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3-methyl-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]pyridin-2-amine
(1S,5R)-N-[(2-fluorophenyl)methyl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-ethyl-N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-5-propyl-1,2-oxazole-3-carboxamide
1-benzyl-4-[(2-methoxy-4-methylphenyl)methyl]-3-methylpiperazin-2-one
4-ethyl-2-methyl-6-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}pyrimidine
N-(furan-3-ylmethyl)-1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-4-amine
5-fluoro-N4,N4-dimethyl-N2-[1-(4-methylphenyl)cyclopropyl]pyrimidine-2,4-diamine
1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
5-[(4-benzylpiperidin-1-yl)methyl]-N-methyl-N-[(1-methylpyrrolidin-2-yl)methyl]-1,2-oxazole-3-carboxamide
2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-N-(2-oxopyrrolidin-3-yl)-1,3-oxazole-4-carboxamide
(1S,5R)-6-(cyclopropylmethyl)-3-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
ethyl 5-(quinoxaline-5-carbonyl)-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-4-phenylbutane-1,4-dione
N3-[2-(3-chlorophenyl)ethyl]-N5-(cyclohexylmethyl)-1-(2-methoxyethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[3-({[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]carbamoyl}methoxy)phenyl]propanamide
3-(cyclohex-1-en-1-ylmethyl)-1-[4-(oxolan-2-ylmethoxy)phenyl]urea
1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-[(3-fluorophenyl)methyl]piperazine
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[2-(pyridin-3-yl)ethyl]acetamide
(3R,5S)-1-benzyl-N-[3-(dimethylamino)propyl]-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
3-(cyclopropylsulfamoyl)-5-(quinolin-8-yl)benzoic acid
1-[1-(pent-4-enoyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
(3S,9aR)-3-(cyclohexylmethyl)-8-(2-phenylethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(oxolane-2-carbonyl)-4-[3-(trifluoromethyl)phenoxy]piperidine
1-[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-{imidazo[1,2-a]pyridin-2-yl}propanamide
1-[(2E)-3-phenylprop-2-en-1-yl]-4-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperazine
(1S,3R)-3-amino-N-[(4-fluorophenyl)methyl]-N-(3-methoxypropyl)cyclopentane-1-carboxamide
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-pentylpyrimidin-2-amine
3-(6-chloro-2-methylpyridin-3-yl)-1-(3-hydroxypropyl)-1-(pyridin-3-ylmethyl)urea
1-[2-(3-fluorophenyl)piperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
methyl 3-[(3S,4R)-1-[(2-chloro-6-fluorophenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]propanoate
3-[5-(benzylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(5-methylthiophen-2-yl)methyl]piperidine
N-[(3R,4S)-1-cyclohexyl-4-cyclopropylpyrrolidin-3-yl]-1,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(1R,3S)-3-(2-hydroxyethoxy)-7-[(2-phenyl-1,3-oxazol-4-yl)methyl]-7-azaspiro[3.5]nonan-1-ol
2-methoxy-1-{4-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1,4-diazepan-1-yl}ethan-1-one
5-ethyl-2,3-dimethyl-N-(pyridin-2-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
(3aS,6aS)-2-(1-benzyl-1H-pyrazole-4-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(naphthalene-2-carbonyl)pyrrolidin-3-yl]methanol
cyclopentyl 4-(4-methyl-1,2,3-thiadiazole-5-amido)benzoate
1-{2-[2-(2,6-difluoro-4-methoxyphenyl)-1H-imidazol-1-yl]ethyl}-4-(propan-2-yl)piperazine
methyl[1-(thiophen-2-yl)ethyl][(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
5-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine-2-carbonitrile
2-[1-({2-phenylimidazo[1,2-a]pyridin-3-yl}methyl)piperidin-3-yl]ethan-1-amine
N-(2,3-dihydro-1H-inden-2-yl)-N,2-dimethyl-6-(piperidin-4-yl)pyrimidin-4-amine
2-({4-[(2-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-5-methoxyphenol
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
1-ethyl-4-{[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
2-{4-[(dimethylamino)methyl]phenyl}-5-methyl-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
1-(1H-indol-3-ylmethyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-(2-methoxyethyl)-8-[(5-methylthiophen-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one