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N-{1-[(2-fluorophenyl)methyl]piperidin-4-yl}-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]-N-[1-(morpholin-4-ylmethyl)cyclopentyl]benzamide
2-methoxy-5-{1-[2-(1H-pyrazol-1-yl)ethyl]-1H-1,2,3-triazol-4-yl}benzoic acid
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-2-(2-oxopiperidin-1-yl)acetamide
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-(2-methylpropyl)-N5-(2-phenoxyethyl)piperidine-3,5-dicarboxamide
methyl 4-{[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylate
1-(2-aminoethyl)-N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
8-{[5-(2-chlorophenyl)furan-2-yl]methyl}-1-ethyl-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S,3R)-2-[({4-[2-(dimethylamino)ethoxy]phenyl}methyl)amino]-3-hydroxybutanamide
(3S,4S)-4-cyclopropyl-1-[(3,5-dichloropyridin-4-yl)methyl]pyrrolidine-3-carboxylic acid
8-[(3,4-difluorophenyl)methyl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
(4aS,8aR)-1-(2-aminoethyl)-6-(2-fluoro-6-methoxybenzoyl)-decahydro-1,6-naphthyridin-2-one
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(3-methylphenyl)methyl]piperidine-3-carboxamide
3-[5-(5-methyl-1,2-oxazol-3-yl)-1,3,4-oxadiazol-2-yl]-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}propanamide
(1S,5R)-6-[(3,5-dimethyl-1H-indol-2-yl)methyl]-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-5-ethylpyrimidin-2-amine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-(propan-2-yl)piperidine-4-carboxamide
7-methyl-N-{1-[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]ethyl}-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
3-[2-(4-chlorophenyl)ethyl]-3,4-dihydropteridin-4-one
N-(3-acetylphenyl)-3-(hydroxymethyl)-3-(3-phenylpropyl)piperidine-1-carboxamide
4-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-1λ6-thiomorpholine-1,1-dione
2-amino-4-(3-ethoxy-4-hydroxyphenyl)-6-(4-hydroxy-3-methoxyphenyl)pyridine-3-carbonitrile
5-[(3-cyclopropyl-1H-1,2,4-triazol-5-yl)methyl]-4,6-dimethylpyrimidin-2-amine
1-(pyridin-3-ylmethyl)-4-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]-1,4-diazepane
(1R,3S)-7-(8-chloroquinoline-2-carbonyl)-3-methoxy-7-azaspiro[3.5]nonan-1-ol
1-cyclohexyl-4-[(1E)-1-(furan-2-yl)prop-1-en-2-yl]-3-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2,3,5-trimethyl-6-{[3-(1-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyrazine
9-cyclopropanecarbonyl-2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecane
3-[3-(4-phenylbenzoyl)piperidin-1-yl]propanoic acid
(1R,5S,8S)-N-(2-chloro-4,6-dimethylphenyl)-8-methoxy-3-azabicyclo[3.2.1]octane-3-carboxamide
1-{3-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
6-methyl-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[(3S,4R)-1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
3-benzyl-8-[(4-hydroxyphenyl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2-methoxyethyl)-N-{[6-methyl-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}thiophene-2-carboxamide
4-methyl-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)pyrimidin-2-amine
6-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}-2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
(benzylsulfamoyl)[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]amine
1-(2-methoxypyridin-3-yl)-3-methyl-3-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]urea
4-{[5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,2-dihydrophthalazin-1-one
N-[4-(3-methoxyphenyl)phenyl]-1-(1,2,4-oxadiazol-3-ylmethyl)piperidine-3-carboxamide
4-{1-[(2,2-dimethyloxan-4-yl)methyl]piperidin-4-yl}-5-methylpyrimidine
2-[1-(1,3-thiazol-4-ylmethyl)azetidin-3-yl]-1H-1,3-benzodiazole
6-(morpholin-4-yl)-N4-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]pyrimidine-2,4-diamine
N,N-dimethyl-2-[(1S,5R)-3-(1-methyl-1H-pyrazole-4-carbonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-1-(4-fluorophenyl)cyclopropane-1-carboxamide
2-[1-(5,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)-N-[(2-methoxyphenyl)methyl]formamido]acetic acid
1-[(6-methoxy-2H-chromen-3-yl)methyl]-4-(pyridin-4-ylmethyl)-1,4-diazepane
6-(furan-3-yl)-2-[3-({methyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
1-[3-methoxy-5-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}urea