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4-ethyl-1-methyl-3-{[1-(2-phenylpropyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-1-[(4-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
(1S,6R)-9-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
(2R)-2-amino-1-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
1-ethyl-N-(furan-2-ylmethyl)-N-methyl-5-[(pyridin-3-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-2,8-dimethylquinoline-3-carboxamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-5-ethyl-N-(prop-2-en-1-yl)-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
6-(2-chlorophenyl)-2-(4-hydroxypiperidine-1-carbonyl)-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
4-[5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carbonyl]thiomorpholine
2-[(dimethyl-4H-1,2,4-triazol-3-yl)methyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
2-(1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-pyrazol-4-yl)ethan-1-ol
1-{3-[1-(3-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]propyl}-1H-pyrazole
{2-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}urea
(2S,3R)-2-amino-3-hydroxy-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylbutanamide
1-[(4-chlorophenyl)methyl]-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
(1S,5R)-3-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-({[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl)carbamoyl}methyl)piperidine-4-carboxamide
(4aS,7aR)-1-(5-chloro-2-methoxybenzoyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-[4-(adamantan-1-yl)piperazin-1-yl]pyridine-2-carboxylic acid
6-(2-chlorophenyl)-7-(cyclopropylmethyl)-N-(3-hydroxypropyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]({[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl})amine
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
(3S,4R)-1-(1,7-dimethyl-1H-indole-2-carbonyl)-N,N-dimethyl-4-propylpyrrolidin-3-amine
methyl (2S,4S)-1-methyl-4-[4-methyl-3-(1H-pyrrol-1-yl)benzamido]pyrrolidine-2-carboxylate
N-(2,4-dimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-4-(2-oxo-1,3-oxazolidin-3-yl)piperidine-1-carboxamide
(2S,4S)-N-[2-(dimethylamino)ethyl]-1-[(2,5-dimethylphenyl)methyl]-4-[(4-fluorophenyl)sulfanyl]pyrrolidine-2-carboxamide
N-[2-(dimethylamino)ethyl]-2-methyl-N-[(3-methylthiophen-2-yl)methyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
(2R,3R)-1'-[(2-methylpyrimidin-5-yl)methyl]-3-(pyrrolidin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-[2-(dimethylamino)ethyl]-5-fluoro-3,4-dihydroquinazolin-4-one
(4aS,7aR)-1-(4-methyl-1H-imidazole-5-carbonyl)-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(2H-1,3-benzodioxol-5-yl)-1H-indole
4-(3-methoxyphenyl)-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]benzamide
8-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-1,3-dimethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3R)-3,4,4-trimethyl-1-(5-propyl-1,2-oxazole-4-carbonyl)pyrrolidin-3-ol
2-(7-fluoro-2-methyl-1H-indol-3-yl)-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
1-methyl-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]-1-{[3-(methylsulfanyl)phenyl]methyl}urea
5-{[2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamido]methyl}-1,2,4-oxadiazole-3-carboxamide
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1H-pyrazole-3-carbonitrile
2-amino-N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-4-methyl-1,3-thiazole-5-carboxamide
methyl 3-[(3S,4R)-1-[(2-hydroxynaphthalen-1-yl)methyl]-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanoate
N-[(2,6-difluoro-3-methylphenyl)methyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-{2-[3-(hydroxymethyl)-3-propylpiperidin-1-yl]-2-oxoethyl}acetamide
1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-2-(pyrrolidin-1-yl)propan-1-one
N-ethyl-3-(4-fluorophenyl)-N-(2-methoxyethyl)-3-phenylpropanamide
8-(2-methoxybutanoyl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{4-[(6-chloropyridin-3-yl)methyl]piperazin-1-yl}-4-(pyridin-3-yl)pyrimidine
1-[2-methoxy-4-({[(2-methoxyphenyl)methyl](methyl)amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-[3-(2-oxopyrrolidin-1-yl)propyl]pyrrolidin-2-one
(1S,6R)-9-(4-methyl-5-phenylthiophene-2-carbonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide