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1-{2-[1-(1-methyl-5-phenyl-1H-pyrazole-3-carbonyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
(1R,5R)-6-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N,N-dimethyl-4-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperazine-1-sulfonamide
(2R,3R,6R)-5-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
6-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-2-carboxylic acid
1-(furan-2-ylmethyl)-N-(isoquinolin-5-ylmethyl)-N-methylpiperidine-4-carboxamide
5-[1-(furan-2-ylmethyl)-4-hydroxypiperidin-4-yl]-N-methyl-N-(quinolin-8-ylmethyl)-1-benzofuran-2-carboxamide
5-(2-fluorophenyl)-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-[2-(4-methoxyphenyl)ethyl]-4-{[(4-methyl-1H-imidazol-5-yl)methyl]amino}pyrrolidin-2-one
4-[4-({3-[(3,4-difluorophenyl)amino]piperidin-1-yl}methyl)phenyl]but-3-yn-1-ol
3-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
1,9-dimethyl-4-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[(4aR,8aR)-7-[2-(2,3-dimethylphenoxy)ethyl]-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-{[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]methyl}propanamide
2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]acetamide
2-({6-[3-(1-methyl-1H-pyrazol-5-yl)phenyl]pyrazin-2-yl}sulfanyl)acetic acid
N-[2-(2-chloro-6-methylphenoxy)ethyl]-N'-(2-methylphenyl)propanediamide
(3S,4R)-1-(2,4-difluoro-3-methoxybenzoyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
(4aS,8aR)-6-[6-(morpholin-4-yl)pyrimidin-4-yl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
N-[(2-ethoxy-3-methoxyphenyl)methyl]-N,1-dimethyl-1H-1,3-benzodiazole-5-carboxamide
3,3-dimethyl-1-[(3S,4R)-1-(4-oxo-1,4-dihydroquinoline-2-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]urea
4-{5-methyl-4-[4-(propan-2-yl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}-3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaene
4-[(5-cyclopentylthiophen-2-yl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(4-{[(1R,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}thiophen-2-yl)ethan-1-one
N-(3-methoxypropyl)-3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
(3S,4S)-4-methyl-1-[(3-phenoxyphenyl)methyl]piperidine-3,4-diol
1-methyl-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[(2-chloro-6-fluorophenyl)methyl]-5-[(2-methoxyethoxy)methyl]-1H-1,2,4-triazole
3-{5-[1-(prop-2-en-1-yl)pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridazine
1-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazole
N-(butan-2-yl)-7-[(thiophen-2-ylmethyl)sulfamoyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
3-cyclopropyl-5-(1-propyl-1H-pyrazol-5-yl)-1H-1,2,4-triazole
2-cyclopentyl-N-{[4-(2,3-dihydro-1H-inden-2-yloxy)phenyl]methyl}-N-[(3S)-2-oxoazepan-3-yl]acetamide
4-(3-hydroxy-3-methylbutyl)-N-[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]benzamide
N-[(1R,3R)-3-aminocyclopentyl]-4-methyl-3-phenyl-1H-pyrazole-5-carboxamide
1-(3-{[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}propyl)piperidin-4-ol
2-[(3,5-difluorophenyl)methyl]-8-[2-(2-methyl-1H-imidazol-1-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
1-(2-phenylethyl)-4-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperazine
7-[2-(1H-1,2,4-triazol-1-yl)benzoyl]-2-oxa-7-azaspiro[4.5]decane
5-[4-({4-[(3,3-dimethylpyrrolidin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}methyl)piperidine-1-carbonyl]pyridin-2-amine
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)pyrrolidine-1-carboxamide
2-{3-[1-(pyridin-3-ylmethyl)-1H-pyrazol-3-yl]phenyl}quinoxaline
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[(2-methanesulfonylethyl)amino]methyl}piperidin-2-one
2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}acetamide
methyl({[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl})(thiophen-2-ylmethyl)amine
methyl 4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidine-1-carboxylate
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
N-benzyl-1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-N-methylpiperidin-4-amine
1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
3-(2-chlorophenyl)-1-(4-fluorophenyl)-4-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-1H-pyrazole