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(1-{[methyl({trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl})amino]methyl}cyclopentyl)methanol
4-phenyl-1-[5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl]piperidine-4-carbonitrile
4-[4-({3-[(4-methoxyphenyl)amino]piperidin-1-yl}methyl)phenyl]but-3-yn-1-ol
(1R,7S)-3-[(5-methylpyrazin-2-yl)methyl]-6-(morpholine-4-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1-(2-methoxyethyl)-6-oxo-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperidine-3-carboxamide
1-(azocan-1-yl)-3-[4-({[(4,6-dimethylpyrimidin-2-yl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
4-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-N-methylpyridin-2-amine
2-[2-(1H-imidazol-4-yl)ethyl]-9-[(2S)-2-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
2-methoxy-1-{1-methyl-4-[3-(5-methylfuran-2-yl)butyl]-1,4,9-triazaspiro[5.5]undecan-9-yl}ethan-1-one
2-methyl-5-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
1-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-(pyridin-3-yl)ethane-1,2-dione
8-methoxy-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-amine
1-[4-(4-acetylphenyl)piperazin-1-yl]-2-(pyrrolidin-3-yl)ethan-1-one
3-(oxolan-3-yl)-5-{4H-thieno[3,2-b]pyrrol-5-yl}-1,2,4-oxadiazole
4-[(2R)-3-hydroxy-2-{[6-(propan-2-yl)pyrimidin-4-yl]amino}propyl]phenol
(2,3-dihydro-1-benzofuran-2-ylmethyl)(methyl)[(1-methyl-1H-imidazol-5-yl)methyl]amine
1-[(3-chlorophenyl)methyl]-4-(1-ethyl-1H-imidazol-2-yl)piperidine
5-(2-methoxy-4-methylphenoxymethyl)-N-(1H-1,2,4-triazol-3-ylmethyl)-1,2-oxazole-3-carboxamide
2-[5-(4-phenyl-1,4-diazepane-1-carbonyl)-1H-1,3-benzodiazol-1-yl]ethan-1-ol
3-methyl-N-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}-1H-pyrazole-5-carboxamide
5-({3-oxo-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-2-yl}methyl)-1,2,4-oxadiazole-3-carboxamide
[(3R,5S)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
N-cyclopropyl-2-[methyl(pyridin-3-ylmethyl)amino]-N-{[4-(methylsulfanyl)phenyl]methyl}acetamide
6-{1-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-4-yl}-2-methylpyrimidin-4-ol
(2S,4S)-4-(2,5-dimethylfuran-3-amido)-N,N-diethyl-1-methylpyrrolidine-2-carboxamide
1-[(3-methylphenyl)methyl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
2-[(2S)-2-amino-3-(1,3-thiazol-4-yl)propanamido]-N-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
1-(2-ethoxybenzoyl)-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
(3aR,6aS)-5-(5-chloropyridin-2-yl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{[3-(2-hydroxyethyl)-4-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-1-yl]methyl}phenol
N-butyl-2-[5-oxo-3-phenyl-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide
1-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one
N-(1-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
4-{[(prop-2-en-1-yl)(pyridin-2-ylmethyl)amino]methyl}benzonitrile
4-{[methyl(2-methylpropyl)amino]methyl}-N-(4-methyl-1,3-thiazol-2-yl)benzamide
1-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-[3-(trifluoromethyl)phenyl]piperazine
2-{3-[(4-acetyl-1,4-diazepan-1-yl)methyl]phenyl}-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
3-(2,2-difluoroethyl)-5-[(3-fluorophenyl)methyl]-5-(piperidin-4-yl)imidazolidine-2,4-dione
4-(pyridin-2-yl)-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}pyrimidin-2-amine
7-methyl-2-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
1-benzyl-N,N-dimethyl-5-{[(5-methylfuran-2-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
2-methyl-5-[1-(4-methylpyridin-2-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]pyrazine
6-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-7-methyl-4-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
N-methyl-2-[methyl(pyridin-3-ylmethyl)amino]-N-[1-(1,2-oxazol-3-yl)ethyl]acetamide
(1-methyl-5-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
2,2-dimethyl-N-(1-{1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}-1H-pyrazol-5-yl)propanamide
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
3-{1-[3-(1-methylpiperidin-3-yl)propanoyl]piperidin-4-yl}benzonitrile
N-ethyl-N-(2-methylprop-2-en-1-yl)-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide