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1-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
4-[(4-fluorophenyl)methyl]-1-(2-methoxyacetyl)-3-(propan-2-yl)-1,4-diazepan-5-one
4-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]-1-(4-methylphenyl)butan-1-one
4-[(4-methyl-1,3-thiazol-5-yl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
5-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}-N-propylpyrimidin-2-amine
2-{5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}pyrimidin-4-amine
(2R)-2-amino-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-phenylacetamide
4-(2,6-dimethoxypyridine-3-carbonyl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
3-chloro-4-fluoro-N-[2-(1H-imidazol-4-yl)ethyl]-1-benzothiophene-2-carboxamide
N-[4-({1-methyl-2,4-dioxo-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decan-8-yl}methyl)phenyl]acetamide
methyl 3-[(3S,4R)-1-[(2-fluorophenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]propanoate
1-(1-benzothiophen-2-ylmethyl)-3-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
4-benzyl-3-ethyl-1-[2-(methylamino)pyridine-4-carbonyl]-1,4-diazepan-5-one
(1S,5R)-6-[(1R,5S,6R)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-3-benzyl-3,6-diazabicyclo[3.2.2]nonane
[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl][(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
2,3,6-trimethyl-N-[1-(1-methyl-1H-imidazol-2-yl)butyl]quinoline-4-carboxamide
(1S,6R)-9-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
6-(2,3-dihydro-1-benzofuran-5-ylmethyl)-N-(furan-2-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
4-{3-[(3S,4R)-3-ethyl-4-hydroxy-4-methylpiperidin-1-yl]-3-oxopropyl}-N-methylbenzene-1-sulfonamide
1-[(3R)-3-cyclopropyl-3-hydroxy-4,4-dimethylpyrrolidin-1-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
4-(2-chlorophenoxy)-1-(3-methyl-1H-pyrazole-5-carbonyl)piperidine
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-[(4-fluoro-2-methoxyphenyl)methyl]-N-methylpiperidin-3-amine
1-[3-(dimethylamino)-2,2-dimethylpropyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-(methylsulfanyl)-3-{3-[3-(trifluoromethyl)benzoyl]piperidine-1-carbonyl}pyridine
4-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-5-methylpyrimidin-2-amine
1-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-3-(2-fluorophenyl)propan-1-one
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxybutan-1-one
2-(2H-1,3-benzodioxol-5-yl)-5-(methanesulfonylmethyl)pyridine
5-[2-(4-methoxyphenyl)piperidine-1-carbonyl]-2-phenylpyrimidin-4-ol
N-({4-[4-(2-methoxyphenyl)piperazin-1-yl]quinazolin-2-yl}methyl)benzenesulfonamide
(1S,5R)-3-(quinolin-2-yl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
7-methyl-4-(thian-4-yl)-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-[(3-methylphenyl)methyl]piperidine
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-methyl-N-[(3-methylpyridin-2-yl)methyl]benzamide
2-{4-[5-(1-methylpiperidin-2-yl)-1,2,4-oxadiazol-3-yl]phenyl}ethan-1-ol
N-methyl-3-[1-(1H-1,2,3,4-tetrazol-5-yl)-1H-pyrazol-4-yl]benzamide
1-(5-chloro-3-phenyl-1H-indole-2-carbonyl)azetidine-2-carboxylic acid
5-({2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}methyl)-N-methylfuran-2-carboxamide
methyl (2S)-2-({[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amino)-2-phenylacetate
1-[4-(4-fluorophenyl)piperazin-1-yl]-3-[(3S,4R)-4-(morpholin-4-yl)-1-(naphthalen-2-ylmethyl)piperidin-3-yl]propan-1-one
ethyl 5-(7-fluoro-2-methylquinoline-4-carbonyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl](methyl){[5-(pyrimidin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}amine
N-[(3R,4R)-3-hydroxy-1-[4-(morpholin-4-yl)butanoyl]piperidin-4-yl]pyridine-2-carboxamide
1-[2-hydroxy-4-(methylsulfanyl)butanoyl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-N-methyl-4-oxo-N-(1H-pyrazol-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-(4-carbamoylpiperidin-1-yl)-2-[6-(piperidin-1-yl)pyridin-3-yl]acetic acid
4-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
5-fluoro-2-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}pyridine
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-(2-phenylpropan-2-yl)piperidine-3-carboxamide