Tips: Press Ctrl key to select multiple functional groups
1-[2-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]ethan-1-one
3-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-1-(1-ethyl-1H-1,2,3-triazol-4-yl)-3-methylurea
(2S,4R)-4-amino-1-{[1-(3-cyanophenyl)-1H-pyrrol-2-yl]methyl}-N-methylpyrrolidine-2-carboxamide
6-[4-(oxolan-3-ylmethyl)piperazin-1-yl]-9H-purine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-5-fluoro-N-methyl-1H-indole-2-carboxamide
(4aR,7aS)-1-(2-methoxyethyl)-4-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]acetamide
N2-{2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-N1-(pyridin-3-yl)ethane-1,2-diamine
2-({4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
5-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine-3-carbonyl)-1-(2-methoxyethyl)piperidin-2-one
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-2-phenyl-1H-imidazole-4-carboxamide
2-ethoxy-N-methyl-N-[(3-methylthiophen-2-yl)methyl]pyridine-3-carboxamide
(8R,9aS)-2-(furan-2-ylmethyl)-8-hydroxy-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
5-(2H-1,3-benzodioxole-5-carbonyl)-3-(4-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-{3-[2-(3,4-difluorophenyl)ethyl]piperidine-1-carbonyl}pyridin-1-ium-1-olate
(2S,4R)-4-{[(3-fluorophenyl)methyl]amino}-N,1-bis(propan-2-yl)pyrrolidine-2-carboxamide
2-methyl-1-[1-(1-methylpiperidine-2-carbonyl)piperidin-4-yl]-5-(trifluoromethyl)-1H-1,3-benzodiazole
N-(5-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]acetamido}-2-methoxyphenyl)benzamide
[(4aS,8aR)-6-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-decahydro-1,6-naphthyridin-4a-yl]methanol
3-(1H-pyrazol-1-ylmethyl)-N-(1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-2-methyl-1,4-diazepan-5-one
N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
(3S,4R)-1-[(4-ethoxy-3-methoxyphenyl)methyl]-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-5,6,7,8-tetrahydroquinoline-3-carboxamide
4-(2-{[(4-fluorophenyl)methyl]carbamoyl}ethyl)-N-(prop-2-en-1-yl)piperidine-1-carboxamide
1-(4-chlorophenyl)-N-[(1-cyclohexylpiperidin-3-yl)methyl]cyclopropane-1-carboxamide
methyl 5-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
4-({1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]piperidin-2-yl}methyl)morpholine
(3S,5R,9R)-11-[(2,4-dimethylphenyl)methyl]-5-hydroxy-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
N-[(3S,4R)-1-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]-4-propylpyrrolidin-3-yl]acetamide
3-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-ol
1-(2-methylphenyl)-4-[3-(piperidin-3-yl)benzoyl]-1,4-diazepane
4-[(3S)-3-ethylmorpholin-4-yl]-1-phenylbutan-1-one
3-oxo-N-phenyl-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecane-9-carboxamide
4-[(1-ethyl-1H-indol-6-yl)methyl]-N,N-dimethylpiperazine-1-sulfonamide
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-3-(pyrrolidin-1-ylmethyl)piperidine
1-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-(morpholin-4-yl)phenyl]ethan-1-one
3-(1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidin-2-yl)pyridine
2-{4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperazin-1-yl}-5-methyl-1,3-benzoxazole
1-[(3-methoxyphenyl)methyl]-4-[(2-methyl-1,3-oxazol-4-yl)methyl]piperazin-2-one
5-(propan-2-yl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-{3,9-diazaspiro[5.6]dodecan-9-yl}-2-(2-methoxyphenyl)ethan-1-one
1-[(3-methoxyphenyl)methyl]-5-[2-(1H-pyrazol-1-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-{[(1R,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}pyridin-2-amine
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2-(methylamino)-1,3-thiazole-4-carboxamide
3-(3-methoxyphenyl)-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1H-pyrazole-5-carboxamide
2-({[(3R,4R)-1-(3-chloro-2-fluorobenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
(1S,5R)-6-benzyl-3-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
N-{4-[({1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}amino)methyl]phenyl}acetamide