[4.5]decan-8-one
1-tert-butyl-4-[3-(2-methylphenoxy)azetidine-1-carbonyl]pyrrolidin-2-one
N-(2-fluorophenyl)-2-{4-[1-(pyridin-2-yl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}acetamide
1-ethyl-4-[3-(2-fluorophenoxy)azetidine-1-carbonyl]pyrrolidin-2-one
N-(1-{7-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylfuran-3-carboxamide
1-[1-(1-benzofuran-5-ylmethyl)piperidin-4-yl]piperidin-4-ol
1-[(3,5-dimethylphenyl)methyl]-4-[2-(4-hydroxyphenyl)acetyl]piperazin-2-one
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-5-ethyl-1,3,4-oxadiazol-2-amine
2-methyl-5-(4-{[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
3,5-dichloro-4-({2-[2-(1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)pyridine
N-[(4-phenylmorpholin-2-yl)methyl]-3-(1H-pyrazol-1-yl)benzamide
2-{4-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]phenyl}-N,N-dimethylacetamide
{4-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-7-yl)methyl]-1,4-oxazepan-6-yl}methanol
3-chloro-4-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)phenol
2-methoxy-1-{4-[3-(piperidin-3-yl)benzoyl]-1,4-diazepan-1-yl}ethan-1-one
methyl (2R,4S)-4-hydroxy-1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidine-2-carboxylate
[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]({[2-(piperidin-1-yl)-2,3-dihydro-1H-inden-2-yl]methyl})amine
6-(azepan-1-yl)-N-[2-(pyridin-3-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
4-benzyl-3-ethyl-1-(6-oxo-1,6-dihydropyridine-3-carbonyl)-1,4-diazepan-5-one
1-{2-[1-(4-methyl-2-phenylpyrimidine-5-carbonyl)piperidin-4-yl]ethyl}pyrrolidin-2-one
2-{[(1-propyl-1H-imidazol-2-yl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
5-chloro-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
1-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}cyclopropan-1-amine
N-[(2S)-1-hydroxy-3-(1H-indol-3-yl)propan-2-yl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
(1S,5R)-6-(pyridin-2-ylmethyl)-3-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl({[1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazol-5-yl]methyl})[2-(pyridin-2-yl)ethyl]amine
1-(azepan-1-yl)-3-[3-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol
(1S,5R)-6-(cyclobutylmethyl)-3-(6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-4-(piperidin-3-yl)benzamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N,6-dimethyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
2-acetyl-N-{[1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]methyl}benzamide
1-(1H-imidazol-4-ylmethyl)-4-(2-methoxyphenyl)piperidine
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-[4-(pyrrolidin-1-yl)benzoyl]piperidine
7-(cyclopropylmethyl)-2-[3-(pyridin-3-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
9-[(4-methyl-1H-imidazol-2-yl)methyl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
ethyl 2-[3-(pyridin-2-yl)azetidin-1-yl]-1,3-oxazole-4-carboxylate
1-[2-(3,4-dimethoxyphenyl)ethyl]-1-methyl-3-(3-oxo-1,3-dihydro-2-benzofuran-5-yl)urea
1-methyl-4-{2-[3-(2-methylpropyl)morpholin-4-yl]-2-oxoethyl}-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-2-(pyridin-3-yl)pyridine
(3S,4S)-4-(dimethylamino)-1-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]pyrrolidin-3-ol
1-{[5-(azetidin-1-ylmethyl)-2-methoxyphenyl]methyl}-1H-pyrazole
2-{5-[1-hydroxy-3-(methylsulfanyl)propyl]-3-methyl-1H-1,2,4-triazol-1-yl}benzoic acid
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-2,6-dimethylquinoline-4-carboxamide
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-5-methyl-1,3,4-oxadiazol-2-amine