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1-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-4-(4-fluorophenyl)butane-1,4-dione
6-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-4-yl)-2-methylpyrimidin-4-ol
2-(5-methylfuran-2-yl)-N,1-bis(propan-2-yl)-1H-1,3-benzodiazole-5-sulfonamide
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
N-[3-(5-amino-3-methyl-1-phenyl-1H-pyrazol-4-yl)phenyl]acetamide
5-tert-butyl-4-{[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]methyl}furan-2-carboxamide
methyl 2-[(6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)formamido]acetate
4-(2-methoxypyridine-4-carbonyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
4-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1λ6-thiane-1,1-dione
3-hydroxy-N-[2-(pyridin-3-yloxy)phenyl]-1-oxa-8-azaspiro[4.5]decane-8-carboxamide
(3E)-1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]hex-3-en-1-one
6-(4-{[4-(propan-2-yl)phenyl]methyl}piperazin-1-yl)-9H-purin-2-amine
N-tert-butyl-2-(2,4-dimethoxypyrimidin-5-yl)benzene-1-sulfonamide
N-[(2S)-1-methoxypropan-2-yl]-4-[methyl(1H-pyrazol-3-ylmethyl)sulfamoyl]benzamide
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
N-[(3S,7S,8aS)-3-[(4-chlorophenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,5-difluorobenzamide
2-[4-(3-methoxyphenyl)piperazine-1-carbonyl]-3,4-dihydroquinazolin-4-one
N-[3-(pyridin-2-yl)propyl]-4-(pyridin-3-yl)pyrimidin-2-amine
5-(1-acetylpiperidine-3-carbonyl)-N,N-dimethyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
1-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}-4-(pyrimidin-2-yl)-1,4-diazepane
N-[(1R,2R)-2-hydroxycyclohexyl]-5-(phenoxymethyl)-N-propyl-1H-pyrazole-3-carboxamide
4-{6-[1-(2,2-dimethylcyclopropanecarbonyl)piperidin-4-yl]-2-methylpyrimidin-4-yl}morpholine
1-(3-{5-methyl-2-[(pyridin-3-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidin-1-yl)-2-(1,3-thiazol-4-yl)ethan-1-one
1-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidin-1-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
1-{2-[(2-chloro-5-acetamidophenyl)formamido]ethyl}piperidine-3-carboxamide
(3R,4S)-1-(2,5-dimethylbenzoyl)-4-propylpyrrolidin-3-amine
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-4-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
4-(2,5-dimethoxyphenyl)-2-[({[2-(trifluoromethyl)phenyl]methyl}amino)methyl]phenol
5-tert-butyl-N-[2-(pyridin-3-yloxy)propyl]-1,3,4-oxadiazol-2-amine
(3R,5S)-5-(3-fluorophenoxymethyl)-1-[(4-hydroxyphenyl)methyl]-N-(2-methylpropyl)piperidine-3-carboxamide
7-(2-methoxyethyl)-2-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-2,7-diazaspiro[4.5]decan-6-one
1-(2-methylpyrimidin-4-yl)-4-(oxan-4-yl)-1,4-diazepan-6-ol
3-methyl-4-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-1-(2-methylpropyl)piperazin-2-one
2-(dimethylamino)-2-(2-methylphenyl)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]acetamide
N-(1-cyclopropanecarbonylpiperidin-3-yl)-2,3,6-trimethylquinoline-4-carboxamide
3-(methoxymethyl)-N-(2-{[(4-methylphenyl)methyl]sulfanyl}phenyl)pyrrolidine-1-carboxamide
({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
N-(adamantan-1-yl)-4-[(pyridin-2-ylmethyl)amino]pyridine-2-carboxamide
(1R,5R)-6-[(3-chloro-4-fluorophenyl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-[(2-methyl-1H-indol-5-yl)methyl]-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
3-methyl-1-[(4-methylphenyl)methyl]-4-(5-methylpyrazine-2-carbonyl)piperazin-2-one
3-(1-cyclooctylpiperidin-4-yl)-1-(4-ethylpiperazin-1-yl)propan-1-one
1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(2H-1,2,3,4-tetrazol-2-yl)ethan-1-one
2-(2-phenylphenyl)-4-(pyrrolidine-1-carbonyl)pyridine
2-[(3,4-difluorophenyl)methyl]-8-(3-methoxypyrazin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
N-[2-(azepan-1-yl)ethyl]-2-(4-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-4-(1H-imidazol-1-yl)butanamide
7-(cyclobutylmethyl)-2-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-butyl-5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-amine
6-(3-ethyl-4-methylpiperazin-1-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide