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N-{[1-(5-chloro-2-methoxyphenyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}acetamide
N-benzyl-N-methyl-3-{[(2S)-4-methyl-2-(propan-2-yl)piperazin-1-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
N-(3-hydroxy-3-methylbutyl)-N-methyl-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-({[(2-methylphenyl)methyl]amino}methyl)piperidin-2-one
(2R)-1-[(3R,5S)-3,5-bis(hydroxymethyl)piperidin-1-yl]-2-hydroxy-2-(naphthalen-2-yl)ethan-1-one
5-chloro-2-[4-(pyridin-3-ylmethyl)-1,4-diazepane-1-carbonyl]phenol
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(methylsulfanyl)ethyl]acetamide
4-[4-(3-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1,3-oxazolidin-2-one
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-[(6-methylpyridin-2-yl)methyl]piperidine-4-carboxamide
3-(2-ethylbutyl)-8-[(2-methyl-1,3-oxazol-4-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-cyclopropyl-4-phenyl-9-(1H-pyrrole-2-carbonyl)-2,9-diazaspiro[5.5]undecane
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-1-phenyl-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
(4aS,7aR)-1-(4-methyl-1H-imidazole-5-carbonyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3aR,6aR)-2-cyclopentyl-5-[(dimethyl-1,3-thiazol-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
ethyl 4-{2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanoyl}piperazine-1-carboxylate
N-(1-{1-[1-(2-fluorophenyl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
N-methyl-2-{8-methyl-3-oxo-2,8-diazaspiro[4.5]decan-2-yl}-N-[(3-methylthiophen-2-yl)methyl]acetamide
N-(1H-1,3-benzodiazol-5-yl)-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine-1-carboxamide
1-[(3,4-dimethylphenyl)methyl]-4-[3-(trimethyl-1H-pyrazol-1-yl)propanoyl]piperazin-2-one
1-{2-hydroxy-3-[4-methoxy-2-({[2-(propan-2-yloxy)ethyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
5-[5-(3,5-dimethylfuran-2-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-[4-(morpholine-4-carbonyl)phenyl]piperidin-4-amine
6-methyl-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-5-(1,4-dioxan-2-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
2-{4-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperazin-1-yl}-6-(piperidine-1-carbonyl)pyrazine
1-(3-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}phenyl)pyrrolidin-2-one
6-(3-{4-[3-(4-ethylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}-3-oxopropyl)-2,3,4,5-tetrahydropyridazin-3-one
1-(4-carbamoylpyridin-2-yl)-4-(4-fluorophenoxy)piperidine-4-carboxylic acid
4-(8-methoxyquinolin-2-yl)-1-methylpiperazine-2-carboxylic acid
2-(6-methoxynaphthalen-2-yl)-4-[5-(propan-2-yl)-1,3-oxazole-4-carbonyl]morpholine
2-[3,5-dimethyl-4-(pyridin-3-yl)-1H-pyrazol-1-yl]-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine
2-[(5-methylpyrazin-2-yl)methyl]-8-(pyridazin-3-yl)-2,8-diazaspiro[5.5]undecan-3-one
2-[(cyclopropylmethyl)sulfanyl]-1-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
2-{1-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]pyrrolidin-2-yl}-5-fluoro-1H-1,3-benzodiazole
4-{[2-(3,4-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}piperazin-2-one
3-({2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-5-yl}methyl)-7-methyl-1,2-dihydroquinolin-2-one
N-cycloheptyl-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-methyl-N-(pyridin-4-ylmethyl)-5-({[3-(trifluoromethyl)phenyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(1-{5-methyl-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperidin-4-yl)-1,2,3,4-tetrahydroisoquinoline
3-(4-hydroxyphenyl)-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}benzamide
2-{4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
N-{[1-(1H-indol-5-ylmethyl)piperidin-3-yl]methyl}-2-(methylsulfanyl)acetamide
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-cyclopropyl-5-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
4-[(1-ethyl-1H-imidazol-2-yl)methyl]-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(4-{3,9-diazaspiro[5.6]dodecan-9-ylmethyl}phenyl)but-3-yn-1-ol
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-(1-methoxypropan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2-methoxyethyl)-3,5-dimethyl-N-(pyridin-4-ylmethyl)-1H-indole-2-carboxamide
1-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-2-methoxy-2-methylpropan-1-one