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5-{[4-(1-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-N-(propan-2-yl)pyrimidin-2-amine
6-methyl-3-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
3-(azetidine-1-carbonyl)-N-[2-(2,5-dimethylphenyl)ethyl]benzene-1-sulfonamide
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[2-(1H-pyrazol-1-yl)ethyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
ethyl 1-{[2-(methoxycarbonyl)phenyl]carbamoyl}-4-(2-phenylethyl)piperidine-4-carboxylate
1-[(4-methoxyphenyl)methyl]-N-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-(2,5-dioxoimidazolidin-4-yl)-N-[3-(trimethyl-1H-pyrazol-1-yl)propyl]acetamide
1-[2-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-oxoethyl]pyrrolidin-2-one
N-(adamantan-1-yl)-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
N-[2-methoxy-2-(thiophen-2-yl)ethyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
N-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-4-amine
ethyl 5-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-1H-imidazole-4-carboxylate
2-{4-[5-(1H-pyrrol-2-yl)-1,2,4-oxadiazol-3-yl]phenyl}ethan-1-ol
3-{2-[3-(dimethylamino)pyrrolidin-1-yl]ethyl}-8-(2-hydroxyacetyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(dimethyl-1,2-oxazol-4-yl)propanamide
N-(1-benzylpiperidin-4-yl)-2-(2,4-dioxo-1,3-diazinan-1-yl)benzamide
3-(furan-2-yl)-3-phenyl-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}propanamide
1-(2-amino-6-methoxypyrimidin-4-yl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-1-[4-(9H-purin-6-yl)piperazin-1-yl]propan-1-one
(2R,3R)-1'-(2-aminopyrimidin-4-yl)-3-(2-methyl-1H-imidazol-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
(3E)-1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}hex-3-en-1-one
3-[3-(4-ethylpiperazin-1-yl)propyl]-8-[(2S)-2-hydroxypropanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{5-[2-(pyridin-2-yl)-1H-imidazol-1-yl]pyridin-2-yl}acetamide
N-(2-methoxyethyl)-7-[1-(methoxymethyl)cyclobutanecarbonyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(1S,5R)-6-(morpholine-4-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-[2-(methylamino)ethyl]acetamide
1,9-dimethyl-4-(2-methyl-1H-pyrrole-3-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
4-{4-[2-(2-hydroxyethyl)pyrrolidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-2-(methylamino)pyridine-4-carboxamide
3-{5-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
8-[2-(2,3-dihydro-1H-inden-5-yloxy)-2-methylpropanoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-[2-(3-methoxyphenoxy)ethyl]benzamide
7-{[ethyl(oxan-4-ylmethyl)amino]methyl}-4-methyl-2H-chromen-2-one
8-(3-cyclopropylpropanoyl)-3-{2-[methyl(2-methylpropyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3aR,6aR)-N-(1H-1,3-benzodiazol-2-ylmethyl)-2-cyclopentyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N3-cyclooctyl-4-oxo-1-(oxolan-2-ylmethyl)-N5-(pyridin-3-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
9-benzyl-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
5-({4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}methyl)-2-(methoxymethyl)pyrimidine
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
1-{4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
{[(1R,5S,6S)-3-[(3-chloro-4-fluorophenyl)methyl]-3-azabicyclo[3.1.0]hexan-6-yl]methyl}dimethylamine
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
1-(azepan-1-yl)-3-(2-methoxy-4-{[methyl(propyl)amino]methyl}phenoxy)propan-2-ol
5-{4-hydroxy-1-[(4-methylphenyl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)-1-benzofuran-2-carboxamide
(1R,3S)-3-(2-hydroxyethoxy)-7-(1H-pyrrole-2-carbonyl)-7-azaspiro[3.5]nonan-1-ol
1-{4-[2-(3,4-dimethoxyphenyl)-5-fluoro-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-(4-fluorophenyl)ethan-1-one
6-{4-[(6-chloropyridin-3-yl)methyl]piperazin-1-yl}pyrazine-2-carboxamide
2-(5-{[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyridine
2-{[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]methyl}-6-methyl-1,4-dihydroquinolin-4-one