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8-fluoro-2-{[(2-methoxyethyl)[(2-methylphenyl)methyl]amino]methyl}quinolin-4-ol
4-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]oxane-4-carbonitrile
4-(2-methoxyphenoxy)-1-(5-methylthiophene-3-carbonyl)piperidine
[5-(1-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-1H-1,2,3-triazol-4-yl)furan-2-yl]methanol
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-methyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)acetamide
6-methoxy-1-[3-(4-methylphenoxymethyl)piperidin-1-yl]hexan-1-one
2-{4-[3-(propan-2-yloxy)phenyl]phenyl}-1,3,4-oxadiazole
N-[(3-hydroxyphenyl)methyl]-N,3,4,7-tetramethyl-1H-indole-2-carboxamide
4-[5-(7-{[ethyl(pyridin-4-ylmethyl)amino]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)furan-2-yl]-2-methylbut-3-yn-2-ol
1-(5-chloropyridin-2-yl)-4-(2,6-dimethoxypyridine-3-carbonyl)piperazine
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]cyclobutanecarboxamide
N-[(2S)-3-(1H-imidazol-4-yl)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-1-oxopropan-2-yl]acetamide
1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)-4-methoxypiperidine
4-{2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}-1H-indole
1-(3-fluoropyridin-2-yl)-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylic acid
1-[6-hydroxy-4-(pyrazin-2-yl)-1,4-diazepan-1-yl]-2-[(2-methoxyethyl)(methyl)amino]ethan-1-one
2,3,6-trimethyl-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]quinoline-4-carboxamide
[1-(1-{1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}piperidin-4-yl)piperidin-3-yl]methanol
1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-2-[2-(pyrrolidin-1-yl)ethyl]piperidine
8-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-dioxa-8-azaspiro[4.5]decan-2-one
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]pyrazolo[1,5-a]pyridine-3-carboxamide
4-{[5-(1-benzyl-5-methyl-1H-1,2,3-triazol-4-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-methylpiperidine
(2R,3R,6R)-5-(4-ethylbenzoyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(2-methoxyethyl)-2-{[2-(2-methoxyphenyl)pyrrolidin-1-yl]methyl}-1H-imidazole
4-{4-[(4-acetylpiperazin-1-yl)methyl]-2-methylphenoxy}thiane-4-carboxylic acid
N-{[1-(dimethylamino)cyclohexyl]methyl}-2-(3-fluorophenyl)-2-hydroxyacetamide
(3R,5R)-5-(morpholine-4-carbonyl)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carboxamide
(1R,5R)-6-(2-methoxyethyl)-3-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]-3,6-diazabicyclo[3.2.2]nonane
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
2-tert-butyl-4-hydroxy-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)pyrimidine-5-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-3-yl]piperazine
3-{[1-(furan-2-ylmethyl)piperidin-3-yl]formamido}-N-(2-methoxyphenyl)propanamide
6-(6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-5,6,7,8-tetrahydro-1,6-naphthyridine
2-(2-chloro-4-fluorophenoxymethyl)-N-methyl-N-(1H-pyrazol-3-ylmethyl)-1,3-oxazole-4-carboxamide
(3R,4S)-1-[(5-fluoro-2-methoxyphenyl)methyl]-3,4-dimethylpiperidin-4-ol
N-{3-[4-(trifluoromethyl)pyrimidin-2-yl]phenyl}acetamide
N-(4-{[2-(2H-1,3-benzodioxol-5-yl)-8-methyl-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}phenyl)acetamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(2-fluorophenyl)-3-phenylpropanamide
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
1-{2-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(1-{[5-(2-chlorophenyl)furan-2-yl]methyl}piperidin-3-yl)methyl]thiophene-2-carboxamide
methyl 5-[6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[(2-phenyl-1,3-thiazol-4-yl)methyl]amine
1-{1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}-N,N-diethylpiperidine-3-carboxamide
methyl (2R,4S)-1-(2,2-diphenylethyl)-4-hydroxypiperidine-2-carboxylate
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-N'-(2,3-dimethylphenyl)-N-methylpropanediamide
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-3-[(oxolan-2-ylmethyl)sulfamoyl]benzamide
1-{5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carbonyl}azocane
N-cyclopentyl-N-(3-phenylprop-2-yn-1-yl)-3-(1H-pyrazol-1-yl)butanamide
1-ethyl-N-[2-(4-fluorobenzenesulfonyl)ethyl]-6-oxopiperidine-3-carboxamide