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3-(5-chloro-2-methoxybenzoyl)-3,9-diazaspiro[5.6]dodecan-10-one
N-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)methyl]-2-(2,3,6-trimethylphenoxy)acetamide
1-ethyl-3-[(3-methoxyphenyl)methyl]-8-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-(3-phenylpropyl)piperidin-3-amine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-2-(diethylamino)-N-methylacetamide
4-(6-cyclopropylpyrimidin-4-yl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
7-[3-(4-methylphenyl)-3-phenylpropanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,4-dimethyl-1,2,5-oxadiazole-3-carboxamide
1'-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
6-{[3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,2-oxazol-5-yl]methoxy}quinoline
N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-2-(4-phenylpiperidin-1-yl)acetamide
3-[2-(4-propanoylphenoxy)acetyl]-3,9-diazaspiro[5.6]dodecan-10-one
N-ethyl-2-(2-fluorophenoxymethyl)-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1,3-oxazole-4-carboxamide
4-ethyl-1-{[4-(methylsulfanyl)phenyl]methyl}-1,4-diazepan-5-one
methyl[(4-methyl-1H-imidazol-5-yl)methyl]{[2-(trifluoromethyl)phenyl]methyl}amine
N-[2-(1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1H-imidazol-4-yl)ethyl]acetamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-{[(1r,4r)-4-hydroxycyclohexyl]amino}pyridine-3-carboxamide
(3S)-3-[5-(2-ethyl-4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]azepan-2-one
N-(pyridin-2-ylmethyl)-5-[(2S)-pyrrolidine-2-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-(1,3-dihydroxypropan-2-yl)-5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole-3-carboxamide
N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-methylpiperidine-3-carboxamide
ethyl 2-{[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxylate
1-ethyl-3-(pyridin-2-ylmethyl)-8-(thian-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(3-hydroxypropyl)-5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
4-(cyclopropylmethyl)-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-3-(propan-2-yl)-1,4-diazepan-5-one
{9-[(1-methyl-1H-imidazol-5-yl)methyl]-3-(1,3-thiazol-4-ylmethyl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
N-{[3-(2H-1,3-benzodioxol-5-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
(2S,4R)-4-{[(3,4-difluorophenyl)methyl]amino}-1-(2,2-diphenylethyl)-N-methylpyrrolidine-2-carboxamide
4-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}piperazine-1-sulfonamide
[(2E)-3-(furan-2-yl)prop-2-en-1-yl](methyl)[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amine
4-methoxy-N-[4-(4-{[2,2,2-trifluoro-1-(furan-2-yl)ethyl]amino}piperidin-1-yl)phenyl]benzamide
4-chloro-N-(3-methoxypropyl)-1,3-dimethyl-N-[(4-methylphenyl)methyl]-1H-pyrazole-5-carboxamide
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
1-(2-methoxyphenyl)-3-(propan-2-yl)-5-[2-(1H-pyrazol-1-yl)ethyl]-1H-1,2,4-triazole
1-[1-(2-fluoro-4-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
2-cyclopropyl-N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]quinoline-4-carboxamide
1-(cyclohex-3-ene-1-carbonyl)-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
7-[3-(2-chlorophenyl)-5-methyl-1,2-oxazole-4-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
(3R,4S)-4-(5-methylfuran-2-yl)-1-(2-propyl-1,3-thiazole-4-carbonyl)pyrrolidin-3-amine
1-{4-[(4aR,8aS)-1-(quinoxaline-6-carbonyl)-decahydro-1,6-naphthyridine-6-carbonyl]thiophen-2-yl}ethan-1-one
4-(propan-2-yl)-N-[(2,4,5-trifluorophenyl)methyl]pyrimidin-2-amine
8-(3,3-dimethylbutanoyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-(2-{1-[3-(4-hydroxyphenyl)benzoyl]piperidin-2-yl}ethyl)acetamide
1-cyclohexyl-4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
1-{1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-3-yl}pyrrolidin-2-one
5-[2-(furan-2-yl)azepane-1-carbonyl]pyrazin-2-ol
1-{1-[3-(4-fluorophenyl)benzoyl]piperidin-4-yl}pyrrolidin-2-one
7-fluoro-2-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}quinoline-4-carboxamide
(3R,5S)-N3-[(1-ethyl-1H-imidazol-5-yl)methyl]-N5-(6-methylpyridin-3-yl)piperidine-3,5-dicarboxamide
N-[4-(3-fluorophenyl)phenyl]-1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidine-3-carboxamide