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4-(1H-pyrazol-4-yl)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butan-1-one
N,N-dimethyl-5-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
8-(2-ethoxybenzoyl)-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
(3R,9aR)-3-[(benzylsulfanyl)methyl]-8-(3,5-difluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-{3-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}-2-methyl-2-phenylpropan-1-one
1-(2-aminopyrimidin-4-yl)-4-(2H-1,3-benzodioxol-5-yloxy)piperidine-4-carboxylic acid
8-fluoro-2-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,4-dihydroquinolin-4-one
(3S,4R)-4-(3-methylthiophen-2-yl)-1-(quinoline-3-carbonyl)piperidin-3-ol
4-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-3-methyl-1H-pyrazole
(3R,4R)-1-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-3,4-dimethylpyrrolidin-3-ol
2-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}quinoxaline
2-(dimethylamino)-2-(2-methylphenyl)-N-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}acetamide
1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-4-(3-methylpyridin-4-yl)-1,4-diazepane
1-(4-{[2-(1-methylpyrrolidin-2-yl)ethyl]amino}-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
N-[(4-fluorophenyl)methyl]-1-methyl-5-{[2-(4-sulfamoylphenyl)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-methylpiperidine
N-[2-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]oxolane-2-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-{3-[4-(2-fluorophenoxy)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
{3-[(3-chlorophenyl)methyl]-1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}methanol
3-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-ol
6-methyl-4-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}quinoline
N,N-dimethyl-2-[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)phenyl]acetamide
6-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-4-methyl-1H-imidazole-5-carboxamide
N-{2-[3-(ethylsulfanyl)-5-oxo-4,5-dihydro-1,2,4-triazin-6-yl]phenyl}-3-methylfuran-2-carboxamide
3-[1-(1,4-dithiepan-6-yl)piperidin-3-yl]-N-(2-fluorophenyl)propanamide
7-(propan-2-yl)-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
4-[(2-fluorophenyl)methyl]-1-[(1-methyl-1H-pyrazol-5-yl)methyl]piperidine
1-(4-chlorophenyl)-N-[(4-hydroxyazepan-4-yl)methyl]cyclobutane-1-carboxamide
(2S,4S)-4-amino-1-{2-[cyclohexyl(methyl)amino]pyridine-3-carbonyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-(2-methyl-1H-imidazol-1-yl)-1-{3-[1-(2-methylpropyl)piperidin-4-yl]pyrrolidin-1-yl}ethan-1-one
(5-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methanol
2-{[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]methyl}benzonitrile
2-(2,4-dioxoimidazolidin-1-yl)-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylacetamide
methyl({2-[2-(4-methylpiperazin-1-yl)ethoxy]phenyl}methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
1-[2-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)ethyl]azepan-2-one
3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(1,3-thiazol-2-yl)piperidine
N-[(1R,3S)-3-[(2-methoxy-6-methylphenyl)carbamoyl]cyclopentyl]pyrrolidine-1-carboxamide
2-methyl-5-{4-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
1-(2-oxo-2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)azepan-2-one
(1R,3S)-7-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-7-azaspiro[3.5]nonane-1,3-diol
4-{1-[2-(2-hydroxyethoxy)ethyl]piperidin-3-yl}benzoic acid
3-[4-(1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl)pyridin-2-yl]phenol
N-(1H-imidazol-2-ylmethyl)-5-{1-[3-(1H-pyrazol-1-yl)propyl]pyrrolidin-2-yl}thiophene-2-carboxamide
1'-(2-benzyl-1,3-benzoxazole-5-carbonyl)spiro[indene-1,4'-piperidine]
(4aR,7aS)-1-(3,5-dichloro-4-methylbenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-methylfuran-2-carboxamide
2-{2-[1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
N-{2-[5-(hydroxymethyl)-1,2,4-oxadiazol-3-yl]ethyl}-4-oxo-3,4-dihydroquinazoline-2-carboxamide
2-(4-hydroxyphenyl)-2-{4-[(4-methylphenyl)methyl]-3-oxopiperazin-1-yl}acetic acid