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4-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-3-(propan-2-yl)piperazin-2-one
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-(3-phenylbutyl)piperidine
5-methyl-2-[3-(pyridine-3-carbonyl)piperidin-1-yl]pyrimidin-4-amine
1-(3-{3-[cyclohexyl(methyl)amino]propyl}-2-oxo-1-oxa-3,8-diazaspiro[4.5]decane-8-carbonyl)cyclopropane-1-carboxamide
1-{4-[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindole-2-carbonyl]phenyl}ethan-1-one
1-ethyl-N-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
4-[2-(benzenesulfonyl)ethyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
(4aR,7aS)-1-benzyl-4-(pyrrolidine-1-sulfonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]imidazo[1,2-a]pyridine-6-carboxamide
N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-2-(1H-pyrazol-1-yl)benzamide
N-[(3S,4R)-1-(4-cyclopentylpyrimidin-2-yl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
1-[2-(1-{8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-yl}piperidin-2-yl)ethyl]pyrrolidin-2-one
methyl 6-[2-(methoxycarbonyl)benzoyl]-2-[(prop-2-en-1-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-tert-butyl-2-methanesulfonyl-N-(thiophen-3-ylmethyl)acetamide
2-(1-{[1-(2-methoxyethyl)-2-(3-methylbutanesulfonyl)-1H-imidazol-5-yl]methyl}piperidin-2-yl)ethan-1-ol
9-[(5-fluoro-2-methoxyphenyl)methyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{4-[3-(2-fluorophenyl)-3-phenylpropanoyl]piperazin-1-yl}-N,N-dimethylacetamide
3-(1-methyl-1H-imidazole-2-carbonyl)-1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidine
N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(oxolan-2-ylmethyl)pyridine-4-carboxamide
5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-N-(pyridin-3-ylmethyl)pyridin-2-amine
1-(2,3-difluoro-4-methylbenzoyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
4-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(4-fluorophenyl)piperazin-2-one
5-chloro-6-(3-fluoro-4-methoxyphenyl)-2-methylpyrimidin-4-ol
N-[(2,3-dimethoxyphenyl)methyl]-5-ethyl-1,3,4-oxadiazol-2-amine
2-cyclopentanecarbonyl-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-methyl-2-{1-[2-phenyl-2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]piperidin-4-yl}acetamide
1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
(4aR,8aR)-2-cyclobutanecarbonyl-7-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}-decahydro-2,7-naphthyridin-4a-ol
7-(3,4-dimethylbenzoyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-{2-[1-(4-cyclopentylpyrimidin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
[4-({[4-(pyrrolidine-1-carbonyl)phenyl]methyl}amino)quinazolin-2-yl]methanol
2-(prop-2-en-1-yl)-9-[3-(pyridin-4-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(3-fluoro-4-hydroxyphenyl)-1-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]ethan-1-one
ethyl (4aS,8aR)-6-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-decahydro-1,6-naphthyridine-4a-carboxylate
1-[1-(2-phenylethyl)-5-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperidin-4-ol
N-{5H,6H,7H-cyclopenta[b]pyridin-7-yl}-1H-1,2,3-triazole-5-carboxamide
N-cyclopentyl-2-({[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}amino)propanamide
5-{[1-(4-chloro-2-methylphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(cyclohexylmethyl)-3-cyclopropyl-5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1H-1,2,4-triazole
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-4-(2-methanesulfonylethyl)piperazine
1-ethyl-4-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-3-methyl-1H-pyrazole
3-{[2-(methoxymethyl)piperidin-1-yl]methyl}-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
(1S,5R)-6-[(4-methylthiophen-2-yl)sulfonyl]-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-(4-fluorophenyl)ethyl]-4-propyl-N-(pyridin-3-ylmethyl)pyrimidine-5-carboxamide
N-(1-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-2-methyl-1-oxopropan-2-yl)acetamide
1-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]-1,4-diazepane-6-carboxylic acid
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
3-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}quinoline
(2S)-1-{[2-(3-chlorophenyl)-6,7-dimethoxyquinolin-3-yl]methyl}pyrrolidine-2-carboxamide
4-[4-(methylamino)pyrimidin-2-yl]-1-(2-phenylethyl)piperazin-2-one