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2-methyl-6-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-4-yl}pyrimidin-4-ol
1-(6-methyl-2-phenylpyrimidin-4-yl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]piperidin-4-amine
N-cyclobutyl-7-(cyclopropylmethyl)-6-(2,5-dimethylfuran-3-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
[2-(dimethyl-1,3-thiazol-2-yl)ethyl][1-(1H-pyrazol-1-yl)propan-2-yl]amine
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2,2-dimethylpropan-1-one
(4-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}-1,4-oxazepan-6-yl)methanol
5-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-3,4-dihydropyrimidin-4-one
4-[(3S,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]benzonitrile
5-[2-(methylsulfanyl)ethyl]-4-phenyl-1-(prop-2-en-1-yl)-1H-imidazole
N,N-diethyl-3-({[(3-methyl-1H-indol-2-yl)methyl]amino}methyl)pyridin-2-amine
(3aS,6aS)-2-ethyl-1-oxo-5-[(1-phenyl-1H-pyrazol-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-tert-butyl-4-[3-(2-fluorophenoxy)azetidine-1-carbonyl]pyrrolidin-2-one
N-[2-(dimethylamino)ethyl]-N-methyl-3-{[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-4-yl]oxy}benzamide
3-[(2-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-1H-imidazol-1-yl)methyl]pyridine
1-ethyl-2-({3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)-1H-1,3-benzodiazole
N-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-1-(pyrimidin-2-yl)piperidin-4-amine
5-{[8-(cyclopropylmethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
2-amino-8-(6-phenoxypyridin-3-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
(3aS,6aS)-2-(2-methoxy-5-methylbenzenesulfonyl)-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
(2R,3R,6R)-5-(5-methoxyfuran-2-carbonyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-[1-(2,8-dimethylquinoline-4-carbonyl)-3-oxopiperazin-2-yl]-N-methylacetamide
3-phenyl-1-[1-(3,6,7-trimethyl-1-benzofuran-2-carbonyl)piperidin-4-yl]propan-1-ol
2-(3-cyclopropyl-1H-1,2,4-triazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinoline
N-methyl-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine
1-{1-[4-(1-benzofuran-2-yl)pyrimidin-2-yl]-5-cyclopropyl-1H-pyrazole-4-carbonyl}-N,N-dimethylpyrrolidin-3-amine
N-[1-(2-chlorophenyl)ethyl]-1-cyclopentyl-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
N-methyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-2,3-dihydro-1H-inden-2-amine
3-(2,5-dimethylphenyl)-4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}-1H-pyrazole
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}formamido)acetic acid
(3aR,6aR)-2-[(1-propyl-1H-imidazol-2-yl)methyl]-5-(thiophen-3-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
(3S,4R)-1-[(3-fluoro-5-methylphenyl)methyl]-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-[(4-methylphenyl)methyl]-1,3-oxazole-4-carboxamide
N-(3-fluoro-4-methylphenyl)-2-{[1-(thiophen-3-yl)propan-2-yl]amino}acetamide
4-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-1,2-dihydroquinazolin-2-one
2-(5-methyl-1H-pyrazol-1-yl)-1-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
3-(5-fluoro-2-methoxyphenyl)-1-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-1-(pyridin-3-ylmethyl)urea
N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]-3-methoxypyridine-2-carboxamide
dimethyl({[(3S,4R)-4-(propan-2-yl)-1-(pyridine-4-carbonyl)pyrrolidin-3-yl]sulfamoyl})amine
3-{1-methyl-4-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]-1H-pyrazolo[3,4-d]pyrimidin-6-yl}pyridine
4-(3-ethoxypropanoyl)-1-(2-phenylphenyl)piperazin-2-one
4,6-dimethyl-2-[9-oxo-8-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-3-carbonitrile
2-methyl-6-[(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)methyl]pyridine
(1R,5S,8S)-8-methoxy-3-[(1-propyl-1H-imidazol-2-yl)methyl]-3-azabicyclo[3.2.1]octane
3-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-4-phenyl-1H-pyrazol-5-amine
2-methyl-9-[(5-phenylthiophen-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-3-(1H-pyrazol-1-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]benzamide
1-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-N-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
4-(1H-imidazol-1-yl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)benzamide