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5-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)pyridine-3-carboxylic acid
2-(5-acetylthiophen-3-yl)-1-[(3S)-3-ethylmorpholin-4-yl]ethan-1-one
3-methyl-3-[3-(1-methyl-1H-imidazol-2-yl)propyl]-1-[3-methyl-4-(2-oxopyrrolidin-1-yl)phenyl]urea
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-[4-(1,3-thiazol-4-yl)phenyl]pyrrolidine-2-carboxamide
3-ethoxy-N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-4-(prop-2-en-1-yloxy)benzamide
3-{2-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-2-oxoethyl}-1λ6-thiolane-1,1-dione
N-(4-acetylphenyl)-3-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidine-1-carboxamide
(1R,9S)-5-amino-3-(2,6-dichloro-3-hydroxyphenyl)-6,12-diazatricyclo[7.2.1.02,7]dodeca-2(7),3,5-triene-4-carbonitrile
N,2,4-trimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]pyrimidine-5-carboxamide
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
5-methyl-N-{4-[2-(morpholin-2-yl)acetamido]phenyl}furan-2-carboxamide
(1S,5R)-1,3,3-trimethyl-N-(4-oxo-4H-chromen-6-yl)-6-azabicyclo[3.2.1]octane-6-carboxamide
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-4-(4H-1,2,4-triazol-4-yl)benzamide
2-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]benzene-1,3-diol
N-(3-chloro-4-methoxyphenyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carboxamide
4-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1-methyl-1H-imidazole-4-sulfonamide
2-amino-4-methyl-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1,3-benzothiazole-6-carboxamide
N-(but-2-yn-1-yl)-N-(furan-2-ylmethyl)-2-(N-phenylmethanesulfonamido)propanamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-6-methoxy-3-methyl-1-benzofuran-2-carboxamide
3-fluoro-6-methyl-N-[3-(3-oxopiperazin-1-yl)propyl]imidazo[1,2-a]pyridine-2-carboxamide
2-(3-methylbut-2-en-1-yl)-8-[4-(1H-pyrazol-4-yl)butanoyl]-2,8-diazaspiro[4.5]decan-3-one
(2-methoxyethyl)(methyl)(2-{[6-(piperidin-1-yl)pyrimidin-4-yl]oxy}hex-5-en-1-yl)amine
3,5-dimethoxy-N-{[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-3-yl]methyl}benzamide
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-2-(propan-2-yloxy)ethan-1-one
N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-4-(1H-1,2,4-triazol-3-yl)benzamide
1-(cyclohexylmethyl)-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-6-oxopiperidine-3-carboxamide
[2-(dimethyl-1,3-thiazol-5-yl)phenyl]methanol
3-[({[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}amino)methyl]piperidin-3-ol
N-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]methanesulfonamide
2-cyclopropyl-N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)acetamide
N,N-dimethyl-5-({methyl[1-(1,3-thiazol-2-yl)ethyl]amino}methyl)pyridin-2-amine
2-(pyridin-3-yl)-N-[2-(thiophen-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
{3-[(2,4-difluorophenyl)methyl]-1-[(4-ethylphenyl)methyl]piperidin-3-yl}methanol
2-[({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amino]pyridine-4-carbonitrile
3-(2-methoxyethyl)-1-(thiophen-3-ylmethyl)piperidine-3-carboxylic acid
1-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-ethoxyethan-1-one
6-methyl-2-{1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carboxamide
1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-4-(pyridin-3-yl)piperazine
N-(3-methyl-1,1-dioxo-1λ6-thiolan-3-yl)-2-(2-methyl-1,3-thiazol-4-yl)-N-(prop-2-en-1-yl)acetamide
1-{1-[1-(3-cyclopropyl-1-phenyl-1H-1,2,4-triazol-5-yl)propan-2-yl]-3,5-dimethyl-1H-pyrazol-4-yl}ethan-1-one
N-[(3R,4S)-4-cyclopropyl-1-(2-methoxyacetyl)pyrrolidin-3-yl]-2-(1-methyl-1H-pyrrol-2-yl)-2-oxoacetamide
(2,1,3-benzoxadiazol-4-ylmethyl)[(dimethyl-1,2-oxazol-4-yl)methyl]methylamine
N-[(3S,4R)-1-(5-chloropyridine-3-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
N,N,1-trimethyl-3-[2-(trifluoromethoxy)phenyl]-1H-1,2,4-triazol-5-amine
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(5-methylthiophen-2-yl)-5-(morpholine-4-sulfonyl)benzamide
2,2-dimethyl-3-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)propan-1-ol
N-{[7-fluoro-5-(quinolin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,5-dimethylfuran-3-carboxamide
N-[1-ethyl-2-(3-methoxyphenyl)-7-(4-propylpiperazine-1-carbonyl)-1H-1,3-benzodiazol-5-yl]acetamide
5-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydropyridin-2-one