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N2-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-N4,N4,5-trimethylpyrimidine-2,4-diamine
ethyl 1-(butylcarbamoyl)-3-[(2,4-difluorophenyl)methyl]piperidine-3-carboxylate
(3aR,6aR)-N-[(2-hydroxyadamantan-2-yl)methyl]-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-3-(3-fluorophenyl)-N-methyl-1H-pyrazole-4-carboxamide
[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl](methyl)[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
2-(1-methyl-1H-pyrrol-2-yl)-2-oxo-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
N'-(2,5-dimethylphenyl)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]propanediamide
(benzylsulfamoyl)[2-(4H-1,2,4-triazol-4-yl)ethyl]amine
3-{5-[(5-cyano-1-methyl-1H-pyrrol-3-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-cyclopropylpropanamide
3-(2-methoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,4S)-1-(5-propyl-1,3,4-oxadiazole-2-carbonyl)-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
2-[benzyl({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amino]ethan-1-ol
2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}acetamide
3-(3-fluorophenyl)-5-[(propan-2-yl)sulfamoyl]benzoic acid
1-(1-carbamoylcyclopropanecarbonyl)-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(pyridin-4-yl)ethan-1-one
N-cyclopropyl-4-methoxy-3-[(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)oxy]benzamide
2-(3-{[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]methyl}phenyl)ethan-1-amine
N-methyl-2,4-dioxo-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-[(2,4-difluoro-3-methoxyphenyl)methyl]-octahydropyrrolo[1,2-a]piperazine
2-{[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]amino}pyridine-3-carbonitrile
1-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
3-butyl-4-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-1-methylpiperazin-2-one
8-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
N-[7-methoxy-2-oxo-4-(6-phenoxypyridin-3-yl)-1,2,3,4-tetrahydroquinolin-6-yl]acetamide
3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}-N-(2-phenylethyl)piperidine-1-carboxamide
8-benzyl-1-ethyl-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(ethanesulfonyl)ethyl]-2,5,6-trimethylpyrimidin-4-amine
1-{6-methylthieno[2,3-d]pyrimidin-4-yl}-N-(3-phenoxypropyl)piperidin-4-amine
dimethyl({4-[1-(1-propyl-1H-pyrazole-5-carbonyl)piperidin-2-yl]phenyl}methyl)amine
2-[4-(hydroxymethyl)-4-(2-phenoxyethyl)piperidin-1-yl]pyridine-3-carbonitrile
N-(1-{1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxybenzamide
2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
2-ethyl-5-[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]pyrimidine
4-methoxy-6-[4-(2-phenylethyl)piperazin-1-yl]pyrimidine
N-[4-(1H-pyrazol-1-yl)butan-2-yl]-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
[(3S,5R)-1-(4-chloro-2-fluorobenzoyl)-5-[(dimethylamino)methyl]piperidin-3-yl]methanol
N-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]-1-methyl-1H-indole-6-carboxamide
6-[4-({2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}amino)piperidin-1-yl]pyridine-3-carbonitrile
3-ethoxy-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
(3S,9aR)-3-ethyl-8-[(4-phenyl-1,3-thiazol-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(3aS,7aR)-5-methyl-2-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
ethyl 2-[2-({1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazol-4-yl}formamido)ethyl]-1,3-thiazole-4-carboxylate
1-cyclopentyl-4-oxo-5-(piperidine-1-carbonyl)-N-[1-(thiophen-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-4-[(2-hydroxyethyl)sulfanyl]benzamide
2-{4-[2-(cyclohex-1-en-1-yl)ethyl]piperazin-1-yl}pyrimidine
4-benzamido-N-(1-butyl-3-methyl-1H-pyrazol-5-yl)piperidine-1-carboxamide
3-fluoro-N,N-bis(2-methoxyethyl)-7-methylimidazo[1,2-a]pyridine-2-carboxamide
3-[1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]pyridine
1-ethyl-5-{methyl[(5-phenyl-1,2-oxazol-3-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid