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2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-(2-methoxyethyl)-N-methylbenzamide
2-(2-{1-[(3-chloro-2-fluorophenyl)methyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
3-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-1-(pyrrolidin-1-yl)propan-1-one
{3-[(2-methylphenyl)methyl]-1-(3-phenylprop-2-yn-1-yl)piperidin-3-yl}methanol
3-{1-[3-(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)propanoyl]piperidin-3-yl}-N,N-dimethylpropanamide
[(3-ethyl-1,2-oxazol-5-yl)methyl][(4-methanesulfonylphenyl)methyl]methylamine
2-{5-[1-methyl-5-(trifluoromethyl)-1H-pyrazol-3-yl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
2-(prop-2-en-1-yl)-9-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}-2,9-diazaspiro[5.5]undecan-3-one
4-(3-fluorophenyl)-3-[(4-methyl-1,3-thiazol-2-yl)methyl]-4H-1,2,4-triazole
1-(5-ethyl-1,3,4-oxadiazol-2-yl)spiro[azepane-4,2'-chromene]
1-(pyrazine-2-carbonyl)-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-4-carboxamide
7-(cyclopropylmethyl)-2-[(3S)-3-hydroxypyrrolidine-1-carbonyl]-6-(4-methoxyphenyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
ethyl 1-[(3,4-difluorophenyl)methyl]-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
N-[(3R,4S)-1-(3-fluoropyridin-2-yl)-4-propylpyrrolidin-3-yl]pyrrolidine-1-sulfonamide
2-(dimethyl-1,3-thiazol-5-yl)-1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
1-(oxan-4-yl)-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
N-[2-(4-fluorobenzenesulfonyl)ethyl]-2,3-dimethyl-1H-indole-7-carboxamide
N-(2-hydroxybutyl)-2-[(isoquinolin-5-yloxy)methyl]-1,3-oxazole-4-carboxamide
12-[(3S,4S)-3-(dimethylamino)-4-hydroxypyrrolidine-1-carbonyl]-8-thia-5-azatricyclo[7.4.0.02,7]trideca-1(13),2(7),9,11-tetraen-6-one
2-[benzyl({[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl})amino]ethan-1-ol
2-(3-fluorophenoxy)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
6-{[4-(1,3-benzothiazol-2-yl)-1,4-diazepan-1-yl]methyl}-1,4-oxazepan-6-ol
1-(1-methylpiperidin-4-yl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}piperidine-3-carboxamide
methyl 4-({1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}carbamoyl)butanoate
1-cyclohexyl-3-(cyclopropylmethyl)-N-methyl-2-oxo-N-[2-(1H-pyrazol-4-yl)ethyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-[2-(4-fluorophenyl)ethyl]-4-{[5-(propan-2-yl)pyrimidin-4-yl]amino}pyrrolidin-2-one
N2,N2-dimethyl-N5-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)-4H,5H,6H,7H-thieno[3,2-c]pyridine-2,5-dicarboxamide
N-[(1-{[4-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)methyl]thiophene-2-carboxamide
(3S,4S)-3-hydroxy-N-[4-(pentyloxy)phenyl]-4-(pyrrolidin-1-yl)pyrrolidine-1-carboxamide
N-[2-(3,4-dimethoxyphenyl)propan-2-yl]-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-({5-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
3-(4-chlorobenzoyl)-1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidine
(2S,4S)-4-{[(2,5-dimethylphenyl)methyl]amino}-N-(2-methoxyethyl)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)-2-(2-oxoazepan-1-yl)acetamide
4-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-methylpyrimidine
(1S,3R)-3-amino-N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}cyclopentane-1-carboxamide
[4-(2-phenoxyethyl)-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-4-yl]methanol
(1R)-1-[(4-methoxyphenyl)methyl]-2-(5-methyl-1,2-oxazole-3-carbonyl)-1,2,3,4,5,6,7,8-octahydroisoquinoline
1-(5-cyclopropyl-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-1H-pyrazole-4-carbonyl)-N,N-dimethylpyrrolidin-3-amine
5-cyano-N-[(3R,4S)-4-cyclopropyl-1-(2-methoxyethyl)pyrrolidin-3-yl]-2-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
methyl 2-{1-[(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)carbamoyl]pyrrolidin-3-yl}acetate
2-(1H-1,3-benzodiazol-1-yl)-N-[(5-methylpyrazin-2-yl)methyl]propanamide
3-(4-methoxyphenyl)-N-(quinolin-3-ylmethyl)-1H-pyrazole-5-carboxamide
N-({5-[(2,3-difluoro-6-methoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
(4aS,8aR)-6-(3-methoxypropanoyl)-1-[2-(5-methylfuran-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-{3-[(2-ethylphenyl)carbamoyl]phenyl}pyridazine-4-carboxamide
6-[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)piperidin-4-yl]-3,4-dihydropyrimidin-4-one
[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)(pyrimidin-2-ylmethyl)amine
8-[(5-acetylthiophen-3-yl)methyl]-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-methyl-6-({4-[methyl(phenyl)amino]phenyl}methyl)-N-(1,3-thiazol-4-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide