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1-({6-[3-(benzyloxy)phenyl]pyridin-3-yl}methyl)-4-methylpiperazine
N-[2-(4-methylbenzenesulfonyl)ethyl]-6-(1-methylpiperidin-4-yl)pyrimidin-4-amine
2-{4-[6-amino-5-cyano-4-(3-fluorophenyl)pyridin-2-yl]-3,5-dimethyl-1H-pyrazol-1-yl}acetic acid
3-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}pyridine-2-carbonitrile
5-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carbonyl]-2-(thiophen-2-yl)pyrimidin-4-ol
5-acetyl-N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-2,4-dimethyl-1H-pyrrole-3-carboxamide
N-benzyl-N-(cyclohexylmethyl)-2-(2,6-dioxo-1,3-diazinan-1-yl)acetamide
1-[6-(3-chloro-4-fluorophenyl)pyridin-2-yl]ethan-1-ol
N-[3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]-4-phenyl-1,2,3,6-tetrahydropyridine-1-carboxamide
N-[(3-hydroxypyrrolidin-3-yl)methyl]-2-(phenylamino)pyrimidine-5-carboxamide
N,N-diethyl-1-{1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(methoxymethyl)-1H-pyrazole-4-carbonyl}pyrrolidin-3-amine
({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)[1-(pyridin-3-yl)propan-2-yl]amine
3-[(3R,4S)-1-(5-ethylthiophene-3-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
2-(2-methylphenyl)-N-[2-(propan-2-yl)-1H-1,3-benzodiazol-5-yl]pyrrolidine-1-carboxamide
1-(azocan-1-yl)-3-[2-methoxy-4-({[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol
6-[5-(trifluoromethyl)-1,2,3,4-tetrahydroisoquinoline-2-carbonyl]piperazin-2-one
3-(2-chlorophenyl)-N-methyl-N-[(3-methylpyridin-4-yl)methyl]-3-phenylpropanamide
5-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}-2,3-dihydro-1H-pyrazol-3-one
5-[4-(3-methoxyphenyl)piperazine-1-carbonyl]-2-methylpyrimidine
2-{3-[1-methyl-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}pyridine
(1S,5R)-3-(3-phenylpropyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(2,2-dimethylpropanoyl)-N-(5-methyl-1,3,4-thiadiazol-2-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
(1R,5R)-6-[(5-methoxy-1,3,4-thiadiazol-2-yl)methyl]-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
(1S,5R)-3-benzyl-6-(dimethyl-1,3-thiazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-cyclohexyl-4-(2-propoxyacetyl)-1,4-diazepane-6-carboxylic acid
1-(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinolin-8-yl)-3-methyl-3-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)urea
1-(2-methylpropanoyl)-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
4-(hydroxymethyl)-1-(4-phenyl-1H-imidazole-5-carbonyl)piperidin-4-ol
methyl 4-[6-amino-5-cyano-4-(oxolan-3-yl)pyridin-2-yl]-5-methylfuran-2-carboxylate
5-methyl-1-(pyridin-2-yl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]-1H-pyrazole-4-carboxamide
N-(furan-3-ylmethyl)-N-methyl-2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carboxamide
N-[2-(morpholin-4-ylmethyl)phenyl]-4-(pyridin-3-yl)piperazine-1-carboxamide
1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
1-(cyclopropylmethyl)-5-[3-(3-methoxyphenyl)propanoyl]-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[3-(3-phenylpropanamido)phenyl]-4-(pyrrolidin-1-yl)butanamide
1-{2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}ethan-1-one
6-(pyrrolidin-1-ylmethyl)-4-[4-(trifluoromethyl)pyridin-2-yl]-1,4-oxazepan-6-ol
2-{1-[1-(3,4-dihydro-2H-1-benzopyran-2-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-methylpropanamide
(1S,4S)-5-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-2-[2-(methylsulfanyl)phenyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
butyl({[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})methylamine
3-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(2-methoxyethyl)-1-(6-methoxypyridin-3-yl)urea
N-methyl-N-(2-phenylethyl)-1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-amine
3-[(2-fluorophenyl)formamido]-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]propanamide
3-({[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]amino}methyl)pyrrolidin-3-ol
1-[(5-methylfuran-2-yl)methyl]-N3-(naphthalen-1-ylmethyl)-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pyridine-2-carboxamide
3-[(3R,4S)-4-(dimethylamino)-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidin-3-yl]propanoic acid
7-cyclopropanecarbonyl-N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[2-(2-fluorophenyl)-2-hydroxyethyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide