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(3S,4S)-3-hydroxy-4-(piperidin-1-yl)-N-[3-(1H-pyrazol-5-yl)phenyl]pyrrolidine-1-carboxamide
9-(5-fluoro-2-methoxybenzoyl)-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-ethyl-N-(furan-3-ylmethyl)-N-methyl-5-(4-methylpiperidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N3-butyl-1-cyclohexyl-N5-[2-methyl-2-(morpholin-4-yl)propyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-({2-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-2,6-dimethylpyridine-4-carboxamide
3-(benzyloxy)-1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine
2-(1H-1,3-benzodiazol-1-yl)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]propan-1-one
4-(1,2,4-oxadiazol-3-yl)-1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidine
2-[(benzylsulfamoyl)amino]benzamide
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
4-({3-azaspiro[5.5]undecan-9-yl}amino)-N,N-dimethylbutanamide
5-[1-(1,4-dioxan-2-ylmethyl)-1H-1,2,3-triazol-4-yl]-2-(2-methoxyphenyl)pyrimidine
4-methyl-2-(pyridin-3-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]pyrimidine-5-carboxamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-1-(2-fluorophenyl)-N-methylcyclopropane-1-carboxamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]morpholine-4-sulfonamide
2-ethyl-8-[(3-methylquinoxalin-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
1-(3-fluorobenzoyl)-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-(1H-1,3-benzodiazol-1-yl)-1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidine-4-carboxylic acid
(3aR,6aR)-2-[2-(1-methyl-1H-indol-3-yl)acetyl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(6-methoxyhexanoyl)-1-(4-methoxyphenyl)piperazin-2-one
4-cyclopentyl-N-methyl-N-[(1-methylpyrrolidin-2-yl)methyl]pyrimidin-2-amine
7-methyl-2-(2-phenylquinazolin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
1,6-dimethyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(2-{[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
2-{[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
2-[5-(4-chloro-2-methylphenoxymethyl)-3-cyclopropyl-1H-1,2,4-triazol-1-yl]acetic acid
N-cyclopentyl-4-(4-{[2-(pyridin-3-yloxy)ethyl]amino}piperidin-1-yl)benzamide
5-chloro-2-[3-(hydroxymethyl)-3-propylpiperidine-1-carbonyl]phenol
3-(2-amino-1,3-thiazol-4-yl)-N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)propanamide
1-{2-[2-(1H-imidazol-1-yl)ethyl]piperidin-1-yl}-4-phenylbutan-1-one
1-[3-(cyclopentyloxy)phenyl]-3-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}urea
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-N-{[7-(methylsulfanyl)-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}thiophene-2-carboxamide
1-[(1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methyl]pyrrolidin-2-one
N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-(2-phenyl-1,3-thiazol-4-yl)acetamide
2-{1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperidin-2-yl}pyridine
4-(4-methyl-4H-1,2,4-triazol-3-yl)-1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidine
2-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-1,2,3,4-tetrahydroisoquinoline
3-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}-7-methoxy-1,2-dihydroquinolin-2-one
N-[(4-fluorophenyl)methyl]-2-(methylamino)-N-(1-phenylethyl)acetamide
6-[4-(3-methylpyridin-2-yl)piperazine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
7-methoxy-3-{[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperazin-1-yl]methyl}-1,2-dihydroquinolin-2-one
(1S,5R)-3-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-(3-propyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
4-chloro-2-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenol
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-(thiophen-2-ylmethyl)-1,4-diazepane
1-{1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]azetidin-3-yl}-3,5-dimethyl-1H-pyrazole
N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[({[3-(prop-2-en-1-yl)-4-(propan-2-yloxy)phenyl]methyl}amino)methyl]-3,4-dihydroquinazolin-4-one
3-(2H-1,3-benzodioxol-5-yl)-1-[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]propan-1-one