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2-(4-{[4-(prop-2-en-1-yl)piperazin-1-yl]methyl}phenyl)-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
N-phenyl-5-[4-(pyrazin-2-yl)piperazine-1-carbonyl]pyrimidin-2-amine
N-[2-(propan-2-yl)-2H-1,2,3-triazol-4-yl]-2-{4-[3-(1H-pyrazol-1-yl)phenyl]-1H-pyrazol-1-yl}acetamide
1,3-dimethyl-N-[4-(1H-pyrazol-1-yl)butan-2-yl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
5-[(4-hydroxypiperidin-1-yl)methyl]-N-[(1S)-1-phenylpropyl]-1,2-oxazole-3-carboxamide
10-methoxy-5-(4-methylpyrimidin-2-yl)-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
1-cyclopentyl-3-methyl-4-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(3R,4R)-1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
3-(cyclopropylmethyl)-5-(4-methanesulfonylphenoxymethyl)-1,2,4-oxadiazole
9-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-propoxyethan-1-one
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3,6-dimethyl-N-{3-[(pyridin-3-yl)amino]propyl}-1-benzofuran-2-carboxamide
2-[(4-chlorophenyl)methyl]-8-(3-methyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2-(2-methoxyethyl)-8-[2-(pyridin-3-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
3-(3,4-diethyl-1-methyl-1H-pyrazol-5-yl)-1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}urea
1-(azepan-1-yl)-3-({2-ethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)propan-2-ol
1-ethyl-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-methyl-N-[2-(5-methyl-1H-indol-3-yl)pyridin-3-yl]propanamide
2-{9-[2-(4-fluorophenoxy)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
3-hydroxy-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1,2-oxazole-5-carboxamide
5-methyl-N-(1,2,2,6,6-pentamethylpiperidin-4-yl)pyrimidin-2-amine
5,7-dimethyl-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]pyrido[2,3-d]pyrimidin-4-amine
(2R,6S)-4-{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}-2,6-dimethylmorpholine
5-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylic acid
2-(3,3-diphenylpiperidin-1-yl)-N-(propan-2-yl)pyridine-4-carboxamide
N-cyclopropyl-5-(phenoxymethyl)-N-(pyridin-2-ylmethyl)-1H-pyrazole-3-carboxamide
(1S,5R)-3-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-ethyl-6-methyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]pyrimidin-4-amine
N-[2-(1,4-dioxo-1,2,3,4-tetrahydrophthalazin-2-yl)ethyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
N-(cyclobutylmethyl)-1-(2-methoxyphenyl)-N-(oxolan-2-ylmethyl)-1H-pyrazole-4-carboxamide
(1H-imidazol-2-ylmethyl)[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]methylamine
N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(oxolan-2-ylmethyl)-3-(pyrazin-2-yl)propanamide
5-(azepane-1-carbonyl)-1-(butan-2-yl)-N-[(3,4-dimethoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
N-[(2-amino-1,3-thiazol-4-yl)methyl]-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
2-methyl-4-(1-{2-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-4-yl)pyrimidine
N-[2-(2-chlorophenyl)-1-{1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-4-yl}ethyl]-N-methylfuran-2-carboxamide
3-[2-oxo-2-(4-phenyl-1,4-diazepan-1-yl)ethyl]-2,3-dihydro-1λ6-thiophene-1,1-dione
N-[(2S,4R,6R)-2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-6-phenyloxan-4-yl]acetamide
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2,5-dimethylbenzamide
2-{[(3-acetylphenyl)formamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
2-(ethoxymethyl)-7-methyl-N-[2-(thiophen-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-5-(4-methyl-1,4-diazepan-1-yl)-2,3-dihydropyridazin-3-one
N-ethyl-2-{4-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperazin-1-yl}acetamide
5-{2-[2-(ethylamino)pyrimidin-5-yl]-1H-imidazol-1-yl}-6-methoxy-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-[4-(1H-1,3-benzodiazol-2-ylmethyl)-1-[(4-ethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
6-(2-fluorophenyl)-N-[2-(3-hydroxypiperidin-1-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-(furan-2-ylmethyl)-4-methyl-2-(propan-2-yl)-N-(pyridin-2-ylmethyl)-1,3-thiazole-5-carboxamide
5-(oxolan-2-yl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}thiophene-2-carboxamide
3-({2-[(2-methoxyethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)pyrrolidin-2-one