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2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
1-(3,5-dimethylphenyl)-4-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperazin-2-one
3-methyl-1-[3-(4-methylphenyl)phenyl]-3-[3-(oxolan-2-yl)propyl]urea
N-cyclobutyl-2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
4-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-[(2S)-2-aminohexanoyl]-N-(pyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
N-(butan-2-yl)-2-[3-(1H-imidazol-1-yl)propyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
5-[(2-carboxy-4,6-dimethoxyphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
methyl (2S,4S,5R)-4-(butylcarbamoyl)-5-(3-chlorophenyl)-1-methylpyrrolidine-2-carboxylate
3-(morpholin-4-yl)-N-(4-phenoxyphenyl)piperidine-1-carboxamide
N-(3-chloro-4-methoxyphenyl)-3-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-3-yl}propanamide
4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]-N,N-dimethylbutanamide
2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl}-5-methylpyrazine
(8R,9aS)-8-hydroxy-2-(2-phenoxyethyl)-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-4-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-[3-(methylsulfanyl)phenyl]-2-(thiomorpholin-4-yl)acetic acid
{2-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}urea
3-({2-[2-(3,5-dimethyl-1-benzofuran-2-yl)-1H-imidazol-1-yl]ethyl}sulfanyl)-4-methyl-4H-1,2,4-triazole
4-{6-[1-(3-methoxypropyl)piperidin-4-yl]-2-methylpyrimidin-4-yl}morpholine
1-(1,3-dioxo-2-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-5-ylmethyl}-2,3-dihydro-1H-isoindol-4-yl)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidine-3-carboxamide
4,4-difluoro-N-{4-[2-(pyridin-2-yl)ethyl]phenyl}piperidine-1-carboxamide
3-{[4-(4-chlorophenoxy)piperidin-1-yl]methyl}pyridine
(3R,4R)-4-ethyl-1-[1-(2-fluorophenyl)cyclopropanecarbonyl]piperidine-3,4-diol
1-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-5-(1-ethyl-1H-pyrazol-3-yl)-4-phenyl-1H-imidazole
1-(5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-N-(4-fluorophenyl)piperazine-2-carboxamide
4-{[1-(2-methyl-3-phenylcycloprop-2-ene-1-carbonyl)piperidin-4-yl]methyl}morpholine
2-{2-[4-(1H-pyrazol-5-yl)phenyl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
1-(furan-2-carbonyl)-4-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazine
methyl 2-(diethylsulfamoyl)-6-[2-(3-methylphenyl)acetyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl][(5-ethyl-1,3,4-oxadiazol-2-yl)methyl](propan-2-yl)amine
1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
ethyl 1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
(4aR,7aS)-1-{2-[(1-benzofuran-2-ylmethyl)amino]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-{4-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]phenyl}-1-phenyl-1H-imidazole
6,7-difluoro-3-[2-(4-methylpiperazin-1-yl)ethyl]-3,4-dihydroquinazolin-4-one
3-{[2-(morpholin-4-ylmethyl)piperidin-1-yl]sulfonyl}benzoic acid
3-[(2-fluorophenyl)methyl]-1-[4-(oxan-2-ylmethoxy)phenyl]urea
N-(2-hydroxy-2-phenylethyl)-2-methyl-2-(thiophen-2-ylformamido)propanamide
7-[(2-fluorophenyl)methyl]-2-(1-methyl-1H-imidazole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
6-cyclopentyl-N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[(2-methoxyphenyl)methyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-methyl-3-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-1-[4-(1H-1,2,4-triazol-1-yl)phenyl]urea
1-(4-methanesulfonylbenzoyl)-3-(2-methylphenoxymethyl)piperidine
4-benzyl-1-[3-(4-fluorophenyl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidine
6-ethyl-N-(2-methoxyethyl)-2-oxo-N-(pyridin-3-ylmethyl)-1,2-dihydropyridine-4-carboxamide
1-{2-[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
(3S,4S)-1-{[5-(cyclohexylsulfanyl)furan-2-yl]methyl}-4-(morpholin-4-yl)pyrrolidin-3-ol
[(3R,4S)-1-[(6-methoxynaphthalen-2-yl)methyl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
3-[(2R,3R,6R)-5-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol