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(1S,5R)-3-(5-methyl-1,3-benzoxazol-2-yl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(2,5-dioxoimidazolidin-1-yl)-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]acetamide
4-(6-chloro-2H-chromen-3-yl)-3-methyl-1-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[(3R,4S)-1-(oxan-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
methyl[(5-methyl-1H-pyrazol-3-yl)methyl]{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
1-benzyl-4-(2,3-dihydro-1H-inden-2-yl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
5-(6-aminopyridin-3-yl)-4-(4-methylphenyl)-N-[1-(pyrimidin-4-yl)ethyl]pyrimidin-2-amine
1-(3-methoxybenzoyl)-4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperazine
4-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}imidazolidin-2-one
4-(4-fluoro-2-methylphenyl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
1-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-4-(1H-pyrazol-1-yl)butan-1-one
3-(4-hydroxyphenyl)-N-[3-(1H-indazol-1-yl)propyl]-1H-pyrazole-5-carboxamide
ethyl 3-[(3-chlorophenyl)methyl]-1-(pyridin-3-ylmethyl)piperidine-3-carboxylate
3-hydroxy-3-({[(3-methylphenyl)methyl]amino}methyl)-1-(2-phenylethyl)piperidin-2-one
2-[(3,5-difluorophenyl)methyl]-8-[(2E)-2-methylbut-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
(3aR,6aR)-2-cyclopropanecarbonyl-5-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propan-1-ol
5-(2,6-dimethylphenoxymethyl)-N-methyl-N-(pyrazin-2-ylmethyl)-1,2-oxazole-3-carboxamide
2-{4-[(6-ethyl-2-methylquinolin-4-yl)methyl]piperazin-1-yl}ethan-1-ol
(1S,5R)-3-benzyl-6-(1H-indole-6-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-{4-[benzyl(methyl)sulfamoyl]morpholin-3-yl}acetamide
N-[(3R,4S)-1-acetyl-4-cyclopropylpyrrolidin-3-yl]-2-methoxy-5-methylbenzene-1-sulfonamide
5-methyl-1-(3-methylphenyl)-4-[4-(trifluoromethyl)benzoyl]piperazin-2-one
[2-(2-chloro-4-fluorophenyl)pyridin-4-yl]methanol
N-[3-(3-methoxyphenyl)phenyl]-1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidine-2-carboxamide
7-(2-cyclohexylethyl)-2-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-2,7-diazaspiro[4.5]decane
N-(3-{1-[(3-methylphenyl)methyl]-1H-1,2,4-triazol-5-yl}propyl)acetamide
N,1,6-trimethyl-4-oxo-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1,4-dihydroquinoline-3-carboxamide
4,6-dimethyl-2-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
1-(4-ethylpiperazin-1-yl)-3-[3-({[2-(2-fluorophenyl)ethyl]amino}methyl)phenoxy]propan-2-ol
8-[1-(4-phenoxyphenyl)-1H-1,2,3,4-tetrazol-5-yl]-1-oxa-8-azaspiro[4.5]decane
1-{1-[1-(2,5-dimethylphenyl)-1H-1,2,4-triazol-5-yl]ethyl}-4-methylpiperazine
N-cyclopropyl-1-{1-[(2,5-dimethoxyphenyl)methyl]piperidin-4-yl}piperidine-4-carboxamide
2-ethoxy-1-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
5-{4-[(3-chlorophenyl)methyl]piperazine-1-carbonyl}-1-cyclopentylpiperidin-2-one
2-(1H-1,3-benzodiazol-1-yl)-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]propanamide
2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
6-tert-butyl-3-[2-(4-hydroxypiperidin-1-yl)ethyl]-3H,4H-thieno[3,2-d]pyrimidin-4-one
2-[(3-{[3-(pyridin-3-yloxy)propyl]carbamoyl}phenyl)amino]acetic acid
N-(2-methoxyethyl)-5-[2-(trifluoromethoxy)phenyl]furan-2-carboxamide
2-[2-(azocan-1-yl)acetamido]-N-(propan-2-yl)acetamide
2-[(2E)-3-phenylprop-2-en-1-yl]-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
1-(5-chloropyridin-2-yl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
1-[2-amino-7-methyl-4-(3-methylphenyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-4-(1H-pyrazol-4-yl)butan-1-one
N-(1-methyl-1H-pyrazol-4-yl)-3-(thiophene-2-carbonyl)piperidine-1-carboxamide
1-methyl-3-{1-[(2E)-2-methylbut-2-en-1-yl]piperidin-3-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[1-(1H-imidazol-4-ylmethyl)piperidin-3-yl]methyl}-2-(methylamino)pyridine-3-carboxamide
N-cyclopropyl-1-[1-(2-methyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
4-(3-fluorophenyl)-N-{[4-(oxolan-2-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)benzamide
1-(5-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}-2-methoxyphenoxy)-3-(piperidin-1-yl)propan-2-ol