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3-(1H-1,2,3,4-tetrazol-1-yl)-1-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}propan-1-one
N3-ethyl-N5-[(4-fluorophenyl)methyl]-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
1-[2-(ethylsulfanyl)-1,3-benzoxazol-6-yl]-3-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]urea
2-[2-(4-fluorophenoxy)ethyl]benzene-1-sulfonamide
2-(5-{[(cyclopropylmethyl)sulfanyl]methyl}-3-methyl-1H-1,2,4-triazol-1-yl)benzoic acid
N-[2-(dimethylamino)ethyl]-N-ethyl-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carboxamide
2-(dimethyl-1,2-oxazol-4-yl)-1-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]ethan-1-one
N-(4-methoxy-2-methylphenyl)-3-{1-[(1-methyl-1H-indol-3-yl)methyl]piperidin-3-yl}propanamide
N-{3-[2-(2-chloro-4-hydroxyphenyl)-1H-imidazol-1-yl]-4-fluorophenyl}acetamide
3-[4-phenyl-5-(2,4,5-trifluorophenyl)-1H-imidazol-1-yl]propan-1-ol
2-(pyrrolidin-1-yl)-8-[4-(1H-1,2,4-triazol-1-yl)phenyl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
3-(3-methoxyphenyl)-N-[1-(pyridin-3-yl)propan-2-yl]-1H-pyrazole-4-carboxamide
4-[4-(3-chloro-4-hydroxybenzoyl)-5-methyl-2-oxopiperazin-1-yl]benzonitrile
ethyl 2-({3-[4-(methylsulfanyl)benzoyl]piperidine-1-carbonyl}amino)acetate
[(3R,4R)-1-({5-[(4-chlorophenyl)sulfanyl]furan-2-yl}methyl)-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
N-[1-(4-chlorophenyl)cyclobutyl]-6-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
2,2-dimethylpropyl 3-oxo-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxylate
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-2-(morpholin-4-yl)ethan-1-one
N-[3-({[3-(1H-imidazol-1-yl)butyl]carbamoyl}amino)phenyl]cyclopentanecarboxamide
[1-(ethylsulfanyl)propan-2-yl]({[2-(1H-imidazol-1-yl)phenyl]methyl})amine
1-(2-phenoxyethyl)-4-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]piperazine
7-methyl-3-(1-methyl-1H-indole-6-carbonyl)-3,7,11-triazaspiro[5.6]dodecan-12-one
8-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
(3S,4R)-4-(4-fluorophenyl)-1-[2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetyl]pyrrolidine-3-carboxylic acid
5-[2-(pyridin-2-yl)piperidine-1-carbonyl]-1,2-oxazol-3-ol
(benzylsulfamoyl)[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]amine
9-{[4-(methylsulfanyl)phenyl]methyl}-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(1-methyl-1H-pyrrol-2-yl)-2-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethane-1,2-dione
1-[3-(5-fluoropyridin-2-yl)phenyl]ethan-1-one
N,N-dimethyl-4-[3-(naphthalene-1-carbonyl)piperidine-1-carbonyl]piperidine-1-carboxamide
5-cyclopropanecarbonyl-1'-[(4-ethoxyphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[4-(furan-2-yl)butan-2-yl]-2-[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
N-{[1-(hydroxymethyl)cyclopentyl]methyl}-1-methanesulfonyl-N-methylpyrrolidine-2-carboxamide
(4aS,8aR)-6-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
methyl 3-{[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]carbamoyl}benzoate
1-{2-[(4-fluoropiperidin-1-yl)methyl]-5-methoxyphenoxy}-3-(4-methylpiperazin-1-yl)propan-2-ol
N-{4-[2-(4-fluorophenyl)morpholine-4-carbonyl]-3-hydroxyphenyl}acetamide
N-{1-[2-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)butanoyl]piperidin-4-yl}methanesulfonamide
N-[(2,3-difluoro-4-methylphenyl)methyl]-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-amine
1-[(2-chlorophenyl)methyl]-3-methyl-5-(oxan-4-yl)-1H,4H-pyrazolo[3,4-d]imidazole
5-{2-[4-(2-methylphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
6-ethyl-2-methyl-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}quinoline-4-carboxamide
1-[(4aR,8aR)-7-[(dimethyl-1,3-thiazol-5-yl)methyl]-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(1-methyl-1H-pyrrole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(2-fluorophenyl)-N-(1-hydroxybutan-2-yl)-N-[(5-methylthiophen-2-yl)methyl]cyclopropane-1-carboxamide
(3aR,6aR)-2-methanesulfonyl-5-[2-(3-methoxyphenyl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{1-[(3-methoxyphenyl)methyl]-4-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
N,3-dicyclopropyl-N-[(2-ethoxyphenyl)methyl]-1H-pyrazole-5-carboxamide
7-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(2-ethoxy-5-{1-[2-(pyridin-4-yl)ethyl]-1H-imidazol-2-yl}phenyl)methanol