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N,N-dimethyl-6-[3-(2-phenylethyl)piperidin-1-yl]pyridine-3-carboxamide
(2S,4R)-4-amino-1-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}-N,N-diethylpyrrolidine-2-carboxamide
ethyl 1-[(2-hydroxyphenyl)methyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
{imidazo[1,2-a]pyrimidin-6-ylmethyl}(methyl)[1-(4-methylpyridin-2-yl)propan-2-yl]amine
1-[(1R,3R,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]-3-(thiophen-2-yl)propan-1-one
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-[(2E)-2-methylbut-2-en-1-yl]piperidin-3-amine
4-(1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}azetidin-3-yl)morpholine
1-[(4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}thiophen-2-yl)methyl]piperazine
1-[1'-(2,4-difluorobenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
(2S,4R)-4-[(1-ethylpiperidin-4-yl)amino]-N-[2-(2-fluorophenyl)ethyl]-1-(propan-2-yl)pyrrolidine-2-carboxamide
1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-phenoxypiperidine-4-carboxylic acid
(1S,5R)-6-propyl-3-[2-(1H-pyrazol-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-methyl-N-(oxan-2-ylmethyl)-2-(1-oxo-1,2-dihydroisoquinolin-2-yl)acetamide
(3S,4R)-3-(dimethylamino)-N-[2-(methylsulfanyl)phenyl]-4-(propan-2-yl)pyrrolidine-1-carboxamide
methyl 5-cyano-2-methyl-6-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}pyridine-3-carboxylate
5-(2-phenylethyl)-5-(piperidin-4-yl)-3-(1,3-thiazol-5-ylmethyl)imidazolidine-2,4-dione
5-({3-[(2H-1,3-benzodioxol-5-yl)amino]piperidin-1-yl}methyl)-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
4-methyl-N-(2-{7-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
(1S,4S)-5-(4-tert-butylbenzoyl)-2-(2-fluorophenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
N-[(5-methylfuran-2-yl)methyl]-3-[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-3-yl]propanamide
2-(2,6-difluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-hydroxypiperidin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
N-(1H-indol-2-ylmethyl)-2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-(naphthalen-2-yloxy)-1-(quinoxalin-2-yl)piperidine-4-carboxylic acid
[5-chloro-7-(1,3-thiazol-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
2,3,5-trimethyl-N-[2-(pyrrolidin-1-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
N,N-diethyl-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[methyl(pyridin-3-ylmethyl)amino]-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl](methyl)[1-(pyridin-2-yl)propan-2-yl]amine
4-(4-chlorophenyl)-1-(oxolane-3-carbonyl)piperidin-4-ol
N-(1-hydroxybutan-2-yl)-2-(phenylamino)-N-(pyridin-3-ylmethyl)pyrimidine-5-carboxamide
8-[1-(hydroxymethyl)cyclopropanecarbonyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
N-(1,1-dioxo-1λ6-thian-4-yl)-N,2,7,8-tetramethylquinoline-4-carboxamide
3-[3-(1H-imidazol-1-yl)pyrrolidine-1-carbonyl]-5-(4-methoxyphenyl)-1H-pyrazole
(1R,5R)-6-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
5-{[(1,4-dioxan-2-ylmethyl)(methyl)amino]methyl}-N-propylpyrimidin-2-amine
3-(hydroxymethyl)-1-({3-[3-(piperidin-1-yl)propoxy]phenyl}methyl)pyrrolidin-3-ol
N-[(1-cyclopropanecarbonylpiperidin-3-yl)methyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-[3-(1H-imidazol-1-yl)propyl]pyrazolo[1,5-a]pyridine-7-carboxamide
3-methyl-4-oxo-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3,4-dihydroquinazoline-7-carboxamide
ethyl 1-(1H-imidazol-2-ylmethyl)-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
2-[2-(aminomethyl)-5-chloro-2,3-dihydro-1-benzofuran-7-yl]-N-cyclopropylpyridine-4-carboxamide
1-benzyl-3-methyl-4-[(2E)-pent-2-en-2-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-{4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-[3-(dimethylamino)-2,2-dimethylpropyl]pyrrolidin-2-one
1-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-2-(3-phenyl-1H-1,2,4-triazol-5-yl)ethan-1-one
(1R,3S)-3-{[1-(3-chlorophenyl)cyclopropyl]carbamoyl}cyclopentane-1-carboxylic acid
N-[(3R,4R)-3-hydroxy-1-[4-(1H-imidazol-1-yl)butanoyl]piperidin-4-yl]pyridine-2-carboxamide
1-(diphenylmethyl)-N-(6-hydroxy-6-methylheptan-2-yl)-1H-1,2,3-triazole-4-carboxamide
4-(2-ethyl-3-methyl-1-benzofuran-7-yl)-4H-1,2,4-triazole
1-[1-(3-aminopropanoyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide