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1-(4-methoxyphenyl)-3-methyl-4-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperazin-2-one
N-ethyl-4-methyl-5-[3-(pyridin-2-yl)azetidine-1-carbonyl]-1,3-thiazol-2-amine
1-[(3-fluorophenyl)methyl]-4-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}piperazine
(3S,4S)-4-(azepan-1-yl)-1-{[2-(propylsulfanyl)pyrimidin-5-yl]methyl}pyrrolidin-3-ol
N-cyclobutyl-2-(dimethylamino)-2-(4-fluorophenyl)acetamide
2-amino-4-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
2-(methylamino)-1-[3-(3-methylphenoxy)azetidin-1-yl]ethan-1-one
4-ethyl-3-[1-(2-phenyl-1H-imidazole-4-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazine-1-sulfonamide
6-[(3-fluorophenyl)methoxy]-1-(2-phenylethyl)-4-[3-(pyrazin-2-yl)propanoyl]-1,4-diazepan-2-one
1-(2-methyl-1,4-oxazepan-4-yl)-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butan-1-one
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(pyrrolidine-1-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[4-(3-fluorophenyl)phenyl]piperidin-4-ol
4-benzyl-1-cyclohexyl-3-hydroxy-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-(2-amino-1,3-thiazol-4-yl)-N-[2-(1H-imidazol-4-yl)ethyl]propanamide
2-amino-6-{4-[(dimethylamino)methyl]thiophen-2-yl}-4-(pyridin-3-yl)pyridine-3-carbonitrile
7-chloro-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-3,5-dimethyl-1-benzofuran-2-carboxamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)furan-3-carboxamide
2-[4-(1H-indol-3-ylmethyl)-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
2-(pyridin-3-yl)-N-[3-(4H-1,2,4-triazol-4-yl)propyl]pyrimidine-5-carboxamide
N-cyclopropyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]imidazo[1,2-a]pyridine-6-carboxamide
(1S,5R)-6-(5-chloro-2-methoxybenzoyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-(1-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl)acetamide
7-(2-methylphenyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
8-(2-amino-6-methoxypyrimidin-4-yl)-2-[(dimethyl-1,2-oxazol-4-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
1-(2,3-dihydro-1H-indene-5-carbonyl)-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
6-[(diethylamino)methyl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-methylpropyl (1S,5R)-7-oxo-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxylate
N-(cyclopropylmethyl)-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
1-[4-({3-hydroxy-1-oxa-8-azaspiro[4.5]decan-8-yl}methyl)thiophen-2-yl]ethan-1-one
4-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-1-methyl-1,2-dihydroquinolin-2-one
N-[2-(4-methylphenyl)propan-2-yl]-4-oxo-1,4-dihydroquinoline-2-carboxamide
(2R)-2-amino-N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-methoxypropanamide
2-[3-(pyridin-4-yl)phenoxy]propanoic acid
3-{9-oxa-2-azaspiro[5.5]undecane-2-sulfonyl}-N-(prop-2-en-1-yl)benzamide
N-({5-[(4-fluoro-2-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
3-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)benzamide
3-(2-hydroxyphenyl)-N-[5-(morpholin-4-yl)pentyl]-1H-pyrazole-5-carboxamide
2-(2-ethyl-1H-imidazol-1-yl)-1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)ethan-1-one
2-[6-hydroxy-4-(oxane-4-carbonyl)-1,4-diazepan-1-yl]pyridine-4-carboxamide
3-(1H-imidazol-2-yl)-1-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidine
[(5-chlorothiophen-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(oxolan-2-ylmethyl)amine
1-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-4-[(4-fluorophenyl)methyl]-1,4-diazepane
1-(2-chloro-4-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazine-7-carbonyl}phenyl)pyrrolidine
N-[(3,4-difluorophenyl)methyl]-3-(1-methyl-1H-pyrazol-5-yl)propanamide
(2,1,3-benzoxadiazol-5-ylmethyl)({[2-(2-methylphenoxy)pyridin-3-yl]methyl})amine
1-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
N-(2-cyclopropylphenyl)-2-(2-methoxyethyl)piperidine-1-carboxamide
4-(1H-pyrazol-1-yl)-1-(quinolin-4-yl)piperidine-4-carboxylic acid
2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one